(Q37296998)

English

Synthesis and evaluation of hetero- and homodimers of ribosome-targeting antibiotics: antimicrobial activity, in vitro inhibition of translation, and drug resistance

scientific article published on July 2013

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scholarly article

1 reference

Europe PubMed Central

PMC publication ID

19 August 2017

Synthesis and evaluation of hetero- and homodimers of ribosome-targeting antibiotics: antimicrobial activity, in vitro inhibition of translation, and drug resistance (English)

1 reference

Europe PubMed Central

PMC publication ID

19 August 2017

antimicrobial resistance

1 reference

based on heuristic

inferred from title

antibiotic resistance

1 reference

based on heuristic

inferred from title

object named as

Micha Fridman

6

0 references

Sylvie Garneau-Tsodikova

object named as

Sylvie Garneau-Tsodikova

5

0 references

author name string

Yifat Berkov-Zrihen

1

1 reference

Europe PubMed Central

PMC publication ID

19 August 2017

Keith D Green

2

1 reference

Europe PubMed Central

PMC publication ID

19 August 2017

Kristin J Labby

3

1 reference

Europe PubMed Central

PMC publication ID

19 August 2017

Mark Feldman

4

1 reference

Europe PubMed Central

PMC publication ID

19 August 2017

language of work or name

0 references

publication date

1 July 2013

1 reference

Europe PubMed Central

PMC publication ID

19 August 2017

Journal of Medicinal Chemistry

1 reference

Europe PubMed Central

PMC publication ID

19 August 2017

56

1 reference

Europe PubMed Central

PMC publication ID

19 August 2017

13

1 reference

Europe PubMed Central

PMC publication ID

19 August 2017

5613-5625

1 reference

Europe PubMed Central

PMC publication ID

19 August 2017

Dual-acting hybrid antibiotics: a promising strategy to combat bacterial resistance

1 reference

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6 September 2017

Click dimers to target HIV TAR RNA conformation

1 reference

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6 September 2017

The structural basis for substrate versatility of chloramphenicol acetyltransferase CATI

1 reference

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6 September 2017

Antibiotics in development targeting protein synthesis

1 reference

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6 September 2017

Recognition of HIV TAR RNA by triazole linked neomycin dimers

1 reference

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6 September 2017

Unusual regioversatility of acetyltransferase Eis, a cause of drug resistance in XDR-TB

1 reference

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6 September 2017

Q&A: Antibiotic resistance: where does it come from and what can we do about it?

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3823688

6 September 2017

Structures of the Escherichia coli ribosome with antibiotics bound near the peptidyl transferase center explain spectra of drug action

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3823688

6 September 2017

The future of aminoglycosides: the end or renaissance?

1 reference

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Controlling the specificity of modularly assembled small molecules for RNA via ligand module spacing: targeting the RNAs that cause myotonic muscular dystrophy

1 reference

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6 September 2017

The use of ribosomal crystal structures in antibiotic drug design.

1 reference

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6 September 2017

Outer membrane permeability and antibiotic resistance

1 reference

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6 September 2017

Design at the atomic level: generation of novel hybrid biaryloxazolidinones as promising new antibiotics

1 reference

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6 September 2017

Expanding the nucleotide repertoire of the ribosome with post-transcriptional modifications

1 reference

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6 September 2017

The Cfr rRNA methyltransferase confers resistance to Phenicols, Lincosamides, Oxazolidinones, Pleuromutilins, and Streptogramin A antibiotics

1 reference

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6 September 2017

Antibiotics and the ribosome.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3823688

6 September 2017

Antibiotics targeting ribosomes: resistance, selectivity, synergism and cellular regulation

1 reference

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6 September 2017

Bacterial resistance to antibiotics: enzymatic degradation and modification

1 reference

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6 September 2017

Molecular basis of bacterial resistance to chloramphenicol and florfenicol

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3823688

6 September 2017

Ribosomal antibiotics: structural basis for resistance, synergism and selectivity

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3823688

6 September 2017

Efflux-mediated drug resistance in bacteria

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3823688

6 September 2017

Structures of five antibiotics bound at the peptidyl transferase center of the large ribosomal subunit

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3823688

6 September 2017

The importance of efflux pumps in bacterial antibiotic resistance

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3823688

6 September 2017

Crystal structure of a complex between the aminoglycoside tobramycin and an oligonucleotide containing the ribosomal decoding a site

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3823688

6 September 2017

Structural basis for the interaction of antibiotics with the peptidyl transferase centre in eubacteria

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3823688

6 September 2017

Crystal structures of complexes of the small ribosomal subunit with tetracycline, edeine and IF3.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3823688

6 September 2017

The structural basis for the action of the antibiotics tetracycline, pactamycin, and hygromycin B on the 30S ribosomal subunit

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3823688

6 September 2017

Functional insights from the structure of the 30S ribosomal subunit and its interactions with antibiotics

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3823688

6 September 2017

Clindamycin in the treatment of streptococcal and staphylococcal toxic shock syndromes

1 reference

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A new resistance gene, linB, conferring resistance to lincosamides by nucleotidylation in Enterococcus faecium HM1025.

1 reference

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6 September 2017

Chloramphenicol toxicity: 25 years of research.

1 reference

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6 September 2017

In vitro activity of chloramphenicol and thiamphenicol analogs

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3823688

14 September 2017

Effects of altering aminoglycoside structures on bacterial resistance enzyme activities

1 reference

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26 June 2018

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1 reference

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26 June 2018

Enhanced RNA binding of dimerized aminoglycosides

1 reference

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26 June 2018

6''-Thioether tobramycin analogues: towards selective targeting of bacterial membranes

1 reference

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2 September 2018

Assessment of 6'- and 6'''-N-acylation of aminoglycosides as a strategy to overcome bacterial resistance.

1 reference

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2 September 2018

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1 reference

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2 September 2018

An approach to enhance specificity against RNA targets using heteroconjugates of aminoglycosides and chloramphenicol (or linezolid).

1 reference

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2 September 2018

Structure–activity relationship in the oxazolidinone–quinolone hybrid series: influence of the central spacer on the antibacterial activity and the mode of action

1 reference

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2 September 2018

Aminoglycosides: a practical review

1 reference

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2 September 2018

Cubic crystals of chloramphenicol phosphotransferase fromStreptomyces venezuelaein complex with chloramphenicol

1 reference

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12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identifiers

10.1021/JM400707F

1 reference

Europe PubMed Central

PMC publication ID

19 August 2017

PMC publication ID

1 reference

Europe PubMed Central

PMC publication ID

19 August 2017

PubMed publication ID

1 reference

Europe PubMed Central

PMC publication ID

19 August 2017

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