(Q37399109)

English

Dipyridamole analogs as pharmacological inhibitors of equilibrative nucleoside transporters. Identification of novel potent and selective inhibitors of the adenosine transporter function of human equilibrative nucleoside transporter 4 (hENT4).

scientific article published on 07 September 2013

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Europe PubMed Central

PMC publication ID

20 August 2017

Dipyridamole analogs as pharmacological inhibitors of equilibrative nucleoside transporters. Identification of novel potent and selective inhibitors of the adenosine transporter function of human equilibrative nucleoside transporter 4 (hENT4). (English)

1 reference

Europe PubMed Central

PMC publication ID

20 August 2017

1 reference

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inferred from title

John K Buolamwini

6

object named as

John K Buolamwini

1 reference

Europe PubMed Central

PMC publication ID

20 August 2017

Hilaire C Playa

3

object named as

Hilaire Playa

1 reference

Europe PubMed Central

PMC publication ID

20 August 2017

author name string

Chunmei Wang

1

1 reference

Europe PubMed Central

PMC publication ID

20 August 2017

Wenwei Lin

2

1 reference

Europe PubMed Central

PMC publication ID

20 August 2017

Shan Sun

4

1 reference

Europe PubMed Central

PMC publication ID

20 August 2017

Keyuna Cameron

5

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Europe PubMed Central

PMC publication ID

20 August 2017

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publication date

7 September 2013

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Europe PubMed Central

PMC publication ID

20 August 2017

Biochemical Pharmacology

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Europe PubMed Central

PMC publication ID

20 August 2017

86

1 reference

Europe PubMed Central

PMC publication ID

20 August 2017

11

1 reference

Europe PubMed Central

PMC publication ID

20 August 2017

1531-1540

1 reference

Europe PubMed Central

PMC publication ID

20 August 2017

Emerging transporters of clinical importance: an update from the International Transporter Consortium

1 reference

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The human concentrative and equilibrative nucleoside transporter families, SLC28 and SLC29.

1 reference

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Human concentrative nucleoside transporter 3 transfection with ultrasound and microbubbles in nucleoside transport deficient HEK293 cells greatly increases gemcitabine uptake

1 reference

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6 September 2017

Adenosine transporter ENT4 is a direct target of EWS/WT1 translocation product and is highly expressed in desmoplastic small round cell tumor

1 reference

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6 September 2017

Dipyridamole, cerebrovascular disease, and the vasculature

1 reference

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6 September 2017

Synthesis, flow cytometric evaluation, and identification of highly potent dipyridamole analogues as equilibrative nucleoside transporter 1 inhibitors

1 reference

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6 September 2017

Dipyridamole, an underestimated vascular protective drug

1 reference

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6 September 2017

Cell entry and export of nucleoside analogues

1 reference

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Clinical effectiveness and cost-effectiveness of clopidogrel and modified-release dipyridamole in the secondary prevention of occlusive vascular events: a systematic review and economic evaluation

1 reference

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Identification and characterization of a novel monoamine transporter in the human brain

1 reference

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6 September 2017

Glycine 154 of the equilibrative nucleoside transporter, hENT1, is important for nucleoside transport and for conferring sensitivity to the inhibitors nitrobenzylthioinosine, dipyridamole, and dilazep

1 reference

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6 September 2017

Mammalian nucleoside transporters

1 reference

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6 September 2017

The equilibrative nucleoside transporter family, SLC29

1 reference

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6 September 2017

Functional and molecular characterization of nucleobase transport by recombinant human and rat equilibrative nucleoside transporters 1 and 2. Chimeric constructs reveal a role for the ENT2 helix 5-6 region in nucleobase translocation

1 reference

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6 September 2017

A single glycine mutation in the equilibrative nucleoside transporter gene, hENT1, alters nucleoside transport activity and sensitivity to nitrobenzylthioinosine

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3866046

6 September 2017

Adenosine, adenosine receptors and myocardial protection: an updated overview

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3866046

6 September 2017

The ENT family of eukaryote nucleoside and nucleobase transporters: recent advances in the investigation of structure/function relationships and the identification of novel isoforms

1 reference

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6 September 2017

Recent advances in the molecular biology of nucleoside transporters of mammalian cells

1 reference

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6 September 2017

Functional production and reconstitution of the human equilibrative nucleoside transporter (hENT1) in Saccharomyces cerevisiae. Interaction of inhibitors of nucleoside transport with recombinant hENT1 and a glycosylation-defective derivative (hENT1/

1 reference

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6 September 2017

Cloning of the human equilibrative, nitrobenzylmercaptopurine riboside (NBMPR)-insensitive nucleoside transporter ei by functional expression in a transport-deficient cell line

1 reference

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6 September 2017

Molecular cloning and functional characterization of nitrobenzylthioinosine (NBMPR)-sensitive (es) and NBMPR-insensitive (ei) equilibrative nucleoside transporter proteins (rENT1 and rENT2) from rat tissues

1 reference

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6 September 2017

Cloning of a human nucleoside transporter implicated in the cellular uptake of adenosine and chemotherapeutic drugs

1 reference

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6 September 2017

Symposium on immunosuppressive drugs. Biochemistry and pharmacology of purine analogues

1 reference

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14 September 2017

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Mutagenicity of cancer chemotherapeutic agents in the Salmonella/microsome test

1 reference

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14 September 2017

Kinetic and pharmacological properties of cloned human equilibrative nucleoside transporters, ENT1 and ENT2, stably expressed in nucleoside transporter-deficient PK15 cells. Ent2 exhibits a low affinity for guanosine and cytidine but a high affinity

1 reference

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Cellular localization and functional characterization of the equilibrative nucleoside transporters of antitumor nucleosides.

1 reference

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2 September 2018

Distribution and functional characterization of equilibrative nucleoside transporter-4, a novel cardiac adenosine transporter activated at acidic pH.

1 reference

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Functional characterization of novel human and mouse equilibrative nucleoside transporters (hENT3 and mENT3) located in intracellular membranes

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Dipyridamole increases the cytotoxicity of cisplatin in human larynx cancer cells in vitro.

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Nucleoside transport inhibitors, dipyridamole and p-nitrobenzylthioinosine, selectively potentiate the antitumor activity of NB1011.

1 reference

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Mutation of residue 33 of human equilibrative nucleoside transporters 1 and 2 alters sensitivity to inhibition of transport by dilazep and dipyridamole

1 reference

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Modulation of atrioventricular nodal function by metabolic and allosteric regulators of endogenous adenosine in guinea pig heart

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Pretreatment with lidoflazine, a calcium-channel blocker. Useful adjunct to heterogeneous cold potassium cardioplegia

1 reference

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The cardioprotective effects of R 75231 and lidoflazine are not caused by adenosine A1 receptor activation

1 reference

https://pubmed.ncbi.nlm.nih.gov/24021350

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Design, synthesis, and evaluation of 2-diethanolamino-4,8-diheptamethyleneimino-2-(N-aminoethyl-N-ethanolamino)-6-(N,N-diethanolamino)pyrimido[5,4-d]pyrimidine-fluorescein conjugate (8MDP-fluor), as a novel equilibrative nucleoside transporter probe

1 reference

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Involvement of multiple transporters in the oral absorption of nucleoside analogues

1 reference

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inferred from PubMed ID database lookup

Identifiers

10.1016/J.BCP.2013.08.063

1 reference

Europe PubMed Central

PMC publication ID

20 August 2017

PMC publication ID

1 reference

Europe PubMed Central

PMC publication ID

20 August 2017

PubMed publication ID

1 reference

Europe PubMed Central

PMC publication ID

20 August 2017

ResearchGate publication ID

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