(Q37502653)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24332089%20AND%20SRC:MED&resulttype=core&format=json

3 March 2020

title

Imidazole-derived agonists for the neurotensin 1 receptor (English)

1 reference

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3 March 2020

9

1 reference

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3 March 2020

Anthony B Pinkerton

13

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24332089%20AND%20SRC:MED&resulttype=core&format=json

3 March 2020

12

Marc G Caron

1 reference

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3 March 2020

author name string

Paul M Hershberger

1

1 reference

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3 March 2020

Michael P Hedrick

2

1 reference

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3 March 2020

Satyamaheshwar Peddibhotla

3

1 reference

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3 March 2020

Arianna Mangravita-Novo

4

1 reference

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3 March 2020

Palak Gosalia

5

1 reference

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3 March 2020

Yujie Li

6

1 reference

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3 March 2020

Wilson Gray

7

1 reference

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3 March 2020

Michael Vicchiarelli

8

1 reference

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3 March 2020

Thomas D Y Chung

10

1 reference

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3 March 2020

James B Thomas

11

1 reference

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3 March 2020

Lawrence S Barak

14

1 reference

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3 March 2020

Gregory P Roth

15

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3 March 2020

language of work or name

English

0 references

publication date

21 November 2013

1 reference

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3 March 2020

number of pages

6

1 reference

Bioorganic & Medicinal Chemistry Letters

inferred from page(s)

published in

1 reference

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3 March 2020

volume

24

1 reference

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3 March 2020

issue

1

1 reference

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3 March 2020

page(s)

262-267

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24332089%20AND%20SRC:MED&resulttype=core&format=json

Discovery of ML314, a Brain Penetrant Non-Peptidic β-Arrestin Biased Agonist of the Neurotensin NTR1 Receptor.

3 March 2020

cites work

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3898338

Response of limbic neurotensin systems to methamphetamine self-administration

23 August 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3898338

Cancer, chemistry, and the cell: molecules that interact with the neurotensin receptors

23 August 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3898338

The identification of nonpeptide neurotensin receptor partial agonists from the potent antagonist SR48692 using a calcium mobilization assay

23 August 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3898338

Biochemical and pharmacological profile of a potent and selective nonpeptide antagonist of the neurotensin receptor

23 August 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3898338

The Isolation of a New Hypotensive Peptide, Neurotensin, from Bovine Hypothalami

23 August 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3898338

Distribution of neurotensin receptors in mammalian brain. What it is telling us about its interactions with other neurotransmitter systems

23 August 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3898338

Distribution of neurotensin and its receptor in the central nervous system

23 August 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3898338

Biochemical and pharmacological activities of SR 142948A, a new potent neurotensin receptor antagonist

14 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3898338

Tissue distribution and cellular localization of the levocabastine-sensitive neurotensin receptor mRNA in adult rat brain

28 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3898338

New bicyclic antidepressant agent. Synthesis and activity of napactadine and related compounds

26 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3898338

The identification of neurotensin NTS1 receptor partial agonists through a ligand-based virtual screening approach

26 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3898338

Bioisosteric replacements of the pyrazole moiety of rimonabant: synthesis, biological properties, and molecular modeling investigations of thiazoles, triazoles, and imidazoles as potent and selective CB1 cannabinoid receptor antagonists

2 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3898338

Immunohistochemical distribution of NTS2 neurotensin receptors in the rat central nervous system

2 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3898338

Synthesis and pharmacological evaluation of 1-[(1,2-diphenyl-1H-4-imidazolyl)methyl]-4-phenylpiperazines with clozapine-like mixed activities at dopamine D(2), serotonin, and GABA(A) receptors.

2 September 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3898338

1,2-Diarylimidazoles as potent, cyclooxygenase-2 selective, and orally active antiinflammatory agents

2 September 2018

1 reference

12 December 2020

SR142948A is a potent antagonist of the cardiovascular effects of neurotensin

1 reference

12 December 2020

Discovery of imidazole carboxamides as potent and selective CCK1R agonists

1 reference

12 December 2020

Optimization of imidazole amide derivatives as cannabinoid-1 receptor antagonists for the treatment of obesity

1 reference

12 December 2020

10.1016/J.BMCL.2013.11.026

Identifiers

DOI

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24332089%20AND%20SRC:MED&resulttype=core&format=json

3 March 2020

1 reference

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3 March 2020

1 reference