(Q38281897)

1 September 2017

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title

KDM4 histone demethylase inhibitors for anti-cancer agents: a patent review (English)

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1 September 2017

Young-Won Chin

1

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1 September 2017

Sun-Young Han

series ordinal

2

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1 September 2017

language of work or name

English

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publication date

3 December 2014

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Expert Opinion on Therapeutic Patents

1 September 2017

published in

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1 September 2017

volume

25

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1 September 2017

issue

2

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1 September 2017

page(s)

135-144

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An operational definition of epigenetics

1 September 2017

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The transcriptional repressor JHDM3A demethylates trimethyl histone H3 lysine 9 and lysine 36.

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The testis-enriched histone demethylase, KDM4D, regulates methylation of histone H3 lysine 9 during spermatogenesis in the mouse but is dispensable for fertility

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Cooperative epigenetic modulation by cancer amplicon genes

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Targeting the JMJD2 histone demethylases to epigenetically control herpesvirus infection and reactivation from latency

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A selective inhibitor and probe of the cellular functions of Jumonji C domain-containing histone demethylases

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Pan-histone demethylase inhibitors simultaneously targeting Jumonji C and lysine-specific demethylases display high anticancer activities.

21 January 2018

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KDM4B as a target for prostate cancer: structural analysis and selective inhibition by a novel inhibitor

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Development of homogeneous luminescence assays for histone demethylase catalysis and binding.

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21 January 2018

Identifiers

DOI

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1 September 2017

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