(Q38647071)

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Cyclopentane-1,3-dione: a novel isostere for the carboxylic acid functional group. Application to the design of potent thromboxane (A2) receptor antagonists

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scholarly article

1 reference

Europe PubMed Central

5 September 2017

Cyclopentane-1,3-dione: a novel isostere for the carboxylic acid functional group. Application to the design of potent thromboxane (A2) receptor antagonists (English)

1 reference

Europe PubMed Central

5 September 2017

John Q. Trojanowski

8

object named as

John Q Trojanowski

1 reference

Europe PubMed Central

5 September 2017

Carlo Ballatore

object named as

Carlo Ballatore

1

0 references

object named as

Donna M Huryn

7

0 references

author name string

James H Soper

2

1 reference

Europe PubMed Central

5 September 2017

Francesco Piscitelli

3

1 reference

Europe PubMed Central

5 September 2017

Michael James

4

1 reference

Europe PubMed Central

5 September 2017

Longchuan Huang

5

1 reference

Europe PubMed Central

5 September 2017

Onur Atasoylu

6

1 reference

Europe PubMed Central

5 September 2017

Virginia M-Y Lee

9

1 reference

Europe PubMed Central

5 September 2017

Kurt R Brunden

10

1 reference

Europe PubMed Central

5 September 2017

Amos B Smith

11

1 reference

Europe PubMed Central

5 September 2017

language of work or name

0 references

publication date

9 September 2011

1 reference

Europe PubMed Central

5 September 2017

Journal of Medicinal Chemistry

1 reference

Europe PubMed Central

5 September 2017

54

1 reference

Europe PubMed Central

5 September 2017

6969-6983

1 reference

Europe PubMed Central

5 September 2017

19

1 reference

Europe PubMed Central

5 September 2017

Synopsis of some recent tactical application of bioisosteres in drug design

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3188681

6 September 2017

From the design to the clinical application of thromboxane modulators

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3188681

6 September 2017

5-Substituted-1H-tetrazoles as carboxylic acid isosteres: medicinal chemistry and synthetic methods

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3188681

6 September 2017

Bioisosterism: A Rational Approach in Drug Design

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3188681

6 September 2017

Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3188681

6 September 2017

The G protein coupled to the thromboxane A2 receptor in human platelets is a member of the novel Gq family

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3188681

6 September 2017

Cloning and expression of cDNA for a human thromboxane A2 receptor

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3188681

6 September 2017

Carboxylic acids and tetrazoles as isosteric replacements for sulfate in cholecystokinin analogues.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3188681

23 June 2018

Radioligand binding methods for membrane preparations and intact cells.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3188681

31 August 2018

Direct amino acid-catalyzed cascade biomimetic reductive alkylations: application to the asymmetric synthesis of Hajos-Parrish ketone analogues

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3188681

31 August 2018

Thromboxane receptor activation mediates isoprostane-induced increases in amyloid pathology in Tg2576 mice

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3188681

31 August 2018

Unusually weak binding interactions in tetrazole-amidine complexes.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3188681

31 August 2018

NMR structure of the thromboxane A2 receptor ligand recognition pocket

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3188681

31 August 2018

Noncovalent interactions between tetrazole and an N,N'-diethyl-substituted benzamidine

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3188681

31 August 2018

Thromboxane modulating agents. 3. 1H-imidazol-1-ylalkyl- and 3-pyridinylalkyl-substituted 3-[2-[(arylsulfonyl)amino]ethyl]benzenepropanoic acid derivatives as dual thromboxane synthase inhibitor/thromboxane receptor antagonists

1 reference

https://pubmed.ncbi.nlm.nih.gov/21863799

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Modeling of human thromboxane A2 receptor and analysis of the receptor-ligand interaction

1 reference

https://pubmed.ncbi.nlm.nih.gov/21863799

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Structures of Cyclopentanepolyones

1 reference

https://pubmed.ncbi.nlm.nih.gov/21863799

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identifiers

10.1021/JM200980U

1 reference

Europe PubMed Central

5 September 2017

1 reference

Europe PubMed Central

5 September 2017

1 reference

Europe PubMed Central

5 September 2017

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