(Q39157688)

9 September 2017

Discovery of the First Potent and Selective Inhibitor of Centromere-Associated Protein E: GSK923295. (English)

1 reference

9 September 2017

6

1 reference

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7 June 2020

Rosanna Tedesco

8

1 reference

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7 June 2020

author name string

Xiangping Qian

1

1 reference

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7 June 2020

Andrew McDonald

2

1 reference

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7 June 2020

Han-Jie Zhou

3

1 reference

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7 June 2020

Nicholas D Adams

4

1 reference

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7 June 2020

Cynthia A Parrish

5

1 reference

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7 June 2020

Duke M Fitch

7

1 reference

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7 June 2020

Luke W Ashcraft

9

1 reference

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7 June 2020

Bing Yao

10

1 reference

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7 June 2020

Hong Jiang

11

1 reference

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7 June 2020

Jennifer K Huang

12

1 reference

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7 June 2020

Melchor V Marin

13

1 reference

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7 June 2020

Carrie E Aroyan

14

1 reference

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7 June 2020

Jianchao Wang

15

1 reference

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7 June 2020

Seyed Ahmed

16

1 reference

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7 June 2020

Joelle L Burgess

17

1 reference

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7 June 2020

Amita M Chaudhari

18

1 reference

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7 June 2020

Carla A Donatelli

19

1 reference

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7 June 2020

Michael G Darcy

20

1 reference

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7 June 2020

Lance H Ridgers

21

1 reference

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7 June 2020

Ken A Newlander

22

1 reference

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7 June 2020

Stanley J Schmidt

23

1 reference

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7 June 2020

Deping Chai

24

1 reference

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7 June 2020

Mariela Colón

25

1 reference

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7 June 2020

Michael N Zimmerman

26

1 reference

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7 June 2020

Latesh Lad

27

1 reference

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7 June 2020

Roman Sakowicz

28

1 reference

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7 June 2020

Stephen Schauer

29

1 reference

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7 June 2020

Lisa Belmont

30

1 reference

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7 June 2020

Ramesh Baliga

31

1 reference

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7 June 2020

Daniel W Pierce

32

1 reference

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7 June 2020

Jeffrey T Finer

33

1 reference

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7 June 2020

Zhengping Wang

34

1 reference

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7 June 2020

Bradley P Morgan

35

1 reference

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7 June 2020

David J Morgans

36

1 reference

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7 June 2020

Kurt R Auger

37

1 reference

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7 June 2020

Chiu-Mei Sung

38

1 reference

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7 June 2020

Jeff D Carson

39

1 reference

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7 June 2020

Lusong Luo

40

1 reference

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7 June 2020

Erin D Hugger

41

1 reference

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7 June 2020

Robert A Copeland

42

1 reference

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7 June 2020

David Sutton

43

1 reference

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7 June 2020

John D Elliott

44

1 reference

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7 June 2020

Jeffrey R Jackson

45

1 reference

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7 June 2020

Kenneth W Wood

46

1 reference

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7 June 2020

Dashyant Dhanak

47

1 reference

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7 June 2020

Gustave Bergnes

48

1 reference

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7 June 2020

Steven D Knight

49

1 reference

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7 June 2020

language of work or name

1 reference

19 January 2010

1 reference

ACS Medicinal Chemistry Letters

9 September 2017

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24900171%20AND%20SRC:MED&resulttype=core&format=json

7 June 2020

volume

1

1 reference

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7 June 2020

issue

1

1 reference

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7 June 2020

page(s)

30-34

1 reference

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Centromere-associated protein E: a motor that puts the brakes on the mitotic checkpoint

7 June 2020

cites work

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4007900

10 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4007900

Recent developments in fragment-based drug discovery

10 September 2017

1 reference

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Targeted anti-mitotic therapies: can we improve on tubulin agents?

10 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4007900

Inhibitors of mitotic kinesins: next-generation antimitotics

10 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4007900

Microtubule capture by CENP-E silences BubR1-dependent mitotic checkpoint signaling

10 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4007900

Mitotic kinesins: prospects for antimitotic drug discovery.

10 September 2017

1 reference

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Functional analysis of human microtubule-based motor proteins, the kinesins and dyneins, in mitosis/cytokinesis using RNA interference

10 September 2017

1 reference

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Gene silencing of CENP-E by small interfering RNA in HeLa cells leads to missegregation of chromosomes after a mitotic delay

10 September 2017

1 reference

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Centromere-associated protein-E is essential for the mammalian mitotic checkpoint to prevent aneuploidy due to single chromosome loss

10 September 2017

1 reference

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The molecular motor toolbox for intracellular transport

10 September 2017

1 reference

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Centromeres and kinetochores: from epigenetics to mitotic checkpoint signaling

10 September 2017

1 reference

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Past and future of the mitotic spindle as an oncology target

10 September 2017

1 reference

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CENP-E is essential for reliable bioriented spindle attachment, but chromosome alignment can be achieved via redundant mechanisms in mammalian cells

10 September 2017

1 reference

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All kinesin superfamily protein, KIF, genes in mouse and human

10 September 2017

1 reference

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Microtubule motors in mitosis

10 September 2017

1 reference

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CENP-E forms a link between attachment of spindle microtubules to kinetochores and the mitotic checkpoint

10 September 2017

1 reference

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The road less traveled: emerging principles of kinesin motor utilization

10 September 2017

1 reference

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CENP-E function at kinetochores is essential for chromosome alignment.

10 September 2017

1 reference

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CENP-E is a plus end-directed kinetochore motor required for metaphase chromosome alignment

10 September 2017

1 reference

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Novel ATP-competitive kinesin spindle protein inhibitors

10 September 2017

1 reference

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A manual method for applying the Hansch approach to drug design

14 September 2017

1 reference

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Ligand efficiency indices as guideposts for drug discovery.

25 September 2017

1 reference

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Ligand binding efficiency: trends, physical basis, and implications

21 August 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/24900171

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1021/ML900018M

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24900171%20AND%20SRC:MED&resulttype=core&format=json

7 June 2020

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24900171%20AND%20SRC:MED&resulttype=core&format=json

7 June 2020

PubMed publication ID

24900171

1 reference