(Q39527868)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:21657832%20AND%20SRC:MED&resulttype=core&format=json

3 February 2020

title

Calcein assay: a high-throughput method to assess P-gp inhibition (English)

1 reference

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3 February 2020

3

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3 February 2020

author name string

H Glavinas

1

1 reference

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3 February 2020

O von Richter

2

1 reference

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3 February 2020

D Mehn

4

1 reference

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3 February 2020

I Wilhelm

5

1 reference

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3 February 2020

T Nagy

6

1 reference

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3 February 2020

J Janossy

7

1 reference

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3 February 2020

I Krizbai

8

1 reference

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3 February 2020

P Couraud

9

1 reference

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3 February 2020

P Krajcsi

10

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3 February 2020

language of work or name

English

0 references

publication date

9 June 2011

1 reference

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3 February 2020

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:21657832%20AND%20SRC:MED&resulttype=core&format=json

3 February 2020

volume

41

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:21657832%20AND%20SRC:MED&resulttype=core&format=json

3 February 2020

issue

8

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3 February 2020

page(s)

712-719

1 reference

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Characterization of beta-adrenoceptor antagonists as substrates and inhibitors of the drug transporter P-glycoprotein

3 February 2020

cites work

1 reference

https://api.crossref.org/works/10.3109%2F00498254.2011.587033

Cholesterol-mediated activation of P-glycoprotein: distinct effects on basal and drug-induced ATPase activities

21 January 2018

1 reference

https://api.crossref.org/works/10.3109%2F00498254.2011.587033

P-glycoprotein and surfactants: effect on intestinal talinolol absorption

21 January 2018

1 reference

https://api.crossref.org/works/10.3109%2F00498254.2011.587033

Characterisation of human tubular cell monolayers as a model of proximal tubular xenobiotic handling

21 January 2018

1 reference

https://api.crossref.org/works/10.3109%2F00498254.2011.587033

Rapid assessment of p-glycoprotein-drug interactions at the blood-brain barrier

21 January 2018

1 reference

https://api.crossref.org/works/10.3109%2F00498254.2011.587033

Refining the in vitro and in vivo critical parameters for P-glycoprotein, [I]/IC50 and [I2]/IC50, that allow for the exclusion of drug candidates from clinical digoxin interaction studies

21 January 2018

1 reference

https://api.crossref.org/works/10.3109%2F00498254.2011.587033

Considerations in the design and development of transport inhibitors as adjuncts to drug therapy

21 January 2018

1 reference

https://api.crossref.org/works/10.3109%2F00498254.2011.587033

N-glycosylation of ABC transporters is associated with functional activity in sandwich-cultured rat hepatocytes.

21 January 2018

1 reference

https://api.crossref.org/works/10.3109%2F00498254.2011.587033

Inhibition of the CYP3A4-mediated metabolism and P-glycoprotein-mediated transport of the HIV-1 protease inhibitor saquinavir by grapefruit juice components

21 January 2018

1 reference

https://api.crossref.org/works/10.3109%2F00498254.2011.587033

Quantification and characterization of P-glycoprotein-substrate interactions

21 January 2018

1 reference

https://api.crossref.org/works/10.3109%2F00498254.2011.587033

Membrane transporters in drug development

21 January 2018

1 reference

https://api.crossref.org/works/10.3109%2F00498254.2011.587033

Functional characterization of glycosylation-deficient human P-glycoprotein using a vaccinia virus expression system

21 January 2018

1 reference

https://api.crossref.org/works/10.3109%2F00498254.2011.587033

Delineating the contribution of secretory transporters in the efflux of etoposide using Madin-Darby canine kidney (MDCK) cells overexpressing P-glycoprotein (Pgp), multidrug resistance-associated protein (MRP1), and canalicular multispecific organic

21 January 2018

1 reference

https://api.crossref.org/works/10.3109%2F00498254.2011.587033

Interaction of imatinib mesilate with human P-glycoprotein

21 January 2018

1 reference

https://api.crossref.org/works/10.3109%2F00498254.2011.587033

Calcein accumulation as a fluorometric functional assay of the multidrug transporter

21 January 2018

1 reference

https://api.crossref.org/works/10.3109%2F00498254.2011.587033

New era in drug interaction evaluation: US Food and Drug Administration update on CYP enzymes, transporters, and the guidance process

21 January 2018

1 reference

https://api.crossref.org/works/10.3109%2F00498254.2011.587033

Drug absorption limited by P-glycoprotein-mediated secretory drug transport in human intestinal epithelial Caco-2 cell layers

21 January 2018

1 reference

https://api.crossref.org/works/10.3109%2F00498254.2011.587033

Absorption properties and P-glycoprotein activity of modified Caco-2 cell lines

21 January 2018

1 reference

https://api.crossref.org/works/10.3109%2F00498254.2011.587033

Decrease in intracellular concentration causes the shift in Km value of efflux pump substrates.

21 January 2018

1 reference

https://api.crossref.org/works/10.3109%2F00498254.2011.587033

P-glycoprotein related drug interactions: clinical importance and a consideration of disease states

21 January 2018

1 reference

https://api.crossref.org/works/10.3109%2F00498254.2011.587033

Pumping of Drugs by P-Glycoprotein: A Two-Step Process?

21 January 2018

1 reference

https://api.crossref.org/works/10.3109%2F00498254.2011.587033

Evidence for a non-MDR1 component in digoxin secretion by human intestinal Caco-2 epithelial layers

21 January 2018

1 reference

https://api.crossref.org/works/10.3109%2F00498254.2011.587033

Evaluation of in vivo P-glycoprotein phenotyping probes: a need for validation

21 January 2018

1 reference

https://api.crossref.org/works/10.3109%2F00498254.2011.587033

Uptake and permeability studies of BBB-targeting immunoliposomes using the hCMEC/D3 cell line

21 January 2018

1 reference

https://api.crossref.org/works/10.3109%2F00498254.2011.587033

Interaction of tomato lectin with ABC transporter in cancer cells: glycosylation confers functional conformation of P-gp.

21 January 2018

1 reference

https://api.crossref.org/works/10.3109%2F00498254.2011.587033

Modulation of P-glycoprotein activity by cannabinoid molecules in HK-2 renal cells

21 January 2018

1 reference

https://api.crossref.org/works/10.3109%2F00498254.2011.587033

Cholesterol potentiates ABCG2 activity in a heterologous expression system: improved in vitro model to study function of human ABCG2.

21 January 2018

1 reference

https://api.crossref.org/works/10.3109%2F00498254.2011.587033

Role of P-glycoprotein on the CNS disposition of amprenavir (141W94), an HIV protease inhibitor

21 January 2018

1 reference

https://api.crossref.org/works/10.3109%2F00498254.2011.587033

ATP-binding cassette B1 transports seliciclib (R-roscovitine), a cyclin-dependent kinase inhibitor

21 January 2018

1 reference

https://api.crossref.org/works/10.3109%2F00498254.2011.587033

In vitro p-glycoprotein inhibition assays for assessment of clinical drug interaction potential of new drug candidates: a recommendation for probe substrates.

21 January 2018

1 reference

https://api.crossref.org/works/10.3109%2F00498254.2011.587033

Comparison of in vitro P-glycoprotein screening assays: recommendations for their use in drug discovery

21 January 2018

1 reference

https://api.crossref.org/works/10.3109%2F00498254.2011.587033

The role of size and charge for blood-brain barrier permeation of drugs and fatty acids

21 January 2018

1 reference

https://api.crossref.org/works/10.3109%2F00498254.2011.587033

Positively cooperative sites for drug transport by P-glycoprotein with distinct drug specificities

21 January 2018

1 reference

https://api.crossref.org/works/10.3109%2F00498254.2011.587033

Are MDCK cells transfected with the human MDR1 gene a good model of the human intestinal mucosa?

21 January 2018

1 reference

https://api.crossref.org/works/10.3109%2F00498254.2011.587033

The elementary mass action rate constants of P-gp transport for a confluent monolayer of MDCKII-hMDR1 cells.

21 January 2018

1 reference

https://api.crossref.org/works/10.3109%2F00498254.2011.587033

A novel screening strategy to identify ABCB1 substrates and inhibitors

21 January 2018

1 reference

https://api.crossref.org/works/10.3109%2F00498254.2011.587033

Grapefruit Juice–Drug Interactions: Grapefruit Juice and Its Components Inhibit P‐Glycoprotein (ABCB1) Mediated Transport of Talinolol in Caco‐2 Cells

21 January 2018

1 reference

https://api.crossref.org/works/10.3109%2F00498254.2011.587033

Blood-brain barrier-specific properties of a human adult brain endothelial cell line

21 January 2018

1 reference

24 May 2022

https://opencitations.net/index/coci/api/v1/citations/10.1096/FJ.04-3458FJE

Identifiers

DOI

10.3109/00498254.2011.587033

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:21657832%20AND%20SRC:MED&resulttype=core&format=json

3 February 2020

1 reference