(Q40629341)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24967388%20AND%20SRC:MED&resulttype=core&format=json

21 March 2020

title

Application of molecular modeling to urokinase inhibitors development (English)

1 reference

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21 March 2020

5

1 reference

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21 March 2020

Irina Beloglazova

7

1 reference

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21 March 2020

Vsevolod Tkachuk

9

1 reference

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21 March 2020

author name string

V B Sulimov

1

1 reference

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21 March 2020

E V Katkova

2

1 reference

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21 March 2020

I V Oferkin

3

1 reference

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21 March 2020

A V Sulimov

4

1 reference

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21 March 2020

A I Roschin

6

1 reference

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21 March 2020

O S Plekhanova

8

1 reference

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21 March 2020

V A Sadovnichiy

10

1 reference

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21 March 2020

language of work or name

English

0 references

publication date

20 May 2014

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24967388%20AND%20SRC:MED&resulttype=core&format=json

BioMed Research International

21 March 2020

published in

1 reference

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21 March 2020

volume

2014

1 reference

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21 March 2020

page(s)

625176

1 reference

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Creative Commons Attribution 3.0 Unported

21 March 2020

copyright license

start time

1 January 2014

1 reference

April 2022 Public Data File from Crossref

copyright status

copyrighted

1 reference

April 2022 Public Data File from Crossref

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The urokinase plasminogen activator system: a target for anti-cancer therapy.

22 September 2017

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Fragment-based discovery of mexiletine derivatives as orally bioavailable inhibitors of urokinase-type plasminogen activator

22 September 2017

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Intraperitoneal injection of a hairpin RNA-expressing plasmid targeting urokinase-type plasminogen activator (uPA) receptor and uPA retards angiogenesis and inhibits intracranial tumor growth in nude mice.

22 September 2017

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Selective urokinase-type plasminogen activator inhibitors. 4. 1-(7-sulfonamidoisoquinolinyl)guanidines

22 September 2017

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Identification of a novel inhibitor of urokinase-type plasminogen activator

22 September 2017

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Uncharged isocoumarin-based inhibitors of urokinase-type plasminogen activator

22 September 2017

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Inhibition of the invasion capacity of carcinoma cells by WX-UK1, a novel synthetic inhibitor of the urokinase-type plasminogen activator system

22 September 2017

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The urokinase plasminogen activator system: role in malignancy

22 September 2017

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CD87 (urokinase-type plasminogen activator receptor), function and pathology in hematological disorders: a review

22 September 2017

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Urokinase plasminogen activator system: a multifunctional role in tumor progression and metastasis.

22 September 2017

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uPAR: a versatile signalling orchestrator

22 September 2017

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Engineering inhibitors highly selective for the S1 sites of Ser190 trypsin-like serine protease drug targets

22 September 2017

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Role of the matrix metalloproteinase and plasminogen activator-plasmin systems in angiogenesis.

22 September 2017

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The plasminogen activator system: biology and regulation

22 September 2017

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Identification of novel inhibitors of urokinase via NMR-based screening

22 September 2017

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Discovering novel ligands for macromolecules using X-ray crystallographic screening

22 September 2017

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Urokinase plasminogen activator enhances neointima growth and reduces lumen size in injured carotid arteries

22 September 2017

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(4-aminomethyl)phenylguanidine derivatives as nonpeptidic highly selective inhibitors of human urokinase

22 September 2017

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22 September 2017

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Folding and binding cascades: shifts in energy landscapes

22 September 2017

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The crystal structure of the catalytic domain of human urokinase-type plasminogen activator

22 September 2017

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22 September 2017

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22 September 2017

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Functional inhibition of endogenously produced urokinase decreases cell proliferation in a human melanoma cell line

22 September 2017

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Methods for Determination of Prekallikrein in Plasma, Glandular Kallikrein and Urokinase

22 September 2017

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22 September 2017

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Amiloride selectively inhibits the urokinase-type plasminogen activator

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Synthetic inhibitors of serine proteinases. 17. The effect of benzamidine derivatives on the activity of urokinase and the reduction of fibrinolysis

15 June 2018

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15 June 2018

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Naphthamidine urokinase plasminogen activator inhibitors with improved pharmacokinetic properties

20 August 2018

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20 August 2018

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Finding more needles in the haystack: A simple and efficient method for improving high-throughput docking results.

20 August 2018

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4-Aminoarylguanidine and 4-aminobenzamidine derivatives as potent and selective urokinase-type plasminogen activator inhibitors

20 August 2018

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Selective urokinase-type plasminogen activator (uPA) inhibitors. Part 1: 2-Pyridinylguanidines

20 August 2018

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Structure-based design, synthesis and SAR of a novel series of thiopheneamidine urokinase plasminogen activator inhibitors.

20 August 2018

1 reference

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20 August 2018

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A Transferable H-Bonding Correction for Semiempirical Quantum-Chemical Methods

21 January 2018

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Antibodies to plasminogen activator inhibit human tumor metastasis

21 January 2018

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12 December 2020

Inhibition of urokinase by 4-substituted benzo[b]thiophene-2-carboxamidines: an important new class of selective synthetic urokinase inhibitor

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12 December 2020

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12 December 2020

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Identifiers

DOI

10.1155/2014/625176

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24967388%20AND%20SRC:MED&resulttype=core&format=json

21 March 2020

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24967388%20AND%20SRC:MED&resulttype=core&format=json

21 March 2020

PubMed publication ID

24967388

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24967388%20AND%20SRC:MED&resulttype=core&format=json