(Q40765666)

23 September 2017

title

Constitutive internalization of constitutively active agiotensin II AT(1A) receptor mutants is blocked by inverse agonists (English)

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23 September 2017

author

Stéphanie Miserey-Lenkei

series ordinal

1

object named as

Stéphanie Miserey-Lenkei

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23 September 2017

4

Pierre Corvol

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23 September 2017

Charles Parnot

2

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23 September 2017

Sabine Bardin

series ordinal

3

1 reference

23 September 2017

Eric Clauser

series ordinal

5

1 reference

23 September 2017

language of work or name

English

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publication date

29 November 2001

1 reference

Journal of Biological Chemistry

23 September 2017

published in

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23 September 2017

volume

277

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23 September 2017

issue

8

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23 September 2017

page(s)

5891-5901

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The Sequence of the Human Genome

23 September 2017

cites work

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Role of carboxyl tail of the rat angiotensin II type 1A receptor in agonist-induced internalization of the receptor

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Short-term desensitization of the angiotensin II receptor of bovine adrenal glomerulosa cells corresponds to a shift from a high to a low affinity state

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Mutation of Asn111 in the third transmembrane domain of the AT1A angiotensin II receptor induces its constitutive activation.

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The conformational change responsible for AT1 receptor activation is dependent upon two juxtaposed asparagine residues on transmembrane helices III and VII.

21 January 2018

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21 January 2018

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Cellular distribution of constitutively active mutant parathyroid hormone (PTH)/PTH-related protein receptors and regulation of cyclic adenosine 3',5'-monophosphate signaling by beta-arrestin2.

21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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Constitutive arrestin-mediated desensitization of a human vasopressin receptor mutant associated with nephrogenic diabetes insipidus

21 January 2018

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Agonist-induced phosphorylation of the angiotensin II (AT(1A)) receptor requires generation of a conformation that is distinct from the inositol phosphate-signaling state

21 January 2018

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Removal of phosphorylation sites from the β2-adrenergic receptor delays onset of agonist-promoted desensitization

21 January 2018

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Inverse agonism and the regulation of receptor number

21 January 2018

1 reference

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Stable expression of a truncated AT1A receptor in CHO-K1 cells. The carboxyl-terminal region directs agonist-induced internalization but not receptor signaling or desensitization.

21 January 2018

1 reference

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Mutation of Asp74 of the rat angiotensin II receptor confers changes in antagonist affinities and abolishes G-protein coupling.

21 January 2018

1 reference

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21 January 2018

Identifiers

DOI

10.1074/JBC.M108398200

1 reference

23 September 2017

1 reference