(Q41985097)

14 October 2017

Discovery of 'molecular switches' within a GIRK activator scaffold that afford selective GIRK inhibitors (English)

1 reference

14 October 2017

8

Craig W Lindsley

1 reference

14 October 2017

Wandong Wen

1

1 reference

14 October 2017

Wenjun Wu

2

1 reference

14 October 2017

Ian M Romaine

3

1 reference

14 October 2017

Kristian Kaufmann

4

1 reference

14 October 2017

Yu Du

5

1 reference

14 October 2017

Gary A Sulikowski

6

1 reference

14 October 2017

C David Weaver

7

1 reference

14 October 2017

language of work or name

English

0 references

publication date

20 June 2013

1 reference

Bioorganic & Medicinal Chemistry Letters

14 October 2017

1 reference

14 October 2017

23

1 reference

14 October 2017

16

1 reference

14 October 2017

4562-4566

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3816575

14 October 2017

1 reference

Naringin directly activates inwardly rectifying potassium channels at an overlapping binding site to tertiapin-Q.

5 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3816575

"Molecular switches" on mGluR allosteric ligands that modulate modes of pharmacology

5 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3816575

Emerging roles for G protein-gated inwardly rectifying potassium (GIRK) channels in health and disease.

5 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3816575

A discrete alcohol pocket involved in GIRK channel activation

5 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3816575

Synthesis and SAR of a mGluR5 allosteric partial antagonist lead: unexpected modulation of pharmacology with slight structural modifications to a 5-(phenylethynyl)pyrimidine scaffold

5 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3816575

Ethanol opens G-protein-activated inwardly rectifying K+ channels

5 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3816575

IRK(1-3) and GIRK(1-4) inwardly rectifying K+ channel mRNAs are differentially expressed in the adult rat brain

5 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3816575

Cloning provides evidence for a family of inward rectifier and G-protein coupled K+ channels in the brain

5 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3816575

The G-protein-gated atrial K+ channel IKACh is a heteromultimer of two inwardly rectifying K(+)-channel proteins

5 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3816575

Molecular cloning of a mouse G-protein-activated K+ channel (mGIRK1) and distinct distributions of three GIRK (GIRK1, 2 and 3) mRNAs in mouse brain

5 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3816575

ML297 (VU0456810), the first potent and selective activator of the GIRK potassium channel, displays antiepileptic properties in mice

5 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3816575

Primary structure and functional expression of a rat G-protein-coupled muscarinic potassium channel

18 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3816575

A comparison of the effects of the D1 receptor antagonists SCH 23390 and SCH 39166 on suppression of feeding behavior by the D1 agonist SKF38393.

18 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3816575

Enantiomer selectivity and the development of tolerance to the behavioral effects of the calcium channel activator BAY K 8644

18 August 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/23838260

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1016/J.BMCL.2013.06.023

1 reference

14 October 2017

1 reference

14 October 2017

PubMed publication ID

23838260

1 reference