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The selectivity of beta-adrenoceptor agonists at human beta1-, beta2- and beta3-adrenoceptors
scientific article published on July 2010
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scholarly article
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Europe PubMed Central
PMCID
2936015
retrieved
31 October 2017
title
The selectivity of beta-adrenoceptor agonists at human beta1-, beta2- and beta3-adrenoceptors
(English)
1 reference
stated in
Europe PubMed Central
PMCID
2936015
retrieved
31 October 2017
author
Jillian G Baker
object named as
Jillian G Baker
series ordinal
1
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language of work or name
English
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publication date
1 July 2010
1 reference
stated in
Europe PubMed Central
PMCID
2936015
retrieved
31 October 2017
published in
British Journal of Pharmacology
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stated in
Europe PubMed Central
PMCID
2936015
retrieved
31 October 2017
volume
160
1 reference
stated in
Europe PubMed Central
PMCID
2936015
retrieved
31 October 2017
issue
5
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stated in
Europe PubMed Central
PMCID
2936015
retrieved
31 October 2017
page(s)
1048-1061
1 reference
stated in
Europe PubMed Central
PMCID
2936015
retrieved
31 October 2017
cites work
The low-affinity site of the beta1-adrenoceptor and its relevance to cardiovascular pharmacology
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PubMed Central
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28 May 2018
Agonist binding, agonist affinity and agonist efficacy at G protein-coupled receptors
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28 May 2018
Evidence for a secondary state of the human beta3-adrenoceptor.
1 reference
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PubMed Central
reference URL
https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2936015
retrieved
28 May 2018
The selectivity of beta-adrenoceptor antagonists at the human beta1, beta2 and beta3 adrenoceptors
1 reference
stated in
PubMed Central
reference URL
https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2936015
retrieved
28 May 2018
Do low-affinity states of beta-adrenoceptors have roles in physiology and medicine?
1 reference
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PubMed Central
reference URL
https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2936015
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28 May 2018
Efficacy as a vector: the relative prevalence and paucity of inverse agonism
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28 May 2018
Agonist and inverse agonist actions of beta-blockers at the human beta 2-adrenoceptor provide evidence for agonist-directed signaling
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PubMed Central
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28 May 2018
Beta-arrestin-mediated activation of MAPK by inverse agonists reveals distinct active conformations for G protein-coupled receptors
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PubMed Central
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28 May 2018
The 'state' of beta-adrenoceptors
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PubMed Central
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28 May 2018
Agonist induction and conformational selection during activation of a G-protein-coupled receptor
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PubMed Central
reference URL
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28 May 2018
Drug efficacy at G protein-coupled receptors
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PubMed Central
reference URL
https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2936015
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28 May 2018
Pharmacological similarities and differences between beta2-agonists
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PubMed Central
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28 May 2018
The putative beta4-adrenergic receptor is a novel state of the beta1-adrenergic receptor
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28 May 2018
Binding properties of beta-blockers at recombinant beta1-, beta2-, and beta3-adrenoceptors
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28 May 2018
Efficacy in drug receptor theory: outdated concept or under-valued tool?
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28 May 2018
Beta-blocker selectivity at cloned human beta 1- and beta 2-adrenergic receptors
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28 May 2018
A three-state receptor model of agonist action
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28 May 2018
Anomalous behavior of CGP 12177A on beta 1-adrenergic receptors
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28 May 2018
Comparison of guinea-pig, bovine and rat alpha 1-adrenoceptor subtypes
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28 May 2018
The two-state model of receptor activation
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28 May 2018
Theoretical and practical problems with the assessment of intrinsic efficacy of agonists: efficacy of reputed beta-1 selective adrenoceptor agonists for beta-2 adrenoceptors
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28 May 2018
Is prenalterol (H133/80) really a selective beta 1 adrenoceptor agonist? Tissue selectivity resulting from differences in stimulus-response relationships
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28 May 2018
Stimulant and blocking effects of optical isomers of pindolol on the sinoatrial node and trachea of guinea pig. Role of ?-adrenoceptor subtypes in the dissociation between blockade and stimulation
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28 May 2018
Influence of rolipram on the cyclic 3',5'-adenosine monophosphate response to histamine and adenosine in slices of guinea-pig cerebral cortex
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Faster onset of action of formoterol versus salmeterol in patients with chronic obstructive pulmonary disease: a multicenter, randomized study
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16 August 2018
Guide to Receptors and Channels (GRAC), 3rd edition
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Site of action of beta-ligands at the human beta1-adrenoceptor
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16 August 2018
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16 August 2018
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16 August 2018
Intrinsic sympathomimetic activity of (-)-pindolol mediated through a (-)-propranolol-resistant site of the beta1-adrenoceptor in human atrium and recombinant receptors
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16 August 2018
Agonist actions of "beta-blockers" provide evidence for two agonist activation sites or conformations of the human beta1-adrenoceptor
1 reference
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PubMed Central
reference URL
https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2936015
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16 August 2018
Pharmacological characterization of CGP 12177 at the human beta(2)-adrenoceptor
1 reference
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PubMed Central
reference URL
https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2936015
retrieved
16 August 2018
The elusive nature of intrinsic efficacy
1 reference
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PubMed Central
reference URL
https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2936015
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16 August 2018
The measurement of efficacy in the drug discovery agonist selection process
1 reference
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PubMed
reference URL
https://pubmed.ncbi.nlm.nih.gov/20590599
retrieved
12 December 2020
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inferred from PubMed ID database lookup
Identifiers
DOI
10.1111/J.1476-5381.2010.00754.X
1 reference
stated in
Europe PubMed Central
PMCID
2936015
retrieved
31 October 2017
PMCID
2936015
1 reference
stated in
Europe PubMed Central
PMCID
2936015
retrieved
31 October 2017
PubMed ID
20590599
1 reference
stated in
Europe PubMed Central
PMCID
2936015
retrieved
31 October 2017
ResearchGate publication ID
44887548
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