(Q42876787)

9 November 2017

title

Potent and selective HIV-1 ribonuclease H inhibitors based on a 1-hydroxy-1,8-naphthyridin-2(1H)-one scaffold (English)

1 reference

9 November 2017

Shankar Venkatraman

3

1 reference

9 November 2017

Geetha Dornadula

17

1 reference

9 November 2017

Peter D. Williams

1

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A20869872

20 July 2024

Donnette D. Staas

2

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A20869872

20 July 2024

H. Marie Loughran

4

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A20869872

20 July 2024

Rowena D. Ruzek

5

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A20869872

20 July 2024

Theresa M. Booth

6

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A20869872

20 July 2024

Terry A. Lyle

7

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A20869872

20 July 2024

John S. Wai

8

1 reference

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20 July 2024

Joseph P. Vacca

9

1 reference

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20 July 2024

Bradley P. Feuston

10

1 reference

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20 July 2024

Linda T. Ecto

11

1 reference

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20 July 2024

Jessica A. Flynn

12

1 reference

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20 July 2024

Daniel J. DiStefano

13

1 reference

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20 July 2024

Daria J. Hazuda

14

1 reference

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20 July 2024

Carolyn M. Bahnck

15

1 reference

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20 July 2024

Amy L. Himmelberger

16

1 reference

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20 July 2024

Renee C. Hrin

18

1 reference

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20 July 2024

Kara A. Stillmock

19

1 reference

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20 July 2024

Marc V. Witmer

20

1 reference

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20 July 2024

Michael D. Miller

21

1 reference

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20 July 2024

Jay A. Grobler

22

1 reference

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20 July 2024

language of work or name

English

0 references

publication date

24 September 2010

1 reference

full work available at URL

9 November 2017

number of pages

4

1 reference

based on heuristic

inferred from page(s)

https://api.elsevier.com/content/article/PII:S0960894X10012710?httpAccept=text/xml

1 reference

https://api.crossref.org/works/10.1016/J.BMCL.2010.08.135

https://api.elsevier.com/content/article/PII:S0960894X10012710?httpAccept=text/plain

20 July 2024

1 reference

https://api.crossref.org/works/10.1016/J.BMCL.2010.08.135

Bioorganic & Medicinal Chemistry Letters

20 July 2024

published in

1 reference

9 November 2017

volume

20

1 reference

9 November 2017

issue

22

1 reference

9 November 2017

page(s)

6754-6757

1 reference

Efficacy and safety of once-daily regimens in the treatment of HIV infection

9 November 2017

cites work

1

1 reference

https://api.crossref.org/works/10.1016/J.BMCL.2010.08.135

RNase H activity: structure, specificity, and function in reverse transcription

20 July 2024

2

1 reference

https://api.crossref.org/works/10.1016/J.BMCL.2010.08.135

Recent progress in the design of small molecule inhibitors of HIV RNase H.

20 July 2024

3

1 reference

https://api.crossref.org/works/10.1016/J.BMCL.2010.08.135

Stepwise analyses of metal ions in RNase H catalysis from substrate destabilization to product release

20 July 2024

4

1 reference

https://api.crossref.org/works/10.1016/J.BMCL.2010.08.135

Inhibition of HIV-1 ribonuclease H by a novel diketo acid, 4-[5-(benzoylamino)thien-2-yl]-2,4-dioxobutanoic acid

20 July 2024

5

1 reference

https://api.crossref.org/works/10.1016/J.BMCL.2010.08.135

Two-metal ion mechanism of RNA cleavage by HIV RNase H and mechanism-based design of selective HIV RNase H inhibitors

20 July 2024

6

1 reference

https://api.crossref.org/works/10.1016/J.BMCL.2010.08.135

Structure of HIV-1 Reverse Transcriptase with the Inhibitor β-Thujaplicinol Bound at the RNase H Active Site

20 July 2024

7

1 reference

https://api.crossref.org/works/10.1016/J.BMCL.2010.08.135

RNase H active site inhibitors of human immunodeficiency virus type 1 reverse transcriptase: design, biochemical activity, and structural information

20 July 2024

8

1 reference

https://api.crossref.org/works/10.1016/J.BMCL.2010.08.135

Structural Basis for the Inhibition of RNase H Activity of HIV-1 Reverse Transcriptase by RNase H Active Site-Directed Inhibitors

20 July 2024

10

1 reference

https://api.crossref.org/works/10.1016/J.BMCL.2010.08.135

Inhibitors of HCV NS5B polymerase: synthesis and structure-activity relationships of N-1-heteroalkyl-4-hydroxyquinolon-3-yl-benzothiadiazines

20 July 2024

11

1 reference

https://api.crossref.org/works/10.1016/J.BMCL.2010.08.135

Dissecting the effects of DNA polymerase and ribonuclease H inhibitor combinations on HIV-1 reverse-transcriptase activities

20 July 2024

12

1 reference

https://api.crossref.org/works/10.1016/J.BMCL.2010.08.135

Diketo acid inhibitor mechanism and HIV-1 integrase: implications for metal binding in the active site of phosphotransferase enzymes

20 July 2024

13

1 reference

https://api.crossref.org/works/10.1016/J.BMCL.2010.08.135

Inhibitors of strand transfer that prevent integration and inhibit HIV-1 replication in cells

20 July 2024

14

1 reference

https://api.crossref.org/works/10.1016/J.BMCL.2010.08.135

Comparison of alamar blue and MTT assays for high through-put screening

20 July 2024

15

1 reference

https://api.crossref.org/works/10.1016/J.BMCL.2010.08.135

L-735,524: an orally bioavailable human immunodeficiency virus type 1 protease inhibitor

20 July 2024

16

1 reference

https://api.crossref.org/works/10.1016/J.BMCL.2010.08.135

20 July 2024

Identifiers

1 reference

9 November 2017

1 reference