(Q44902867)

7 December 2017

title

Solid-phase intramolecular N-acyliminium Pictet-Spengler reactions as crossroads to scaffold diversity (English)

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7 December 2017

2

Morten Meldal

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7 December 2017

Thomas E Nielsen

1

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7 December 2017

language of work or name

English

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publication date

1 May 2004

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Journal of Organic Chemistry

7 December 2017

published in

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7 December 2017

volume

69

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7 December 2017

issue

11

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7 December 2017

page(s)

3765-3773

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Comprehensive survey of combinatorial library synthesis: 2000.

7 December 2017

cites work

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Development of highly potent inhibitors of Ras farnesyltransferase possessing cellular and in vivo activity.

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Recent advances in the preparation of heterocycles on solid support: a review of the literature

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3HPropyl ?-Carboline-3-Carboxylate as a Selective Radioligand for the BZ1Benzodiazepine Receptor Subclass

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Design and synthesis of somatostatin analogues with topographical properties that lead to highly potent and specific mu opioid receptor antagonists with greatly reduced binding at somatostatin receptors

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Tetrahydroisoquinoline derivatives containing a benzenesulfonamide moiety as potent, selective human beta3 adrenergic receptor agonists

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Neuromuscular blocking activity and therapeutic potential of mixed-tetrahydroisoquinolinium halofumarates and halosuccinates in rhesus monkeys

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Recent developments in combinatorial organic synthesis.

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2-Amino- and 2-guanidino-1,2,3,4-tetrahydro-1,4-epoxynaphthalenes as conformationally defined analogues of alpha-adrenergic agents

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Identification of (3R)-7-hydroxy-N-((1S)-1-[[(3R,4R)-4-(3-hydroxyphenyl)- 3,4-dimethyl-1-piperidinyl]methyl]-2-methylpropyl)-1,2,3,4-tetrahydro- 3-isoquinolinecarboxamide as a novel potent and selective opioid kappa receptor antagonist.

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6-Methylergoline-8-carboxylic acid esters as serotonin antagonists: N1-substituent effects on 5HT2 receptor affinity

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Urinary and brain beta-carboline-3-carboxylates as potent inhibitors of brain benzodiazepine receptors

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The recent impact of solid-phase synthesis on medicinally relevant benzoannelated nitrogen heterocycles.

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High-speed combinatorial synthesis utilizing microwave irradiation

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Chemistry and biology of the tetrahydroisoquinoline antitumor antibiotics

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Solid-Phase Synthesis of Tetrahydro-β-carbolinehydantoins via theN-Acyliminium Pictet−Spengler Reaction and Cyclative Cleavage

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Amino Acid-Derived Heterocycles as Combinatorial Library Targets: Bicyclic Aminal Lactones

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HR22C16: a potent small-molecule probe for the dynamics of cell division

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11 October 2022

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beta-Turned dipeptoids as potent and selective CCK(1) receptor antagonists.

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11 October 2022

https://opencitations.net/index/coci/api/v1/references/10.1021/JO049918P

Identifiers

DOI

10.1021/JO049918P

0 references

1 reference