(Q45127785)

English

Use of photoaffinity labeling and site-directed mutagenesis for identification of the key residue responsible for extraordinarily high affinity binding of UCN-01 in human alpha1-acid glycoprotein.

scientific article published on 27 October 2004

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scholarly article

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Europe PubMed Central

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:15509559%20AND%20SRC:MED&resulttype=core&format=json

4 January 2020

Use of photoaffinity labeling and site-directed mutagenesis for identification of the key residue responsible for extraordinarily high affinity binding of UCN-01 in human alpha1-acid glycoprotein (English)

1 reference

Europe PubMed Central

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:15509559%20AND%20SRC:MED&resulttype=core&format=json

4 January 2020

Victor Tuan Giam Chuang

2

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:15509559%20AND%20SRC:MED&resulttype=core&format=json

4 January 2020

Noriyuki Yamaotsu

6

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4 January 2020

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Masaaki Katsuki

1

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4 January 2020

Koji Nishi

3

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4 January 2020

Kohichi Kawahara

4

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4 January 2020

Hitoshi Nakayama

5

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4 January 2020

Shuichi Hirono

7

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4 January 2020

Masaki Otagiri

8

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4 January 2020

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27 October 2004

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4 January 2020

Journal of Biological Chemistry

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4 January 2020

280

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4 January 2020

2

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4 January 2020

1384-1391

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4 January 2020

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UCN-01-induced cell cycle arrest requires the transcriptional induction of p21(waf1/cip1) by activation of mitogen-activated protein/extracellular signal-regulated kinase kinase/extracellular signal-regulated kinase pathway

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UCN-01 (7-hydroxystaurosporine) enhances 5-fluorouracil cytotoxicity through down-regulation of thymidylate synthetase messenger RNA.

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The binding of selected therapeutic drugs to human serum alpha-1 acid glycoprotein and to human serum albumin in vitro

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21 January 2018

Evaluation of the protein binding ratio of drugs by a micro-scale ultracentrifugation method

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21 January 2018

Tryptophan residues play an important role in the extraordinarily high affinity binding interaction of UCN-01 to human alpha-1-acid glycoprotein

1 reference

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21 January 2018

Photoaffinity labeling in drug discovery and developments: chemical gateway for entering proteomic frontier

1 reference

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21 January 2018

Identification of a critical ankyrin-binding loop on the cytoplasmic domain of erythrocyte membrane band 3 by crystal structure analysis and site-directed mutagenesis

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Amino acid mutagenesis of the ligand binding site and the dimer interface of the metabotropic glutamate receptor 1. Identification of crucial residues for setting the activated state

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21 January 2018

Construction of expression system for human alpha 1-acid glycoprotein in Pichia pastoris and evaluation of its drug-binding properties

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21 January 2018

Linearization of the Bradford protein assay increases its sensitivity: theoretical and experimental studies

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Analysis of peptide mixtures by capillary high performance liquid chromatography: a practical guide to small-scale separations

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21 January 2018

Structure of human alpha1-acid glycoprotein and its high-affinity binding site

1 reference

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21 January 2018

Structural basis for Chk1 inhibition by UCN-01

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21 January 2018

A fast flexible docking method using an incremental construction algorithm.

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21 January 2018

Development and validation of a genetic algorithm for flexible docking

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21 January 2018

A general and fast scoring function for protein-ligand interactions: a simplified potential approach.

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A geometric approach to macromolecule-ligand interactions

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Empirical scoring functions: I. The development of a fast empirical scoring function to estimate the binding affinity of ligands in receptor complexes.

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21 January 2018

Human alpha-1-glycoprotein and its interactions with drugs

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Hydrophobic and ionic factors in the binding of local anesthetics to the major variant of human alpha1-acid glycoprotein

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The plasma protein binding of basic drugs

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Structural basis for UCN-01 (7-hydroxystaurosporine) specificity and PDK1 (3-phosphoinositide-dependent protein kinase-1) inhibition

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12 April 2024

https://opencitations.net/index/api/v1/citations/10.7164/ANTIBIOTICS.40.1782

Identifiers

10.1074/JBC.M411076200

1 reference

Europe PubMed Central

PubMed publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:15509559%20AND%20SRC:MED&resulttype=core&format=json

4 January 2020

PubMed publication ID

1 reference

Europe PubMed Central

PubMed publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:15509559%20AND%20SRC:MED&resulttype=core&format=json

4 January 2020

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