(Q46248926)

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SLV313 (1-(2,3-dihydro-benzo[1,4]dioxin-5-yl)-4- [5-(4-fluoro-phenyl)-pyridin-3-ylmethyl]-piperazine monohydrochloride): a novel dopamine D2 receptor antagonist and 5-HT1A receptor agonist potential antipsychotic drug.

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Europe PubMed Central

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:16710314%20AND%20SRC:MED&resulttype=core&format=json

21 January 2020

SLV313 (1-(2,3-dihydro-benzo[1,4]dioxin-5-yl)-4- [5-(4-fluoro-phenyl)-pyridin-3-ylmethyl]-piperazine monohydrochloride): a novel dopamine D2 receptor antagonist and 5-HT1A receptor agonist potential antipsychotic drug (English)

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Europe PubMed Central

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:16710314%20AND%20SRC:MED&resulttype=core&format=json

21 January 2020

Jeffrey C Glennon

2

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21 January 2020

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Andrew C McCreary

1

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21 January 2020

Charles R Ashby

3

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21 January 2020

Herbert Y Meltzer

4

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21 January 2020

Zhu Li

5

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21 January 2020

Jan-Hendrik Reinders

6

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21 January 2020

Mayke B Hesselink

7

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21 January 2020

Stephen K Long

8

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21 January 2020

Arnoud H Herremans

9

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21 January 2020

Herman van Stuivenberg

10

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21 January 2020

Rolf W Feenstra

11

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21 January 2020

Chris G Kruse

12

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21 January 2020

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17 May 2006

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21 January 2020

Neuropsychopharmacology

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21 January 2020

32

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21 January 2020

1

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21 January 2020

78-94

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21 January 2020

Contrasting contribution of 5-hydroxytryptamine 1A receptor activation to neurochemical profile of novel antipsychotics: frontocortical dopamine and hippocampal serotonin release in rat brain

1 reference

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21 January 2018

The 5-HT1A receptor in schizophrenia: a promising target for novel atypical neuroleptics?

1 reference

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21 January 2018

Selective activation of 5HT1A receptors induces lower lip retraction in the rat.

1 reference

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21 January 2018

Direct evidence for an important species difference in the mechanism of 8-OH-DPAT-induced hypothermia

1 reference

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21 January 2018

The pharmacology and distribution of human 5‐hydroxytryptamine2B (5‐HT2b) receptor gene products: comparison with 5‐HT2a and 5‐HT2c receptors

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1301098

21 January 2018

Cloning and expression of a rat D2 dopamine receptor cDNA

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1301098

21 January 2018

5-HT1A and 5-HT2A receptor mRNAs and binding site densities are differentially altered in schizophrenia

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1301098

21 January 2018

Dopamine-containing neurons in the mammalian central nervous system: electrophysiology and pharmacology

1 reference

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21 January 2018

Reversal of haloperidol-induced extrapyramidal side effects in cebus monkeys by 8-hydroxy-2-(di-n-propylamino)tetralin and its enantiomers

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1301098

21 January 2018

Clozapine increases both acetylcholine and dopamine release in rat ventral hippocampus: role of 5-HT1A receptor agonism

1 reference

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21 January 2018

SSR181507, a dopamine D2 receptor antagonist and 5-HT1A receptor agonist. II: Behavioral profile predictive of an atypical antipsychotic activity

1 reference

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21 January 2018

Heterogeneity of [3H]-mepyramine binding sites in guinea pig cerebellum and lung

1 reference

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21 January 2018

The hippocampus, memory, and place cells: is it spatial memory or a memory space?

1 reference

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21 January 2018

Human declarative memory formation: segregating rhinal and hippocampal contributions.

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1301098

21 January 2018

Cloning of the cDNA and gene for a human D2 dopamine receptor

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1301098

21 January 2018

Binding characteristics of 3H-prazosin to rat brain α-adrenergic receptors

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1301098

21 January 2018

Alterations in the cortical serotonergic system in schizophrenia: a postmortem study

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1301098

21 January 2018

Serotonergic and histaminergic mechanisms involved in intralipid drinking?

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1301098

21 January 2018

Studies of cognitive change in patients with schizophrenia following novel antipsychotic treatment

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1301098

21 January 2018

The 5-HT1A receptor agonist flesinoxan shares discriminative stimulus properties with some 5-HT2 receptor antagonists.

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1301098

21 January 2018

Risperidone: regional effects in vivo on release and metabolism of dopamine and serotonin in the rat brain

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1301098

21 January 2018

Characterization of a human 5-hydroxytryptamine3 receptor type A (h5-HT3R-AS) subunit stably expressed in HEK 293 cells

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1301098

21 January 2018

Atypical, but not typical, antipsychotic drugs increase cortical acetylcholine release without an effect in the nucleus accumbens or striatum

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1301098

21 January 2018

5-HT(2A) and D(2) receptor blockade increases cortical DA release via 5-HT(1A) receptor activation: a possible mechanism of atypical antipsychotic-induced cortical dopamine release

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1301098

21 January 2018

Preclinical neurochemical and electrophysiological profile of 1192U90, a potential antipsychotic

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1301098

21 January 2018

The antipsychotic aripiprazole is a potent, partial agonist at the human 5-HT1A receptor

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1301098

21 January 2018

Dopamine D3 receptor antagonists as therapeutic agents

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1301098

21 January 2018

Clozapine inhibits serotoninergic transmission by an action at alpha 1-adrenoceptors not at 5-HT1A receptors

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1301098

21 January 2018

Aripiprazole, a novel antipsychotic drug, preferentially increases dopamine release in the prefrontal cortex and hippocampus in rat brain

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1301098

21 January 2018

Characterization of the human dopamine D3 receptor expressed in transfected cell lines

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1301098

21 January 2018

The role of serotonin in antipsychotic drug action

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1301098

21 January 2018

Serotonin receptors: their key role in drugs to treat schizophrenia

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1301098

21 January 2018

The effects of clozapine, risperidone, and olanzapine on cognitive function in schizophrenia

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1301098

21 January 2018

Pharmacological characterization of the human 5-HT(4(d)) receptor splice variant stably expressed in Chinese hamster ovary cells

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1301098

21 January 2018

Acute effects of typical and atypical antipsychotic drugs on the release of dopamine from prefrontal cortex, nucleus accumbens, and striatum of the rat: an in vivo microdialysis study

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1301098

21 January 2018

The putative 5-HT1A receptor antagonist DU125530 blocks the discriminative stimulus of the 5-HT1A receptor agonist flesinoxan in pigeons

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1301098

21 January 2018

The acute and chronic administration of (+/-)-8-hydroxy-2-(Di-n-propylamino)tetralin significantly alters the activity of spontaneously active midbrain dopamine neurons in rats: an in vivo electrophysiological study

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1301098

21 January 2018

Clozapine is a partial agonist at cloned, human serotonin 5-HT1A receptors.

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1301098

21 January 2018

Efficacy of antipsychotic agents at human 5-HT(1A) receptors determined by [3H]WAY100,635 binding affinity ratios: relationship to efficacy for G-protein activation

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1301098

21 January 2018

Systemic administration of amperozide, a new atypical antipsychotic drug, preferentially increases dopamine release in the rat medial prefrontal cortex

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1301098

21 January 2018

The atypical antipsychotic drug amperozide enhances rat cortical and striatal dopamine efflux

1 reference

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21 January 2018

Effects of dopamine antagonists in a two-way active avoidance procedure in rats: interactions with 8-OH-DPAT, ritanserin, and prazosin.

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1301098

21 January 2018

Repeated treatment with 8-OH-DPAT induces tolerance to its ability to produce the 5-HT1A behavioural syndrome, but not to its ability to attenuate haloperidol-induced catalepsy

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1301098

21 January 2018

Association of antipsychotic drug-induced weight gain with a 5-HT2C receptor gene polymorphism

1 reference

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21 January 2018

5-HT(1A) receptor activation contributes to ziprasidone-induced dopamine release in the rat prefrontal cortex

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1301098

21 January 2018

Clozapine increases dopamine release in prefrontal cortex by 5-HT1A receptor activation

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1301098

21 January 2018

A highly sensitive adenylate cyclase assay

1 reference

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21 January 2018

Antipsychotic drug doses and neuroleptic/dopamine receptors

1 reference

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21 January 2018

A comparative profile analysis of neuropsychological functioning in patients with schizophrenia and bipolar psychoses.

1 reference

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21 January 2018

Effects of typical and atypical antipsychotics and receptor selective compounds on acetylcholine efflux in the hippocampus of the rat.

1 reference

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21 January 2018

Comparison of the novel antipsychotic ziprasidone with clozapine and olanzapine: inhibition of dorsal raphe cell firing and the role of 5-HT1A receptor activation

1 reference

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21 January 2018

Enhancement of cognitive performance in schizophrenia by addition of tandospirone to neuroleptic treatment

1 reference

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21 January 2018

The effect of tandospirone, a serotonin(1A) agonist, on memory function in schizophrenia

1 reference

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21 January 2018

Pharmacological profile of antidepressants and related compounds at human monoamine transporters

1 reference

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21 January 2018

The involvement of subtypes of the 5-HT1 receptor and of catecholaminergic systems in the behavioural response to 8-hydroxy-2-(di-n-propylamino)tetralin in the rat.

1 reference

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21 January 2018

Rat spinal cord alpha 2-adrenoceptors are of the alpha 2A-subtype: comparison with alpha 2A- and alpha 2B-adrenoceptors in rat spleen, cerebral cortex and kidney using 3H-RX821002 ligand binding

1 reference

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21 January 2018

Multiple dopamine D4 receptor variants in the human population

1 reference

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21 January 2018

Serotonergic mechanisms in neuroleptic-induced catalepsy in the rat.

1 reference

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21 January 2018

Effects of local application of 5-hydroxytryptamine into the dorsal or median raphe nuclei on haloperidol-induced catalepsy in the rat

1 reference

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21 January 2018

Cortical maldevelopment, anti-psychotic drugs, and schizophrenia: a search for common ground

1 reference

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21 January 2018

Corticotropin-peptide regulation of intracellular cyclic AMP production in cortical neurons in primary culture

1 reference

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21 January 2018

Differential Effects of Classical and Atypical Antipsychotic Drugs on A9 and A10 Dopamine Neurons

1 reference

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21 January 2018

Intra-prefrontal 8-OH-DPAT and M100907 improve visuospatial attention and decrease impulsivity on the five-choice serial reaction time task in rats.

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1301098

21 January 2018

Decreased 5-HT1A receptor binding in amygdala of schizophrenia

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1301098

21 January 2018

Effect of tandospirone on tardive dyskinesia and parkinsonian symptoms.

1 reference

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21 January 2018

Typical and atypical neuroleptics: differential effects of chronic administration on the activity of A9 and A10 midbrain dopaminergic neurons

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1301098

7 January 2021

based on heuristic

inferred from DOI database lookup

SSR181507, a dopamine D(2) receptor antagonist and 5-HT(1A) receptor agonist. I: Neurochemical and electrophysiological profile.

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1301098

7 January 2021

based on heuristic

inferred from DOI database lookup

The cortical dopamine system: role in memory and cognition

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1301098

7 January 2021

based on heuristic

inferred from DOI database lookup

Interactions between neuroleptics and 5-HT(1A) ligands in preclinical behavioral models for antipsychotic and extrapyramidal effects

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1301098

7 January 2021

based on heuristic

inferred from DOI database lookup

Antipsychotic-like profile of combined treatment with raclopride and 8-OH-DPAT in the rat: enhancement of antipsychotic-like effects without catalepsy

1 reference

https://api.crossref.org/works/10.1038%2FSJ.NPP.1301098

7 January 2021

based on heuristic

inferred from DOI database lookup

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