(Q53503547)

14 May 2018

title

Interrogating 7TM receptors: does texture in the question yield greater texture in the answer? (English)

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14 May 2018

author name string

Terry Kenakin

series ordinal

1

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14 May 2018

publication date

1 January 2009

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14 May 2018

Journal of Receptors and Signal Transduction

published in

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14 May 2018

volume

29

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14 May 2018

issue

3-4

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14 May 2018

page(s)

132-139

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14 May 2018

Intrinsic disorder in transcription factors

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Functionally selective M1 muscarinic agonists. 3. Side chains and azacycles contributing to functional muscarinic selectivity among pyrazinylazacycles

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Ligand-selective receptor conformations revisited: the promise and the problem

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Illuminating insights into protein-protein interactions using bioluminescence resonance energy transfer (BRET).

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Functional Selectivity and Classical Concepts of Quantitative Pharmacology

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Regulation of receptor-coupling to (multiple) G proteins. A challenge for basic research and drug discovery

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A novel, conformation-specific allosteric inhibitor of the tachykinin NK2 receptor (NK2R) with functionally selective properties

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Distinct receptor activity-modifying protein domains differentially modulate interaction with calcitonin receptors

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Beta-arrestin-mediated activation of MAPK by inverse agonists reveals distinct active conformations for G protein-coupled receptors

21 January 2018

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Agonist and inverse agonist actions of beta-blockers at the human beta 2-adrenoceptor provide evidence for agonist-directed signaling

21 January 2018

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Distinct signaling profiles of beta1 and beta2 adrenergic receptor ligands toward adenylyl cyclase and mitogen-activated protein kinase reveals the pluridimensionality of efficacy

21 January 2018

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Historical review: a brief history and personal retrospective of seven-transmembrane receptors

21 January 2018

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Transduction of receptor signals by beta-arrestins

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New roles for beta-arrestins in cell signaling: not just for seven-transmembrane receptors

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Bombesin and substance P analogues differentially regulate G-protein coupling to the bombesin receptor. Direct evidence for biased agonism

21 January 2018

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21 January 2018

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The ligand paradox between affinity and efficacy: can you be there and not make a difference?

21 January 2018

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10.1080/10799890903050829

21 January 2018

Identifiers

DOI

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14 May 2018

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14 May 2018