(Q54242505)

26 May 2018

title

Selective ligands for rat A3 adenosine receptors: structure-activity relationships of 1,3-dialkylxanthine 7-riboside derivatives. (English)

1 reference

26 May 2018

author name string

H O Kim

1

1 reference

26 May 2018

X D Ji

2

1 reference

26 May 2018

N Melman

3

1 reference

26 May 2018

M E Olah

4

1 reference

26 May 2018

G L Stiles

5

1 reference

26 May 2018

K A Jacobson

6

1 reference

26 May 2018

language of work or name

English

0 references

publication date

1 November 1994

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26 May 2018

Journal of Medicinal Chemistry

published in

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26 May 2018

volume

37

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26 May 2018

issue

23

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26 May 2018

page(s)

4020-4030

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26 May 2018

Structure-activity relationships of 8-styrylxanthines as A2-selective adenosine antagonists

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1 reference

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8-(3-Chlorostyryl)caffeine (CSC) is a selective A2-adenosine antagonist in vitro and in vivo

26 May 2018

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Adenosine A3 receptors mediate hypotension in the angiotensin II-supported circulation of the pithed rat.

26 May 2018

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The A3 adenosine receptor is the unique adenosine receptor which facilitates release of allergic mediators in mast cells

26 May 2018

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A role for central A3-adenosine receptors. Mediation of behavioral depressant effects

26 May 2018

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Molecular cloning and characterization of the human A3 adenosine receptor

26 May 2018

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125I-4-aminobenzyl-5'-N-methylcarboxamidoadenosine, a high affinity radioligand for the rat A3 adenosine receptor

26 May 2018

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Structure-activity relationships of N6-benzyladenosine-5'-uronamides as A3-selective adenosine agonists

26 May 2018

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A binding site model and structure-activity relationships for the rat A3 adenosine receptor

26 May 2018

1 reference

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Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

26 May 2018

1 reference

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Iodine-125-labeled 8-phenylxanthine derivatives: antagonist radioligands for adenosine A1 receptors

26 May 2018

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8-Aryl-and 8-cycloalkyl-1,3-dipropylxanthines: further potent and selective antagonists for A1-adenosine receptors

26 May 2018

1 reference

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8-Substituted xanthines as antagonists at A1- and A2-adenosine receptors.

26 May 2018

1 reference

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A functionalized congener approach to adenosine receptor antagonists: amino acid conjugates of 1,3-dipropylxanthine

26 May 2018

1 reference

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Functionalized congeners of 1,3-dialkylxanthines: preparation of analogues with high affinity for adenosine receptors

26 May 2018

1 reference

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Sulfur-containing 1,3-dialkylxanthine derivatives as selective antagonists at A1-adenosine receptors.

26 May 2018

1 reference

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[3H]CGS 21680, a selective A2 adenosine receptor agonist directly labels A2 receptors in rat brain

26 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5875426

Activation of phospholipase C via adenosine receptors provides synergistic signals for secretion in antigen-stimulated RBL-2H3 cells. Evidence for a novel adenosine receptor.

26 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5875426

RDC8 codes for an adenosine A2 receptor with physiological constitutive activity.

26 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5875426

Structure and function of A1 adenosine receptors

26 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5875426

Adenosine receptors: pharmacology, structure-activity relationships, and therapeutic potential

26 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5875426

Molecular cloning of a novel putative G-protein coupled receptor expressed during rat spermiogenesis

26 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5875426

The orphan receptor cDNA RDC7 encodes an A1 adenosine receptor

26 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5875426

26 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5875426

Molecular cloning and characterization of an adenosine receptor: the A3 adenosine receptor

26 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5875426

Molecular cloning and functional expression of a sheep A3 adenosine receptor with widespread tissue distribution.

26 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=5875426

Characterization of adenosine receptors in rat brain by (?)[3H]N6-phenylisopropyladenosine

13 August 2018

1 reference

12 December 2020

Evidence that the adenosine A3 receptor may mediate the protection afforded by preconditioning in the isolated rabbit heart

1 reference

12 December 2020

BW-A522 blocks adenosine A3 receptor-mediated hypotensive responses in the rat

1 reference

12 December 2020

Effect of trifluoromethyl and other substituents on activity of xanthines at adenosine receptors

1 reference

12 December 2020

Photoisomerization of a potent and selective adenosine A2 antagonist, (E)-1,3-Dipropyl-8-(3,4-dimethoxystyryl)-7-methylxanthine

1 reference

12 December 2020

Identifiers

DOI

10.1021/JM00049A021

1 reference

26 May 2018

PMC publication ID

5875426

1 reference

26 May 2018

PubMed publication ID

7966162

1 reference

26 May 2018