(Q63423653)

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Synthesis and Structure-Activity Relationships of FAAH Inhibitors: Cyclohexylcarbamic Acid Biphenyl Esters with Chemical Modulation at the Proximal Phenyl Ring

scientific article published on 01 January 2006

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scholarly article

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Europe PubMed Central

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28 December 2019

Synthesis and structure-activity relationships of FAAH inhibitors: cyclohexylcarbamic acid biphenyl esters with chemical modulation at the proximal phenyl ring (English)

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28 December 2019

Giovanni Piersanti

4

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28 December 2019

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28 December 2019

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28 December 2019

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28 December 2019

Satish Kathuria

10

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Satish Kathuria

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28 December 2019

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Andrea Duranti

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28 December 2019

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Andrea Tontini

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28 December 2019

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Giorgio Tarzia

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28 December 2019

Pier Vincenzo Plazzi

8

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Pier Vincenzo Plazzi

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28 December 2019

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Giuseppe Gatti

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28 December 2019

Daniele Piomelli

11

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28 December 2019

publication date

1 January 2006

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28 December 2019

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28 December 2019

1

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28 December 2019

1

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28 December 2019

130-139

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28 December 2019

The molecular logic of endocannabinoid signalling

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Fatty acid amide hydrolase: an emerging therapeutic target in the endocannabinoid system

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Anandamide hydrolysis: a new target for anti-anxiety drugs?

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Fatty acid sulfonyl fluorides inhibit anandamide metabolism and bind to the cannabinoid receptor

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Methyl arachidonyl fluorophosphonate: a potent irreversible inhibitor of anandamide amidase

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Trifluoromethyl ketone inhibitors of fatty acid amide hydrolase: a probe of structural and conformational features contributing to inhibition

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alpha-Keto heterocycle inhibitors of fatty acid amide hydrolase: carbonyl group modification and alpha-substitution

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7 January 2021

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Discovery of a potent, selective, and efficacious class of reversible alpha-ketoheterocycle inhibitors of fatty acid amide hydrolase effective as analgesics

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7 January 2021

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Discovery of an exceptionally potent and selective class of fatty acid amide hydrolase inhibitors enlisting proteome-wide selectivity screening: concurrent optimization of enzyme inhibitor potency and selectivity

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7 January 2021

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Design, synthesis, and structure-activity relationships of alkylcarbamic acid aryl esters, a new class of fatty acid amide hydrolase inhibitors.

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7 January 2021

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Cyclohexylcarbamic acid 3'- or 4'-substituted biphenyl-3-yl esters as fatty acid amide hydrolase inhibitors: synthesis, quantitative structure-activity relationships, and molecular modeling studies

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7 January 2021

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Characterization of the fatty acid amide hydrolase inhibitor cyclohexyl carbamic acid 3'-carbamoyl-biphenyl-3-yl ester (URB597): effects on anandamide and oleoylethanolamide deactivation.

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Tandem mass spectrometric data-FAAH inhibitory activity relationships of some carbamic acid O-aryl esters

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QM/MM modelling of oleamide hydrolysis in fatty acid amide hydrolase (FAAH) reveals a new mechanism of nucleophile activation.

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Identifiers

10.1002/CMDC.200500017

1 reference

Europe PubMed Central

PubMed publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:16892344%20AND%20SRC:MED&resulttype=core&format=json

28 December 2019

PubMed publication ID

1 reference

Europe PubMed Central

PubMed publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:16892344%20AND%20SRC:MED&resulttype=core&format=json

28 December 2019

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