(Q27632621)

1

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Maria Paola Costi

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ORCID Public Data File 2021

author name string

R A Powers

2

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M C Negri

4

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J Blázquez

5

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M P Costi

6

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B K Shoichet

The crisis in antibiotic resistance

7

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publication date

June 2001

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published in

Chemistry and Biology

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volume

8

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issue

6

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page(s)

593-611

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cites work

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2801%2900034-5

7 January 2021

Evolution of antibiotic resistance

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7 January 2021

Beta-lactamase inhibitors and reversal of antibiotic resistance

1 reference

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7 January 2021

beta-Lactamases of gram-negative bacteria: new challenges for new drugs

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7 January 2021

Inactivation of antibiotics and the dissemination of resistance genes

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7 January 2021

The inhibition of class C beta-lactamases by boronic acids

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2801%2900034-5

7 January 2021

Structure-based design of a potent transition state analogue for TEM-1 beta-lactamase

1 reference

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7 January 2021

Structure-based enhancement of boronic acid-based inhibitors of AmpC beta-lactamase.

1 reference

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7 January 2021

The complexed structure and antimicrobial activity of a non-β-lactam inhibitor of AmpC β-lactamase

1 reference

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7 January 2021

Structure-based design guides the improved efficacy of deacylation transition state analogue inhibitors of TEM-1 beta-Lactamase(,)

1 reference

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7 January 2021

Energetic, structural, and antimicrobial analyses of beta-lactam side chain recognition by beta-lactamases

1 reference

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7 January 2021

Three-dimensional structure of AmpC beta-lactamase from Escherichia coli bound to a transition-state analogue: possible implications for the oxyanion hypothesis and for inhibitor design

1 reference

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7 January 2021

Refined crystal structure of beta-lactamase from Citrobacter freundii indicates a mechanism for beta-lactam hydrolysis

1 reference

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7 January 2021

Crystallographic structure of a phosphonate derivative of the Enterobacter cloacae P99 cephalosporinase: mechanistic interpretation of a beta-lactamase transition-state analog

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2801%2900034-5

7 January 2021

Synthesis and Applications of Small Molecule Libraries

1 reference

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7 January 2021

Structure-based design and combinatorial chemistry yield low nanomolar inhibitors of cathepsin D.

1 reference

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7 January 2021

Structure-based discovery and in-parallel optimization of novelcompetitive inhibitors of thymidylate synthase

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2801%2900034-5

7 January 2021

Flexible ligand docking using conformational ensembles

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2801%2900034-5

7 January 2021

A quick method for the determination of inhibition constants

1 reference

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7 January 2021

Automated docking with grid-based energy evaluation

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2801%2900034-5

7 January 2021

Structure of the extended-spectrum class C beta-lactamase of Enterobacter cloacae GC1, a natural mutant with a tandem tripeptide insertion

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2801%2900034-5

7 January 2021

PROCHECK: a program to check the stereochemical quality of protein structures

1 reference

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7 January 2021

Molecular structure of the acyl-enzyme intermediate in beta-lactam hydrolysis at 1.7 A resolution

1 reference

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7 January 2021

Structure of a phosphonate-inhibited beta-lactamase. An analog of the tetrahedral transition state/intermediate of beta-lactam hydrolysis

1 reference

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7 January 2021

Beta-lactamase inhibitors. The inhibition of serine beta-lactamases by specific boronic acids

1 reference

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7 January 2021

Structure-based drug design: progress, results and challenges

1 reference

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7 January 2021

Structure-based drug design

1 reference

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7 January 2021

What makes a binding site a binding site?

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2801%2900034-5

7 January 2021

Structure-based discovery of inhibitors of thymidylate synthase

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2801%2900034-5

7 January 2021

Predicting the structure of protein complexes: a step in the right direction

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2801%2900034-5

7 January 2021

Molecular docking programs successfully predict the binding of a beta-lactamase inhibitory protein to TEM-1 beta-lactamase

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2801%2900034-5

7 January 2021

Kinetic properties of the binding of alpha-lytic protease to peptide boronic acids

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2801%2900034-5

7 January 2021

Iterative partial equalization of orbital electronegativity—a rapid access to atomic charges

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2801%2900034-5

7 January 2021

Molecular docking using shape descriptors

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2801%2900034-5

7 January 2021

Calculation of electrostatic potentials in an enzyme active site

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2801%2900034-5

7 January 2021

Processing of X-ray diffraction data collected in oscillation mode

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2801%2900034-5

7 January 2021

Crystallography & NMR System: A New Software Suite for Macromolecular Structure Determination

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2801%2900034-5

7 January 2021

Improved methods for building protein models in electron density maps and the location of errors in these models

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2801%2900034-5

7 January 2021

Noncovalent Adducts of Poly(ethylene glycols) with Proteins

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2801%2900034-5

7 January 2021

Synthesis of a fluorescent boronic acid which reversibly binds to cell walls and a diboronic acid which agglutinates erythrocytes

1 reference

https://api.crossref.org/works/10.1016%2FS1074-5521%2801%2900034-5

7 January 2021