(Q27667313)

22 June 2017

Turning a protein kinase on or off from a single allosteric site via disulfide trapping (English)

1 reference

22 June 2017

5

Matthew P Jacobson

Matthew P

Jacobson

1 reference

22 June 2017

Dennis W Wolan

3

Dennis W

Wolan

1 reference

19 October 2023

Jack D Sadowsky

1

Jack D

Sadowsky

1 reference

22 June 2017

Mark A Burlingame

series ordinal

2

author given names

Mark A

author last names

Burlingame

1 reference

22 June 2017

Christopher L McClendon

series ordinal

4

author given names

Christopher L

author last names

McClendon

1 reference

22 June 2017

James A Wells

series ordinal

6

author given names

James A

author last names

Wells

1 reference

22 June 2017

language of work or name

English

0 references

publication date

23 March 2011

1 reference

Proceedings of the National Academy of Sciences of the United States of America

22 June 2017

6

1 reference

based on heuristic

inferred from page(s)

published in

1 reference

22 June 2017

108

1 reference

22 June 2017

6056-6061

1 reference

22 June 2017

15

1 reference

PHENIX: a comprehensive Python-based system for macromolecular structure solution

22 June 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3076885

The impact of GPCR structures on pharmacology and structure-based drug design

20 March 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3076885

Structure and allosteric effects of low-molecular-weight activators on the protein kinase PDK1

20 March 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3076885

An allosteric mechanism for activation of the kinase domain of epidermal growth factor receptor

20 March 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3076885

Pulse proteolysis: A simple method for quantitative determination of protein stability and ligand binding

20 March 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3076885

Interactions of LY333531 and other bisindolyl maleimide inhibitors with PDK1

20 March 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3076885

Structural basis of Aurora-A activation by TPX2 at the mitotic spindle

20 March 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3076885

Crystal structure of an activated Akt/protein kinase B ternary complex with GSK3-peptide and AMP-PNP

20 March 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3076885

A phosphoserine/threonine-binding pocket in AGC kinases and PDK1 mediates activation by hydrophobic motif phosphorylation

20 March 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3076885

High resolution crystal structure of the human PDK1 catalytic domain defines the regulatory phosphopeptide docking site

20 March 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3076885

Site-directed ligand discovery

20 March 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3076885

Identification of a pocket in the PDK1 kinase domain that interacts with PIF and the C-terminal residues of PKA

20 March 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3076885

Mechanism of CDK activation revealed by the structure of a cyclinA-CDK2 complex

20 March 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3076885

Features and development of Coot

20 March 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3076885

The PIF-binding pocket in PDK1 is essential for activation of S6K and SGK, but not PKB.

20 March 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3076885

A Common Mechanism Underlying Promiscuous Inhibitors from Virtual and High-Throughput Screening

20 March 2017

1 reference

Crossref

https://api.crossref.org/works/10.1073/PNAS.1102376108

Regulation of protein kinases; controlling activity through activation segment conformation

22 April 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3076885

Lining the pockets of kinases and phosphatases.

7 April 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3076885

A common allosteric site and mechanism in caspases

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3076885

Disulfide trapping to localize small-molecule agonists and antagonists for a G protein-coupled receptor

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3076885

Structure and regulation of Src family kinases

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3076885

Discovery of an allosteric site in the caspases

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3076885

Tethering: fragment-based drug discovery

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3076885

Protein analysis by hydrogen exchange mass spectrometry

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3076885

Kinetic and catalytic mechanisms of protein kinases

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3076885

A phosphoserine-regulated docking site in the protein kinase RSK2 that recruits and activates PDK1.

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3076885

Effect of detergent on "promiscuous" inhibitors

29 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3076885

Site-specific disulfide capture of agonist and antagonist peptides on the C5a receptor

2 June 2018

1 reference

Crossref

https://api.crossref.org/works/10.1073%2FPNAS.1102376108

Identification of promiscuous small molecule activators in high-throughput enzyme activation screens

21 January 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/21430264

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1073/PNAS.1102376108

1 reference

OpenCitations bibliographic resource ID

22 June 2017

0 references

4697241

1 reference

Consolidated OpenCitations Corpus – April 2017

OpenCitations bibliographic resource ID

1 reference

Consolidated OpenCitations Corpus – April 2017

OpenCitations bibliographic resource ID

1 reference