(Q27667460)

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Structure of Estradiol Metal Chelate and Estrogen Receptor Complex: The Basis for Designing a New Class of Selective Estrogen Receptor Modulators

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scholarly article

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Structure of Estradiol Metal Chelate and Estrogen Receptor Complex: The Basis for Designing a New Class of Selective Estrogen Receptor Modulators (English)

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1 reference

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Joel L. Sussman

object named as

Joel L Sussman

9

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7

object named as

David Milstein

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8

object named as

Hadassa Degani

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5

object named as

Adi Pais

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author name string

Min-Jun Li

1

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Harry M Greenblatt

2

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Orly Dym

3

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Shira Albeck

4

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Chidambaram Gunanathan

6

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language of work or name

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publication date

26 May 2011

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Journal of Medicinal Chemistry

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54

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10

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3575-80

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PHENIX: a comprehensive Python-based system for macromolecular structure solution

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MolProbity: all-atom structure validation for macromolecular crystallography

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Structural plasticity in the oestrogen receptor ligand-binding domain

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1 reference

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Estrogen receptors and human disease

1 reference

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Crystal structure of a mutant hERalpha ligand-binding domain reveals key structural features for the mechanism of partial agonism

1 reference

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1 reference

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1 reference

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Optimal description of a protein structure in terms of multiple groups undergoing TLS motion

1 reference

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20 March 2017

electronic Ligand Builder and Optimization Workbench (eLBOW): a tool for ligand coordinate and restraint generation

1 reference

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7 April 2017

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1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3112352

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1 reference

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Water-soluble contrast agents targeted at the estrogen receptor for molecular magnetic resonance imaging.

1 reference

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Preclinical and clinical studies on the use of platinum complexes for breast cancer treatment.

1 reference

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Conformational dynamics of the estrogen receptor alpha: molecular dynamics simulations of the influence of binding site structure on protein dynamics.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3112352

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Capitalizing on the complexities of estrogen receptor pharmacology in the quest for the perfect SERM.

1 reference

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Different ligands-different receptor conformations: modeling of the hER alpha LBD in complex with agonists and antagonists

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3112352

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1 reference

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1 reference

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29 September 2017

Carboxymethylation of the human estrogen receptor ligand-binding domain-estradiol complex: HPLC/ESMS peptide mapping shows that cysteine 447 does not react with iodoacetic acid

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1 reference

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1 reference

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27 November 2018

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1 reference

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1 reference

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Molecular sensors of estrogen receptor conformations and dynamics

1 reference

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12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Processing of X-ray diffraction data collected in oscillation mode

1 reference

https://pubmed.ncbi.nlm.nih.gov/21473635

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identifiers

10.1021/JM200192Y

1 reference

Consolidated OpenCitations Corpus – April 2017

OpenCitations bibliographic resource ID

OpenCitations bibliographic resource ID

1 reference

Consolidated OpenCitations Corpus – April 2017

OpenCitations bibliographic resource ID

1 reference

Consolidated OpenCitations Corpus – April 2017

OpenCitations bibliographic resource ID

1 reference

Consolidated OpenCitations Corpus – April 2017

OpenCitations bibliographic resource ID

ResearchGate publication ID

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