(Q31572098)

3 September 2017

Combinatorial target-guided ligand assembly: identification of potent subtype-selective c-Src inhibitors (English)

1 reference

3 September 2017

2

I C Choong

1 reference

3 September 2017

D J Maly

1

1 reference

PMCID

15944

3 September 2017

J A Ellman

series ordinal

3

1 reference

PMCID

15944

3 September 2017

language of work or name

English

0 references

publication date

1 March 2000

1 reference

Proceedings of the National Academy of Sciences of the United States of America

3 September 2017

6

1 reference

based on heuristic

inferred from page(s)

published in

1 reference

3 September 2017

97

1 reference

3 September 2017

2419-2424

1 reference

3 September 2017

6

1 reference

Synthesis and Applications of Small Molecule Libraries

3 September 2017

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=15944

Comprehensive survey of combinatorial library synthesis: 1998.

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=15944

Acquisition of inhibitor-sensitive protein kinases through protein design

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=15944

Comprehensive survey of chemical libraries yielding enzyme inhibitors, receptor agonists and antagonists, and other biologically active agents: 1992 through 1997.

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=15944

Rapid identification of subtype-selective agonists of the somatostatin receptor through combinatorial chemistry

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=15944

Synthesis and biological activities of potent peptidomimetics selective for somatostatin receptor subtype 2

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=15944

Protein kinase inhibitors: the tyrosine-specific protein kinases

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=15944

Small molecule inhibitors of the platelet-derived growth factor receptor, the fibroblast growth factor receptor, and Src family tyrosine kinases

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=15944

Future pathways for combinatorial chemistry

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=15944

Structure-based design and combinatorial chemistry yield low nanomolar inhibitors of cathepsin D.

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=15944

Discovering high-affinity ligands for proteins: SAR by NMR

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=15944

SRC as a target for anti-cancer drugs

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=15944

Fluvoxamine. An updated review of its pharmacology, and therapeutic use in depressive illness

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=15944

The Src family of tyrosine protein kinases in hemopoietic signal transduction

28 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=15944

Exploiting chemical libraries, structure, and genomics in the search for kinase inhibitors

28 July 2018

1 reference

Crossref

https://api.crossref.org/works/10.1073%2FPNAS.97.6.2419

Synthesis of Alkoxylamines by Alkoxide Amination with 3,3'-Di-tert-butyloxaziridine

21 January 2018

1 reference

Crossref

https://api.crossref.org/works/10.1073%2FPNAS.97.6.2419

Discovery of a novel, potent, and Src family-selective tyrosine kinase inhibitor. Study of Lck- and FynT-dependent T cell activation

21 January 2018

1 reference

Crossref

https://api.crossref.org/works/10.1073%2FPNAS.97.6.2419

21 January 2018

1 reference

https://pubmed.ncbi.nlm.nih.gov/10716979

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Erratum [McMahon G, Sun L, Liang C, Tang C: Protein kinase inhibitors: structural determinants for target specificity. Current Opin Drug Discovery Dev (1998) 1(2):131-146. Correction to the structure of Compound 74 (SU-5874) in Figure 9]

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/10716979

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1073/PNAS.97.6.2419

1 reference

3 September 2017

0 references

1 reference

3 September 2017

1 reference

PMCID

15944