(Q33221506)

24 July 2017

title

Homogeneous high-throughput screening assays for HIV-1 integrase 3beta-processing and strand transfer activities (English)

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high-throughput screening

24 July 2017

main subject

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2

Heath Klock

1 reference

24 July 2017

Yu Wang

1

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24 July 2017

Hong Yin

3

1 reference

24 July 2017

Karen Wolff

4

1 reference

24 July 2017

Kimberly Bieza

5

1 reference

24 July 2017

Kirk Niswonger

6

1 reference

24 July 2017

Jason Matzen

7

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24 July 2017

Drew Gunderson

8

1 reference

24 July 2017

Joanna Hale

9

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24 July 2017

Scott Lesley

10

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24 July 2017

Kelli Kuhen

11

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24 July 2017

Jeremy Caldwell

12

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24 July 2017

Achim Brinker

13

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24 July 2017

publication date

1 August 2005

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Journal of Biomolecular Screening

24 July 2017

published in

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24 July 2017

volume

10

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24 July 2017

issue

5

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24 July 2017

page(s)

456-462

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https://api.crossref.org/works/10.1177%2F1087057105275212

24 July 2017

1 reference

New developments in anti-HIV chemotherapy

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105275212

HIV-1 integration as a target for antiretroviral therapy: a review

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105275212

Design and development of integrase inhibitors as anti-HIV agents

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105275212

Three new structures of the core domain of HIV-1 integrase: an active site that binds magnesium

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105275212

Metal-dependent inhibition of HIV-1 integrase

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105275212

Inhibitors of strand transfer that prevent integration and inhibit HIV-1 replication in cells

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105275212

Differential inhibition of HIV-1 preintegration complexes and purified integrase protein by small molecules

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105275212

Structural determinants for HIV-1 integrase inhibition by beta-diketo acids

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105275212

Structure activity of 3-aryl-1,3-diketo-containing compounds as HIV-1 integrase inhibitors.

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105275212

A naphthyridine carboxamide provides evidence for discordant resistance between mechanistically identical inhibitors of HIV-1 integrase

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105275212

Small-molecule HIV-1 integrase inhibitors: the 2001-2002 update

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105275212

In vitro human immunodeficiency virus type 1 integrase assays

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105275212

A rapid in vitro assay for HIV DNA integration

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105275212

Integration complexes derived from HIV vectors for rapid assays in vitro

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105275212

Rapid microtiter assays for poxvirus topoisomerase, mammalian type IB topoisomerase and HIV-1 integrase: application to inhibitor isolation

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105275212

A novel assay for the DNA strand-transfer reaction of HIV-1 integrase

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105275212

Structure of the HIV-1 integrase catalytic domain complexed with an inhibitor: a platform for antiviral drug design

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105275212

Interacting residues in the extracellular region of the common beta subunit of the human granulocyte-macrophage colony-stimulating factor, interleukin (IL)-3, and IL-5 receptors involved in constitutive activation.

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105275212

Structural genomics of the Thermotoga maritima proteome implemented in a high-throughput structure determination pipeline

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105275212

A Simple Statistical Parameter for Use in Evaluation and Validation of High Throughput Screening Assays

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105275212

Efficient human immunodeficiency virus-based vector transduction of unstimulated human mobilized peripheral blood CD34+ cells in the SCID-hu Thy/Liv model of human T cell lymphopoiesis

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105275212

Efficient concerted integration by recombinant human immunodeficiency virus type 1 integrase without cellular or viral cofactors

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105275212

Human immunodeficiency virus type-1 integrase containing a glycine to serine mutation at position 140 is attenuated for catalysis and resistant to integrase inhibitors

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105275212

Metal-dependent inhibition of HIV-1 integrase by beta-diketo acids and resistance of the soluble double-mutant (F185K/C280S).

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105275212

Antiretroviral agents as inhibitors of both human immunodeficiency virus type 1 integrase and protease.

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105275212

HIV-1 integrase pharmacophore model derived from diverse classes of inhibitors.

21 January 2018

1 reference

https://api.crossref.org/works/10.1177%2F1087057105275212

21 January 2018

Identifiers

DOI

10.1177/1087057105275212

1 reference

24 July 2017

1 reference