(Q33536202)

English

Implementation of a fluorescence-based screening assay identifies histamine H3 receptor antagonists clobenpropit and iodophenpropit as subunit-selective N-methyl-D-aspartate receptor antagonists

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scholarly article

1 reference

Europe PubMed Central

PubMed publication ID

27 July 2017

Implementation of a fluorescence-based screening assay identifies histamine H3 receptor antagonists clobenpropit and iodophenpropit as subunit-selective N-methyl-D-aspartate receptor antagonists (English)

1 reference

Europe PubMed Central

PubMed publication ID

27 July 2017

1 reference

ChEBI release 2020-05-28

Hans Bräuner-Osborne

18

object named as

Hans Bräuner-Osborne

0 references

object named as

Kevin K Ogden

9

0 references

Kasper B. Hansen

object named as

Kasper B Hansen

1

0 references

12

object named as

Iestyn Lewis

1 reference

Europe PubMed Central

PubMed publication ID

27 July 2017

8

object named as

Trine Kvist

1 reference

Europe PubMed Central

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27 July 2017

Stephen Traynelis

19

object named as

Stephen F Traynelis

1 reference

Europe PubMed Central

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27 July 2017

author name string

Praseeda Mullasseril

2

1 reference

Europe PubMed Central

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27 July 2017

Sara Dawit

3

1 reference

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27 July 2017

Natalie L Kurtkaya

4

1 reference

Europe PubMed Central

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27 July 2017

Hongjie Yuan

5

1 reference

Europe PubMed Central

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27 July 2017

Katie M Vance

6

1 reference

Europe PubMed Central

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27 July 2017

Anna G Orr

7

1 reference

Europe PubMed Central

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27 July 2017

Phuong Le

10

1 reference

Europe PubMed Central

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27 July 2017

Kimberly M Vellano

11

1 reference

Europe PubMed Central

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27 July 2017

Serdar Kurtkaya

13

1 reference

Europe PubMed Central

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27 July 2017

Yuhong Du

14

1 reference

Europe PubMed Central

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27 July 2017

Min Qui

15

1 reference

Europe PubMed Central

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27 July 2017

T J Murphy

16

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Europe PubMed Central

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27 July 2017

James P Snyder

17

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27 July 2017

language of work or name

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publication date

2 March 2010

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Europe PubMed Central

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27 July 2017

Journal of Pharmacology and Experimental Therapeutics

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Europe PubMed Central

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27 July 2017

333

1 reference

Europe PubMed Central

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27 July 2017

3

1 reference

Europe PubMed Central

PubMed publication ID

27 July 2017

650-662

1 reference

Europe PubMed Central

PubMed publication ID

27 July 2017

Glutamate receptor ion channels: structure, regulation, and function

1 reference

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Control of NMDA receptor function by the NR2 subunit amino-terminal domain

1 reference

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1 reference

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Synthesis, structural activity-relationships, and biological evaluation of novel amide-based allosteric binding site antagonists in NR1A/NR2B N-methyl-D-aspartate receptors

1 reference

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An innovative design to establish proof of concept of the antidepressant effects of the NR2B subunit selective N-methyl-D-aspartate antagonist, CP-101,606, in patients with treatment-refractory major depressive disorder.

1 reference

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21 June 2018

Histamine in the nervous system

1 reference

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Pharmacological characterization of ligands at recombinant NMDA receptor subtypes by electrophysiological recordings and intracellular calcium measurements

1 reference

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Pharmacological characterization of JNJ-28583867, a histamine H(3) receptor antagonist and serotonin reuptake inhibitor

1 reference

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21 June 2018

The histamine H3 receptor antagonist clobenpropit enhances GABA release to protect against NMDA-induced excitotoxicity through the cAMP/protein kinase A pathway in cultured cortical neurons

1 reference

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21 June 2018

Subunit-specific mechanisms and proton sensitivity of NMDA receptor channel block.

1 reference

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Detection of multiple H3 receptor affinity states utilizing [3H]A-349821, a novel, selective, non-imidazole histamine H3 receptor inverse agonist radioligand

1 reference

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The role of N-methyl-D-asparate receptors in neurogenesis

1 reference

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21 June 2018

Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist

1 reference

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Potential energy functions for atomic-level simulations of water and organic and biomolecular systems

1 reference

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N-methyl-D-aspartate receptor subtypes: multiple roles in excitotoxicity and neurological disease

1 reference

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21 June 2018

Long-term potentiation: outstanding questions and attempted synthesis

1 reference

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21 June 2018

Channel blockers acting at N-methyl-D-aspartate receptors: differential effects of mutations in the vestibule and ion channel pore.

1 reference

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21 June 2018

Cloning and pharmacological characterization of a fourth histamine receptor (H(4)) expressed in bone marrow

1 reference

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Ligands for glutamate receptors: design and therapeutic prospects

1 reference

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21 June 2018

A Simple Statistical Parameter for Use in Evaluation and Validation of High Throughput Screening Assays

1 reference

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21 June 2018

Control of voltage-independent zinc inhibition of NMDA receptors by the NR1 subunit.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2879924

21 June 2018

Functional and pharmacological differences between recombinant N-methyl-D-aspartate receptors

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2879924

21 June 2018

Evaluation of the receptor selectivity of the H3 receptor antagonists, iodophenpropit and thioperamide: an interaction with the 5-HT3 receptor revealed

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2879924

21 June 2018

Histamine potentiates N-methyl-D-aspartate receptors by interacting with an allosteric site distinct from the polyamine binding site

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2879924

31 October 2018

Structural basis of NR2B-selective antagonist recognition by N-methyl-D-aspartate receptors.

1 reference

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Different effects of two N-methyl-D-aspartate receptor antagonists on seizures, spontaneous behavior, and motor performance in immature rats

1 reference

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Peripheral tackykinin and excitatory amino acid receptors mediate hyperalgesia induced by Phoneutria nigriventer venom

1 reference

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Mapping the binding site of the neuroprotectant ifenprodil on NMDA receptors.

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1 reference

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31 October 2018

Enhancement by histamine of NMDA-mediated synaptic transmission in the hippocampus

1 reference

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31 October 2018

Ifenprodil prevents glutamate cytotoxicity via polyamine modulatory sites of N-methyl-D-aspartate receptors in cultured cortical neurons.

1 reference

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31 October 2018

Subunit-specific potentiation of recombinant N-methyl-D-aspartate receptors by histamine.

1 reference

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Optimal expression of cloned NMDAR1/NMDAR2A heteromeric glutamate receptors: a biochemical characterization

1 reference

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Effect of clobenpropit, a centrally acting histamine H3-receptor antagonist, on electroshock- and pentylenetetrazol-induced seizures in mice

1 reference

https://pubmed.ncbi.nlm.nih.gov/20197375

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Histamine potentiates N-methyl-D-aspartate responses in acutely isolated hippocampal neurons

1 reference

https://pubmed.ncbi.nlm.nih.gov/20197375

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Inhibition and induction of cytochrome P450 and the clinical implications

1 reference

https://pubmed.ncbi.nlm.nih.gov/20197375

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identifiers

10.1124/JPET.110.166256

1 reference

Europe PubMed Central

PubMed publication ID

27 July 2017

PMC publication ID

1 reference

Europe PubMed Central

PubMed publication ID

27 July 2017

PubMed publication ID

1 reference

Europe PubMed Central

PubMed publication ID

27 July 2017

ResearchGate publication ID

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