(Q33547071)

28 July 2017

title

Prospective validation of a comprehensive in silico hERG model and its applications to commercial compound and drug databases (English)

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28 July 2017

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Adriaan P Ijzerman

4

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Andreas Bender

5

object named as

Andreas Bender

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28 July 2017

author name string

Munikumar R Doddareddy

1

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28 July 2017

Elisabeth C Klaasse

2

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28 July 2017

Shagufta

3

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28 July 2017

publication date

1 May 2010

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28 July 2017

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28 July 2017

volume

5

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28 July 2017

issue

5

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28 July 2017

page(s)

716-729

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Modeling promiscuity based on in vitro safety pharmacology profiling data

28 July 2017

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21 January 2018

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21 January 2018

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21 January 2018

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21 January 2018

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Clemastine, a conventional antihistamine, is a high potency inhibitor of the HERG K+ channel

21 January 2018

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Flunarizine is a highly potent inhibitor of cardiac hERG potassium current

21 January 2018

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Potent inhibition of human cardiac potassium (HERG) channels by the anti-estrogen agent clomiphene-without QT interval prolongation

21 January 2018

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The phenothiazine drugs inhibit hERG potassium channels

21 January 2018

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hERG classification model based on a combination of support vector machine method and GRIND descriptors

21 January 2018

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Prediction of Hydrophobic (Lipophilic) Properties of Small Organic Molecules Using Fragmental Methods: An Analysis of ALOGP and CLOGP Methods

21 January 2018

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Molecular determinants of HERG channel block.

21 January 2018

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.201000024

Structural determinants of HERG channel block by clofilium and ibutilide.

21 January 2018

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.201000024

Validation of a [3H]astemizole binding assay in HEK293 cells expressing HERG K+ channels

21 January 2018

1 reference

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A high-throughput HERG potassium channel function assay: an old assay with a new look

21 January 2018

1 reference

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Identifiers

DOI

10.1002/CMDC.201000024

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28 July 2017

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