(Q33589171)

28 July 2017

title

Identification of broad-based HIV-1 protease inhibitors from combinatorial libraries (English)

1 reference

28 July 2017

Max W Chang

1

0 references

Sukwon Hong

object named as

Sukwon Hong

6

0 references

author name string

Michael J Giffin

2

1 reference

28 July 2017

Rolf Muller

3

1 reference

28 July 2017

Jeremiah Savage

4

1 reference

28 July 2017

Ying C Lin

5

1 reference

28 July 2017

Wei Jin

7

1 reference

28 July 2017

Landon R Whitby

8

1 reference

28 July 2017

John H Elder

9

1 reference

28 July 2017

Dale L Boger

10

1 reference

28 July 2017

Bruce E Torbett

11

1 reference

28 July 2017

language of work or name

English

0 references

publication date

1 August 2010

1 reference

28 July 2017

number of pages

6

1 reference

based on heuristic

inferred from page(s)

published in

Biochemical Journal

1 reference

28 July 2017

volume

429

1 reference

28 July 2017

issue

3

1 reference

28 July 2017

page(s)

527-532

1 reference

Fragment-Based Screen against HIV Protease

28 July 2017

cites work

1 reference

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21 June 2018

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Drug resistance mutations for surveillance of transmitted HIV-1 drug-resistance: 2009 update

21 June 2018

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Discovery of inhibitors of aberrant gene transcription from Libraries of DNA binding molecules: inhibition of LEF-1-mediated gene transcription and oncogenic transformation

21 June 2018

1 reference

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Viral protease inhibitors

21 June 2018

1 reference

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A copper(I)-catalyzed 1,2,3-triazole azide-alkyne click compound is a potent inhibitor of a multidrug-resistant HIV-1 protease variant

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3084599

Solution kinetics measurements suggest HIV-1 protease has two binding sites for darunavir and amprenavir

21 June 2018

1 reference

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Targeting the open-flap conformation of HIV-1 protease with pyrrolidine-based inhibitors

21 June 2018

1 reference

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Unique small molecule entry inhibitors of hemorrhagic fever arenaviruses

21 June 2018

1 reference

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A poke in the eye: inhibiting HIV-1 protease through its flap-recognition pocket

21 June 2018

1 reference

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HIV-1 protease folding and the design of drugs which do not create resistance

21 June 2018

1 reference

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An in vitro and in vivo disconnect uncovered through high-throughput identification of botulinum neurotoxin A antagonists.

21 June 2018

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High-throughput assays for promiscuous inhibitors.

21 June 2018

1 reference

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Beta-lactam compounds as apparently uncompetitive inhibitors of HIV-1 protease

21 June 2018

1 reference

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Development of low molecular weight HIV-1 protease dimerization inhibitors

21 June 2018

1 reference

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HIV-1 protease molecular dynamics of a wild-type and of the V82F/I84V mutant: possible contributions to drug resistance and a potential new target site for drugs

21 June 2018

1 reference

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Solution‐Phase Combinatorial Libraries: Modulating Cellular Signaling by Targeting Protein–Protein or Protein–DNA Interactions

21 June 2018

1 reference

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21 June 2018

1 reference

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A Common Mechanism Underlying Promiscuous Inhibitors from Virtual and High-Throughput Screening

21 June 2018

1 reference

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Viral evolution in response to the broad-based retroviral protease inhibitor TL-3.

21 June 2018

1 reference

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Polyoxometalate HIV-1 protease inhibitors. A new mode of protease inhibition.

21 June 2018

1 reference

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Analysis of the interactions between an enzyme and multiple inhibitors using combination plots

21 June 2018

1 reference

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A solution-phase strategy for the synthesis of chemical libraries containing small organic molecules: a universal and dipeptide mimetic template

21 June 2018

1 reference

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Subsite preferences of retroviral proteinases

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3084599

Human immunodeficiency virus has an aspartic-type protease that can be inhibited by pepstatin A

21 June 2018

1 reference

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Stability and activity of human immunodeficiency virus protease: comparison of the natural dimer with a homologous, single-chain tethered dimer

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3084599

Crystallographic analysis of a complex between human immunodeficiency virus type 1 protease and acetyl-pepstatin at 2.0-A resolution

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3084599

A simple, continuous fluorometric assay for HIV protease

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3084599

Switching between allosteric and dimerization inhibition of HIV-1 protease

21 June 2018

1 reference

Crossref

https://api.crossref.org/works/10.1042%2FBJ20091645

Automatic generation of 3D-atomic coordinates for organic molecules

21 January 2018

1 reference

Crossref

https://api.crossref.org/works/10.1042%2FBJ20091645

Analysis of the combined effect of two linear inhibitors on a single enzyme

21 January 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3084599

Synergistic binding of inhibitors to the protease from HIV type 1.

31 October 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3084599

STUDIES ON LIVER ALCOHOL HYDROGENASE COMPLEXES. 3. MULTIPLE INHIBITION KINETICS IN THE PRESENCE OF TWO COMPETITIVE INHIBITORS

31 October 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/20507280

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Evaluation of enzyme inhibitors in drug discovery. A guide for medicinal chemists and pharmacologists

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/20507280

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1042/BJ20091645

1 reference

28 July 2017

1 reference

28 July 2017

1 reference