(Q33598591)

28 July 2017

title

Cyclopropyl Carboxamides: A New Oral Antimalarial Series Derived from the Tres Cantos Anti-Malarial Set (TCAMS). (English)

1 reference

28 July 2017

0 references

0 references

Lourdes Rueda

1

1 reference

28 July 2017

Isabel Castellote

2

1 reference

28 July 2017

Julia Castro-Pichel

3

1 reference

28 July 2017

Maria J Chaparro

4

1 reference

28 July 2017

Juan Carlos de la Rosa

5

1 reference

28 July 2017

Adolfo Garcia-Perez

6

1 reference

28 July 2017

Mariola Gordo

7

1 reference

28 July 2017

Maria Belen Jimenez-Diaz

8

1 reference

28 July 2017

Albane Kessler

9

1 reference

28 July 2017

Simon J F Macdonald

10

1 reference

28 July 2017

Maria Santos Martinez

11

1 reference

28 July 2017

Laura M Sanz

12

1 reference

28 July 2017

Francisco Javier Gamo

13

1 reference

28 July 2017

Esther Fernandez

14

1 reference

28 July 2017

publication date

29 August 2011

1 reference

ACS Medicinal Chemistry Letters

28 July 2017

published in

1 reference

28 July 2017

volume

2

1 reference

28 July 2017

issue

11

1 reference

28 July 2017

page(s)

840-844

1 reference

An Invitation to Open Innovation in Malaria Drug Discovery: 47 Quality Starting Points from the TCAMS

28 July 2017

cites work

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4017974

β-Branched acyclic nucleoside analogues as inhibitors of Plasmodium falciparum dUTPase

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4017974

Evaluation of Diarylureas for Activity Against Plasmodium falciparum.

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4017974

Synthesis and structure-activity relationships of novel benzoxaboroles as a new class of antimalarial agents

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4017974

Road towards new antimalarials - overview of the strategies and their chemical progress

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4017974

Endoperoxide carbonyl falcipain 2/3 inhibitor hybrids: toward combination chemotherapy of malaria through a single chemical entity

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4017974

Discovery of potent small-molecule inhibitors of multidrug-resistant Plasmodium falciparum using a novel miniaturized high-throughput luciferase-based assay

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4017974

Chemical genetics of Plasmodium falciparum

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4017974

Thousands of chemical starting points for antimalarial lead identification

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4017974

New medicines to improve control and contribute to the eradication of malaria

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4017974

Improved murine model of malaria using Plasmodium falciparum competent strains and non-myelodepleted NOD-scid IL2Rgammanull mice engrafted with human erythrocytes

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4017974

In silico activity profiling reveals the mechanism of action of antimalarials discovered in a high-throughput screen

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4017974

A murine model of falciparum-malaria by in vivo selection of competent strains in non-myelodepleted mice engrafted with human erythrocytes

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4017974

Antimalarial drug discovery: efficacy models for compound screening

21 June 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4017974

Chromatographic Hydrophobicity Index by Fast-Gradient RP-HPLC: A High-Throughput Alternative to log P/log D

21 June 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/24900273

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1021/ML2001517

1 reference

28 July 2017

1 reference

28 July 2017

1 reference