(Q33992426)

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Design, synthesis, and biological evaluation of resveratrol analogues as aromatase and quinone reductase 2 inhibitors for chemoprevention of cancer.

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20558073%20AND%20SRC:MED&resulttype=core&format=json

5 February 2020

Design, synthesis, and biological evaluation of resveratrol analogues as aromatase and quinone reductase 2 inhibitors for chemoprevention of cancer (English)

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Europe PubMed Central

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20558073%20AND%20SRC:MED&resulttype=core&format=json

5 February 2020

Andrew D. Mesecar

6

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5 February 2020

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John M Pezzuto

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5 February 2020

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Bin Sun

1

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5 February 2020

Juma Hoshino

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5 February 2020

Katie Jermihov

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5 February 2020

Laura Marler

4

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5 February 2020

Mark Cushman

7

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5 February 2020

language of work or name

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publication date

24 May 2010

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5 February 2020

Bioorganic & Medicinal Chemistry

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5 February 2020

18

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5 February 2020

14

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5 February 2020

5352-5366

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Europe PubMed Central

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5 February 2020

Synthesis and multidrug resistance reversal activity of dihydroptychantol A and its novel derivatives

1 reference

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Separation of alpha-glucosidase-inhibitory and liver X receptor-antagonistic activities of phenethylphenyl phthalimide analogs and generation of LXRalpha-selective antagonists.

1 reference

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Synthesis, structural characterisation and biological evaluation of fluorinated analogues of resveratrol

1 reference

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5 July 2018

Synthesis of Casimiroin and Optimization of Its Quinone Reductase 2 and Aromatase Inhibitory Activities

1 reference

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5 July 2018

Structural basis for androgen specificity and oestrogen synthesis in human aromatase

1 reference

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Second-generation DBFOX ligands for the synthesis of beta-substituted alpha-amino acids via enantioselective radical conjugate additions

1 reference

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Synthesis and biological evaluation of a library of resveratrol analogues as inhibitors of COX-1, COX-2 and NF-kappaB.

1 reference

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5 July 2018

Cancer statistics, 2008

1 reference

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Kinetic, thermodynamic and X-ray structural insights into the interaction of melatonin and analogues with quinone reductase 2

1 reference

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Reduction of mitomycin C is catalysed by human recombinant NRH:quinone oxidoreductase 2 using reduced nicotinamide adenine dinucleotide as an electron donating co-factor

1 reference

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5 July 2018

Therapeutic potential of resveratrol: the in vivo evidence

1 reference

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5 July 2018

The red wine polyphenol resveratrol displays bilevel inhibition on aromatase in breast cancer cells

1 reference

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5 July 2018

Molecular tools to study melatonin pathways and actions.

1 reference

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Coot: model-building tools for molecular graphics

1 reference

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5 July 2018

Crystal structure of quinone reductase 2 in complex with resveratrol

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2903642

5 July 2018

Refinement of macromolecular structures by the maximum-likelihood method

1 reference

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5 July 2018

The CCP4 suite: programs for protein crystallography

1 reference

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5 July 2018

Likelihood-enhanced fast rotation functions

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2903642

5 July 2018

Biological rationale for endocrine therapy in breast cancer

1 reference

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5 July 2018

Aromatase inhibitors: mechanism of action and role in the treatment of breast cancer

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2903642

5 July 2018

Improved protein-ligand docking using GOLD

1 reference

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5 July 2018

The evolving role of aromatase inhibitors in breast cancer

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2903642

5 July 2018

Prevention and treatment of breast cancer by suppressing aromatase activity and expression

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2903642

5 July 2018

Nonsteroidal aromatase inhibitors: recent advances

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2903642

5 July 2018

Aromatase inhibitors continue their ATAC on tamoxifen

1 reference

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5 July 2018

Molecular pharmacology of aromatase and its regulation by endogenous and exogenous agents

1 reference

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Selective estrogen receptor modulators (SERMS) and their roles in breast cancer prevention

1 reference

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Molecular perspectives on selective estrogen receptor modulators (SERMs): progress in understanding their tissue-specific agonist and antagonist actions

1 reference

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5 July 2018

Bioactivation of 5-(aziridin-1-yl)-2,4-dinitrobenzamide (CB 1954) by human NAD(P)H quinone oxidoreductase 2: a novel co-substrate-mediated antitumor prodrug therapy

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2903642

5 July 2018

Resveratrol, a phytoestrogen found in red wine. A possible explanation for the conundrum of the 'French paradox'?

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2903642

5 July 2018

Development and validation of a genetic algorithm for flexible docking

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2903642

5 July 2018

Recent developments in aromatase inhibition as a potential treatment for oestrogen-dependent breast cancer.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=2903642

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Synthesis and evaluation of stilbene and dihydrostilbene derivatives as potential anticancer agents that inhibit tubulin polymerization

1 reference

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Nazarov cyclizations of an allenyl vinyl ketone with interception of the oxyallyl cation intermediate for the formation of carbon-carbon bonds.

1 reference

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29 October 2018

trans-Directing ability of the amide group: enabling the enantiocontrol in the synthesis of 1,1-dicarboxy cyclopropanes. Reaction development, scope, and synthetic applications.

1 reference

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Cytotoxic constituents of Soymida febrifuga from Myanmar.

1 reference

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Fast three dimensional pharmacophore virtual screening of new potent non-steroid aromatase inhibitors.

1 reference

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The design, synthesis, and anti-tumor mechanism study of N-phosphoryl amino acid modified resveratrol analogues

1 reference

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Algicidal activity of stilbene analogues

1 reference

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1 reference

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1 reference

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1 reference

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12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Aromatase inhibitors in breast cancer therapy

1 reference

https://pubmed.ncbi.nlm.nih.gov/20558073

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Synthesis of hydroxystilbenes and their derivatives via Heck reaction

1 reference

https://pubmed.ncbi.nlm.nih.gov/20558073

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Synthesis and Biological Evaluation of (±)-Abyssinone II and Its Analogues as Aromatase Inhibitors for Chemoprevention of Breast Cancer

1 reference

https://pubmed.ncbi.nlm.nih.gov/20558073

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Imidazolylmethylbenzophenones as highly potent aromatase inhibitors

1 reference

https://pubmed.ncbi.nlm.nih.gov/20558073

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Processing of X-ray diffraction data collected in oscillation mode

1 reference

https://pubmed.ncbi.nlm.nih.gov/20558073

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identifiers

10.1016/J.BMC.2010.05.042

1 reference

Europe PubMed Central

PMC publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20558073%20AND%20SRC:MED&resulttype=core&format=json

5 February 2020

PMC publication ID

1 reference

Europe PubMed Central

PMC publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20558073%20AND%20SRC:MED&resulttype=core&format=json

5 February 2020

PubMed publication ID

1 reference

Europe PubMed Central

PMC publication ID

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20558073%20AND%20SRC:MED&resulttype=core&format=json

5 February 2020

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