(Q34376764)

1 August 2017

title

Identification of novel functionally selective κ-opioid receptor scaffolds (English)

1 reference

1 August 2017

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Marie-Laure Rives

3

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Peter J. Brown

object named as

Peter J Brown

6

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Jordan Zjawiony

object named as

Jordan K Zjawiony

9

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Jonathan Javitch

object named as

Jonathan A Javitch

8

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author name string

Kate L White

1

1 reference

1 August 2017

Alex P Scopton

2

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1 August 2017

Ruslan V Bikbulatov

4

1 reference

1 August 2017

Prabhakar R Polepally

5

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1 August 2017

Terrance Kenakin

7

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1 August 2017

Bryan L Roth

10

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1 August 2017

publication date

10 October 2013

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1 August 2017

published in

Molecular Pharmacology

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1 August 2017

volume

85

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1 August 2017

issue

1

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1 August 2017

page(s)

83-90

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Functional selectivity of 6'-guanidinonaltrindole (6'-GNTI) at κ-opioid receptors in striatal neurons

1 August 2017

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6 July 2018

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6'-Guanidinonaltrindole (6'-GNTI) is a G protein-biased κ-opioid receptor agonist that inhibits arrestin recruitment

6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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Activation of the kappa opioid receptor in the dorsal raphe nucleus mediates the aversive effects of stress and reinstates drug seeking

6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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Galpha-subunits differentially alter the conformation and agonist affinity of kappa-opioid receptors

6 July 2018

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The dysphoric component of stress is encoded by activation of the dynorphin kappa-opioid system

6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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The interaction of a constitutively active arrestin with the arrestin-insensitive 5-HT(2A) receptor induces agonist-independent internalization

6 July 2018

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6 July 2018

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6 July 2018

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Salvinorin A: a potent naturally occurring nonnitrogenous kappa opioid selective agonist

6 July 2018

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The dynamin-dependent, arrestin-independent internalization of 5-hydroxytryptamine 2A (5-HT2A) serotonin receptors reveals differential sorting of arrestins and 5-HT2A receptors during endocytosis

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3868907

Confirmation of primary active substances from high throughput screening of chemical and biological populations: a statistical approach and practical considerations

6 July 2018

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Agonist-induced phosphorylation of the kappa-opioid receptor

6 July 2018

1 reference

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Agonist-receptor efficacy. II. Agonist trafficking of receptor signals

6 July 2018

1 reference

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Operational models of pharmacological agonism.

6 July 2018

1 reference

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Psychotomimesis mediated by kappa opiate receptors

6 July 2018

1 reference

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Kappa-opioid receptors and analgesia

6 July 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3868907

Conformational ensembles in GPCR activation

6 July 2018

1 reference

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Psychotomimetic effects of kappa opioid receptor agonists

27 October 2018

1 reference

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Effects of the long-lasting kappa opioid 2-(3,4-dichlorophenyl)-N-methyl-N-[(1S)-1-(3-isothiocyanatophenyl)-2-(1-pyrrolidinyl) ethyl] acetamide in a drug discrimination and warm water tail-withdrawal procedure

27 October 2018

1 reference

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[(11)C]-GR89696, a potent kappa opiate receptor radioligand; in vivo binding of the R and S enantiomers

27 October 2018

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27 October 2018

Identifiers

DOI

10.1124/MOL.113.089649

1 reference

1 August 2017

1 reference

1 August 2017

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