(Q34395031)

24380043

1 August 2017

title

Design, synthesis, and evaluation of hydroxamic acid-based molecular probes for in vivo imaging of histone deacetylase (HDAC) in brain (English)

1 reference

1 August 2017

0 references

Changning Wang

1

1 reference

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31 May 2020

Thomas E Eessalu

2

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31 May 2020

Charles H Mitch

4

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31 May 2020

Florence F Wagner

5

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31 May 2020

Ramesh Neelamegam

7

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31 May 2020

Frederick A Schroeder

8

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31 May 2020

Edward B Holson

9

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31 May 2020

Stephen J Haggarty

10

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31 May 2020

Jacob M Hooker

11

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31 May 2020

publication date

15 December 2013

1 reference

24380043

American journal of nuclear medicine and molecular imaging

1 August 2017

published in

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24380043%20AND%20SRC:MED&resulttype=core&format=json

31 May 2020

volume

4

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31 May 2020

issue

1

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31 May 2020

page(s)

29-38

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A selective HDAC 1/2 inhibitor modulates chromatin and gene expression in brain and alters mouse behavior in two mood-related tests

31 May 2020

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6 July 2018

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6 July 2018

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6 July 2018

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Class I HDAC imaging using [ (3)H]CI-994 autoradiography

6 July 2018

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HDAC3-selective inhibitor enhances extinction of cocaine-seeking behavior in a persistent manner

6 July 2018

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6 July 2018

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6 July 2018

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HDAC6 regulates glucocorticoid receptor signaling in serotonin pathways with critical impact on stress resilience

6 July 2018

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6 July 2018

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In vivo PET imaging of histone deacetylases by 18F-suberoylanilide hydroxamic acid (18F-SAHA).

6 July 2018

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Histone deacetylase inhibitor, MS-275, exhibits poor brain penetration: PK studies of [C]MS-275 using Positron Emission Tomography

6 July 2018

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Inhibition of specific HDACs and sirtuins suppresses pathogenesis in a Drosophila model of Huntington's disease.

6 July 2018

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A novel histone deacetylase 8 (HDAC8)-specific inhibitor PCI-34051 induces apoptosis in T-cell lymphomas

6 July 2018

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Epigenetic targets of HDAC inhibition in neurodegenerative and psychiatric disorders.

6 July 2018

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Dimethyl sulfoxide to vorinostat: development of this histone deacetylase inhibitor as an anticancer drug

6 July 2018

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Anticancer activities of histone deacetylase inhibitors

6 July 2018

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A phase I study of intravenous LBH589, a novel cinnamic hydroxamic acid analogue histone deacetylase inhibitor, in patients with refractory hematologic malignancies

6 July 2018

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6 July 2018

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Remodeling chromatin and stress resistance in the central nervous system: histone deacetylase inhibitors as novel and broadly effective neuroprotective agents.

6 July 2018

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Histone deacetylation in epigenetics: an attractive target for anticancer therapy

6 July 2018

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Trichostatin A-like hydroxamate histone deacetylase inhibitors as therapeutic agents: toxicological point of view

6 July 2018

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Pharmacodynamic response and inhibition of growth of human tumor xenografts by the novel histone deacetylase inhibitor PXD101.

6 July 2018

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Modulation of histone acetylation by [4-(acetylamino)-N-(2-amino-phenyl) benzamide] in HCT-8 colon carcinoma.

6 July 2018

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Histone deacetylases (HDACs): characterization of the classical HDAC family

6 July 2018

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Histone deacetylase inhibitors arrest polyglutamine-dependent neurodegeneration in Drosophila

6 July 2018

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Histone deacetylase is a direct target of valproic acid, a potent anticonvulsant, mood stabilizer, and teratogen

6 July 2018

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6 July 2018

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6 July 2018

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6 July 2018

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27 October 2018

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27 October 2018

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Histone deacetylase inhibitors exhibit anti-inflammatory and neuroprotective effects in a rat permanent ischemic model of stroke: multiple mechanisms of action.

27 October 2018

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Pharmacological inhibition of histone deacetylases by suberoylanilide hydroxamic acid specifically alters gene expression and reduces ischemic injury in the mouse brain

27 October 2018

1 reference

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Differential contributions of Caenorhabditis elegans histone deacetylases to huntingtin polyglutamine toxicity.

27 October 2018

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Use of LC/MS to assess brain tracer distribution in preclinical, in vivo receptor occupancy studies: dopamine D2, serotonin 2A and NK-1 receptors as examples

27 October 2018

1 reference

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Sodium phenylbutyrate prolongs survival and regulates expression of anti-apoptotic genes in transgenic amyotrophic lateral sclerosis mice

27 October 2018

1 reference

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Valproic acid reduces brain damage induced by transient focal cerebral ischemia in rats: potential roles of histone deacetylase inhibition and heat shock protein induction

27 October 2018

1 reference

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Heterocyclic ketones as inhibitors of histone deacetylase.

27 October 2018

1 reference

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Trifluoromethyl ketones as inhibitors of histone deacetylase

27 October 2018

1 reference

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27 October 2018

Identifiers

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24380043%20AND%20SRC:MED&resulttype=core&format=json

31 May 2020

24380043

1 reference