(Q34583185)

English

Solid-phase peptide head-to-side chain cyclodimerization: Discovery of C2-symmetric cyclic lactam hybrid α-melanocyte-stimulating hormone (MSH)/agouti-signaling protein (ASIP) analogues with potent activities at the human melanocortin receptors

scientific article published on August 3, 2010

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3 August 2017

Solid-phase peptide head-to-side chain cyclodimerization: discovery of C(2)-symmetric cyclic lactam hybrid α-melanocyte-stimulating hormone (MSH)/agouti-signaling protein (ASIP) analogues with potent activities at the human melanocortin receptors (English)

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PubMed publication ID

3 August 2017

Solid-phase peptide head-to-side chain cyclodimerization: Discovery of C2-symmetric cyclic lactam hybrid α-melanocyte-stimulating hormone (MSH)/agouti-signaling protein (ASIP) analogues with potent activities at the human melanocortin receptors (English)

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10.1016/J.PEPTIDES.2010.06.026

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17 June 2024

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Minying Cai

2

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3 August 2017

Zhihua Liu

4

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3 August 2017

Josef Vagner

6

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3 August 2017

Dev Trivedi

7

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3 August 2017

Alexander V. Mayorov

1

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Erin S. Palmer

3

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James P. Cain

5

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Victor J. Hruby

8

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3 August 2010

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3 August 2017

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10.1016/J.PEPTIDES.2010.06.026

https://api.crossref.org/works/10.1016/J.PEPTIDES.2010.06.026

17 June 2024

https://api.elsevier.com/content/article/PII:S0196978110002706?httpAccept=text/plain

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10.1016/J.PEPTIDES.2010.06.026

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17 June 2024

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3 August 2017

31

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3 August 2017

10

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3 August 2017

1894-1905

1 reference

Europe PubMed Central

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3 August 2017

pA, a new scale for the measurement of drug antagonism

1 reference

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1 reference

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1 reference

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Structure-activity relationships of cyclic lactam analogues of alpha-melanocyte-stimulating hormone (alpha-MSH) targeting the human melanocortin-3 receptor

1 reference

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1 reference

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Melanocortin receptors, melanotropic peptides and penile erection

1 reference

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1 reference

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1 reference

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Design, synthesis, and biological evaluation of new cyclic melanotropin peptide analogues selective for the human melanocortin-4 receptor

1 reference

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1 reference

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Design, synthesis, and biological evaluation of a new class of small molecule peptide mimetics targeting the melanocortin receptors

1 reference

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1 reference

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Effects of macrocycle size and rigidity on melanocortin receptor-1 and -5 selectivity in cyclic lactam alpha-melanocyte-stimulating hormone analogs

1 reference

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Development of cyclic gamma-MSH analogues with selective hMC3R agonist and hMC3R/hMC5R antagonist activities

1 reference

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Targeting melanocortin receptors as potential novel therapeutics

1 reference

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The melanocortin system and energy balance

1 reference

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Melanocortin peptide therapeutics: historical milestones, clinical studies and commercialization

1 reference

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Interactions between gut peptides and the central melanocortin system in the regulation of energy homeostasis

1 reference

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The regulation of food intake by selective stimulation of the type 3 melanocortin receptor (MC3R).

1 reference

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1 reference

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A review of melanocortin receptor small molecule ligands

1 reference

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Design of cyclic and other templates for potent and selective peptide alpha-MSH analogues

1 reference

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Chimeras of the agouti-related protein: insights into agonist and antagonist selectivity of melanocortin receptors

1 reference

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Design of novel melanotropin agonists and antagonists with high potency and selectivity for human melanocortin receptors

1 reference

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Novel 3D pharmacophore of alpha-MSH/gamma-MSH hybrids leads to selective human MC1R and MC3R analogues

1 reference

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Over one hundred peptide-activated G protein-coupled receptors recognize ligands with turn structure.

1 reference

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Structures of the agouti signaling protein

1 reference

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Head-to-tail peptide cyclodimerization by copper-catalyzed azide-alkyne cycloaddition

1 reference

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Chimeric NDP-MSH and MTII melanocortin peptides with agouti-related protein (AGRP) Arg-Phe-Phe amino acids possess agonist melanocortin receptor activity

1 reference

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Melanocortin-5 receptor deficiency promotes defensive behavior in male mice

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Molecular interaction of Agouti protein and Agouti-related protein with human melanocortin receptors

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Agouti protein is an antagonist of the melanocyte-stimulating-hormone receptor

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Cyclic lactam alpha-melanotropin analogues of Ac-Nle4-cyclo[Asp5, D-Phe7,Lys10] alpha-melanocyte-stimulating hormone-(4-10)-NH2 with bulky aromatic amino acids at position 7 show high antagonist potency and selectivity at specific melanocortin recep

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half-Cys4,half-Cys10-alpha-Melanocyte-stimulating hormone: a cyclic alpha-melanotropin exhibiting superagonist biological activity

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Functional group contributions to drug-receptor interactions.

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Corticotropin inhibits food intake in rats.

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Inhibition of feeding by ACTH-(1-24): behavioral and pharmacological aspects

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Emerging approaches in the molecular design of receptor-selective peptide ligands: conformational, topographical and dynamic considerations

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Central administration of selective melanocortin 4 receptor antagonist HS014 prevents morphine tolerance and withdrawal hyperalgesia.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3041174

27 October 2018

Potent and selective agonists of human melanocortin receptor 5: cyclic analogues of alpha-melanocyte-stimulating hormone

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3041174

27 October 2018

Central receptors mediating the cardiovascular actions of melanocyte stimulating hormones

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3041174

27 October 2018

Synthesis and biological activity of the first cyclic biphalin analogues.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3041174

27 October 2018

De novo design, synthesis, and pharmacology of alpha-melanocyte stimulating hormone analogues derived from somatostatin by a hybrid approach

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3041174

27 October 2018

Inverse agonist activity of agouti and agouti-related protein.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3041174

27 October 2018

Exploring the stereostructural requirements of peptide ligands for the melanocortin receptors

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3041174

27 October 2018

Structure-activity studies of the melanocortin peptides: discovery of potent and selective affinity antagonists for the hMC3 and hMC4 receptors.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3041174

27 October 2018

Design and pharmacology of N-[(3R)-1,2,3,4-tetrahydroisoquinolinium- 3-ylcarbonyl]-(1R)-1-(4-chlorobenzyl)- 2-[4-cyclohexyl-4-(1H-1,2,4-triazol- 1-ylmethyl)piperidin-1-yl]-2-oxoethylamine (1), a potent, selective, melanocortin subtype-4 receptor ago

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3041174

27 October 2018

Melanocortin antagonists define two distinct pathways of cardiovascular control by alpha- and gamma-melanocyte-stimulating hormones.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3041174

27 October 2018

Total Solid-Phase Synthesis of Marine Cyclodepsipeptide IB-01212

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=3041174

9 December 2018

Conformational restrictions of biologically active peptides via amino acid side chain groups

1 reference

https://pubmed.ncbi.nlm.nih.gov/20688117

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Color test for detection of free terminal amino groups in the solid-phase synthesis of peptides

1 reference

https://pubmed.ncbi.nlm.nih.gov/20688117

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Proceedings of the 5th International Melanocortin Meeting. August 25-28, 2002. Sunriver, Oregon, USA

1 reference

https://pubmed.ncbi.nlm.nih.gov/20688117

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Ligand binding efficiency: trends, physical basis, and implications

1 reference

https://pubmed.ncbi.nlm.nih.gov/20688117

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

alpha-Melanotropin: the minimal active sequence in the frog skin bioassay

1 reference

https://pubmed.ncbi.nlm.nih.gov/20688117

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Gramicidin S and its use in the Treatment of Infected Wounds

27

1 reference

10.1016/J.PEPTIDES.2010.06.026

https://api.crossref.org/works/10.1016/J.PEPTIDES.2010.06.026

17 June 2024

Unequivocal synthesis and characterization of a parallel and an antiparallel bis-cystine peptide

80

1 reference

10.1016/J.PEPTIDES.2010.06.026

https://api.crossref.org/works/10.1016/J.PEPTIDES.2010.06.026

17 June 2024

Semianalytical treatment of solvation for molecular mechanics and dynamics

87

1 reference

10.1016/J.PEPTIDES.2010.06.026

https://api.crossref.org/works/10.1016/J.PEPTIDES.2010.06.026

17 June 2024

Use of Alloc-amino acids in solid-phase peptide synthesis. Tandem deprotection-coupling reactions using neutral conditions

88

1 reference

10.1016/J.PEPTIDES.2010.06.026

https://api.crossref.org/works/10.1016/J.PEPTIDES.2010.06.026

17 June 2024

Identifiers

10.1016/J.PEPTIDES.2010.06.026

1 reference

Europe PubMed Central

PubMed publication ID

3 August 2017

PMC publication ID

1 reference

Europe PubMed Central

PubMed publication ID

3 August 2017

PubMed publication ID

1 reference

Europe PubMed Central

PubMed publication ID

3 August 2017

ResearchGate publication ID

0 references

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