(Q35181966)

7 August 2017

title

High content screening of diverse compound libraries identifies potent modulators of tubulin dynamics (English)

1 reference

7 August 2017

David R Spring

6

0 references

author name string

Luca Laraia

1

1 reference

7 August 2017

Jamie Stokes

2

1 reference

7 August 2017

Amy Emery

3

1 reference

7 August 2017

Grahame J McKenzie

4

1 reference

7 August 2017

Ashok R Venkitaraman

5

1 reference

7 August 2017

publication date

24 February 2014

1 reference

ACS Medicinal Chemistry Letters

7 August 2017

published in

1 reference

7 August 2017

volume

5

1 reference

7 August 2017

issue

5

1 reference

7 August 2017

page(s)

598-603

1 reference

Biology-oriented synthesis of a tetrahydroisoquinoline-based compound collection targeting microtubule polymerization

7 August 2017

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28 July 2018

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28 July 2018

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Identification of Simple Compounds with Microtubule-Binding Activity That Inhibit Cancer Cell Growth with High Potency

28 July 2018

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28 July 2018

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28 July 2018

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28 July 2018

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28 July 2018

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28 July 2018

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28 July 2018

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Microtubules and resistance to tubulin-binding agents

28 July 2018

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Development of a benzopyran-containing androgen receptor antagonist to treat antiandrogen-resistant prostate cancer

28 July 2018

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Microtubule inhibitors: Differentiating tubulin-inhibiting agents based on mechanisms of action, clinical activity, and resistance

28 July 2018

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Direct coupling of catharanthine and vindoline to provide vinblastine: total synthesis of (+)- and ent-(-)-vinblastine

28 July 2018

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Paclitaxel from primary taxanes: a perspective on creative invention in organozirconium chemistry

28 July 2018

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28 July 2018

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28 July 2018

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28 July 2018

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28 July 2018

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A strategy for the diversity-oriented synthesis of macrocyclic scaffolds using multidimensional coupling

27 September 2018

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A natural product inspired tetrahydropyran collection yields mitosis modulators that synergistically target CSE1L and tubulin.

27 September 2018

1 reference

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UA62784 Is a cytotoxic inhibitor of microtubules, not CENP-E.

27 September 2018

1 reference

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Diversity-oriented synthesis of macrocyclic peptidomimetics

27 September 2018

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Anti-MRSA agent discovery using diversity-oriented synthesis

27 September 2018

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Structural basis for the regulation of tubulin by vinblastine

27 September 2018

1 reference

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Insight into tubulin regulation from a complex with colchicine and a stathmin-like domain.

27 September 2018

1 reference

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Total synthesis of (+)-discodermolide: a highly convergent fourth-generation approach

27 September 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/24900887

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1021/ML5000564

1 reference

7 August 2017

1 reference

7 August 2017

1 reference