(Q36742217)

English

Distinct roles of β-arrestin 1 and β-arrestin 2 in ORG27569-induced biased signaling and internalization of the cannabinoid receptor 1 (CB1).

scientific article published on 28 February 2013

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scholarly article

1 reference

Europe PubMed Central

PMC publication ID

16 August 2017

Distinct roles of β-arrestin 1 and β-arrestin 2 in ORG27569-induced biased signaling and internalization of the cannabinoid receptor 1 (CB1). (English)

1 reference

Europe PubMed Central

PMC publication ID

16 August 2017

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cannabinoid receptor

0 references

author name string

Kwang H Ahn

1

1 reference

Europe PubMed Central

PMC publication ID

16 August 2017

Mariam M Mahmoud

2

1 reference

Europe PubMed Central

PMC publication ID

16 August 2017

Joong-Youn Shim

3

1 reference

Europe PubMed Central

PMC publication ID

16 August 2017

Debra A Kendall

4

1 reference

Europe PubMed Central

PMC publication ID

16 August 2017

language of work or name

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publication date

28 February 2013

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Europe PubMed Central

PMC publication ID

16 August 2017

Journal of Biological Chemistry

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Europe PubMed Central

PMC publication ID

16 August 2017

288

1 reference

Europe PubMed Central

PMC publication ID

16 August 2017

14

1 reference

Europe PubMed Central

PMC publication ID

16 August 2017

9790-9800

1 reference

Europe PubMed Central

PMC publication ID

16 August 2017

describes a project that uses

1 reference

Europe PubMed Central

11 June 2022

https://www.ebi.ac.uk/europepmc/webservices/rest/PMC3617280/fullTextXML

based on heuristic

inferred from PubMed Central ID database lookup

CB(1) receptor allosteric modulators display both agonist and signaling pathway specificity.

1 reference

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1 reference

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29 September 2017

Allosteric modulator ORG27569 induces CB1 cannabinoid receptor high affinity agonist binding state, receptor internalization, and Gi protein-independent ERK1/2 kinase activation

1 reference

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Crystal structure of the β2 adrenergic receptor-Gs protein complex

1 reference

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1 reference

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1 reference

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Hydrophobic residues in helix 8 of cannabinoid receptor 1 are critical for structural and functional properties

1 reference

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Contrasting effects of allosteric and orthosteric agonists on m1 muscarinic acetylcholine receptor internalization and down-regulation

1 reference

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Allosteric modulators of g protein-coupled receptors: future therapeutics for complex physiological disorders.

1 reference

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Dual role of the second extracellular loop of the cannabinoid receptor 1: ligand binding and receptor localization

1 reference

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Positive allosteric modulation of the human cannabinoid (CB) receptor by RTI-371, a selective inhibitor of the dopamine transporter

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1 reference

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Identification of a putative intracellular allosteric antagonist binding-site in the CXC chemokine receptors 1 and 2.

1 reference

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Hepatocyte growth factor and c-Met promote dendritic maturation during hippocampal neuron differentiation via the Akt pathway

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A unique mechanism of beta-blocker action: carvedilol stimulates beta-arrestin signaling

1 reference

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PSNCBAM-1, a novel allosteric antagonist at cannabinoid CB1 receptors with hypophagic effects in rats

1 reference

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Beta-arrestins and cell signaling

1 reference

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Small-molecule agonists for the glucagon-like peptide 1 receptor

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A guided tour into subcellular colocalization analysis in light microscopy

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mGluR7 undergoes rapid internalization in response to activation by the allosteric agonist AMN082.

1 reference

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Distinct signaling profiles of beta1 and beta2 adrenergic receptor ligands toward adenylyl cyclase and mitogen-activated protein kinase reveals the pluridimensionality of efficacy

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Allosteric agonists of 7TM receptors: expanding the pharmacological toolbox

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Mutations of CB1 T210 produce active and inactive receptor forms: correlations with ligand affinity, receptor stability, and cellular localization

1 reference

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beta-arrestin-dependent, G protein-independent ERK1/2 activation by the beta2 adrenergic receptor

1 reference

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29 September 2017

Allosteric modulation of the cannabinoid CB1 receptor

1 reference

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Functional antagonism of different G protein-coupled receptor kinases for beta-arrestin-mediated angiotensin II receptor signaling

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Different G protein-coupled receptor kinases govern G protein and beta-arrestin-mediated signaling of V2 vasopressin receptor

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Constitutive endocytic cycle of the CB1 cannabinoid receptor.

1 reference

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beta-Arrestin inhibits NF-kappaB activity by means of its interaction with the NF-kappaB inhibitor IkappaBalpha.

1 reference

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Reciprocal regulation of angiotensin receptor-activated extracellular signal-regulated kinases by beta-arrestins 1 and 2.

1 reference

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Desensitization, internalization, and signaling functions of beta-arrestins demonstrated by RNA interference

1 reference

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Activation and targeting of extracellular signal-regulated kinases by beta-arrestin scaffolds

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1 reference

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1 reference

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1 reference

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Constitutive activation of a single effector pathway: evidence for multiple activation states of a G protein-coupled receptor.

1 reference

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Biased signaling pathways in β2-adrenergic receptor characterized by 19F-NMR.

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Signal transduction through MAP kinase cascades

1 reference

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28 June 2018

Allosteric modulation of muscarinic acetylcholine receptors.

1 reference

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Allosteric modulators affect the internalization of human adenosine A1 receptors

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1 reference

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1 reference

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5 September 2018

alpha-Thrombin induces rapid and sustained Akt phosphorylation by beta-arrestin1-dependent and -independent mechanisms, and only the sustained Akt phosphorylation is essential for G1 phase progression

1 reference

https://pubmed.ncbi.nlm.nih.gov/23449980

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Linkage of G protein-coupled receptors to the MAPK signaling pathway through PI 3-kinase gamma

1 reference

https://pubmed.ncbi.nlm.nih.gov/23449980

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Internalization and Recycling of the CB1 Cannabinoid Receptor

1 reference

https://pubmed.ncbi.nlm.nih.gov/23449980

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identifiers

10.1074/JBC.M112.438804

1 reference

Europe PubMed Central

PMC publication ID

16 August 2017

PMC publication ID

1 reference

Europe PubMed Central

PMC publication ID

16 August 2017

PubMed publication ID

1 reference

Europe PubMed Central

PMC publication ID

16 August 2017

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