(Q37590090)

21 August 2017

1 reference

title

Protein methyltransferases as a target class for drug discovery (English)

1 reference

21 August 2017

1 reference

Robert A Copeland

1

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PubMed ID

19721445

21 August 2017

Michael E Solomon

series ordinal

2

1 reference

PubMed ID

19721445

21 August 2017

Victoria M Richon

series ordinal

3

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21 August 2017

1 September 2009

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Nature Reviews Drug Discovery

21 August 2017

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21 August 2017

8

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21 August 2017

724-732

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21 August 2017

9

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https://scigraph.springernature.com/pub.10.1038/nrd2974

21 August 2017

0 references

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31 March 2020

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The polycomb group protein EZH2 is involved in progression of prostate cancer

31 March 2020

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31 March 2020

1 reference

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31 March 2020

1 reference

Involvement of arginine methyltransferase CARM1 in androgen receptor function and prostate cancer cell viability

31 March 2020

1 reference

CARM1 regulates estrogen-stimulated breast cancer growth through up-regulation of E2F1.

31 March 2020

1 reference

PRMT5-mediated methylation of histone H4R3 recruits DNMT3A, coupling histone and DNA methylation in gene silencing.

31 March 2020

1 reference

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31 March 2020

1 reference

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31 March 2020

1 reference

Identification of a specific inhibitor of the histone methyltransferase SU(VAR)3-9.

31 March 2020

1 reference

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31 March 2020

1 reference

Evaluation of enzyme inhibitors in drug discovery. A guide for medicinal chemists and pharmacologists

31 March 2020

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/19721445

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Catalytic roles for carbon-oxygen hydrogen bonding in SET domain lysine methyltransferases

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/19721445

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1038/NRD2974

1 reference

21 August 2017

1 reference

PubMed ID

19721445