(Q37780549)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20716022%20AND%20SRC:MED&resulttype=core&format=json

10 February 2020

review article

1 reference

title

Recent advances in histamine H3 receptor antagonists/inverse agonists (English)

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20716022%20AND%20SRC:MED&resulttype=core&format=json

Katarzyna Kiec-Kononowicz

10 February 2020

author

series ordinal

2

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20716022%20AND%20SRC:MED&resulttype=core&format=json

10 February 2020

author name string

Dorota Łazewska

series ordinal

1

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20716022%20AND%20SRC:MED&resulttype=core&format=json

10 February 2020

language of work or name

English

0 references

publication date

1 September 2010

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20716022%20AND%20SRC:MED&resulttype=core&format=json

Expert Opinion on Therapeutic Patents

10 February 2020

published in

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20716022%20AND%20SRC:MED&resulttype=core&format=json

10 February 2020

volume

20

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20716022%20AND%20SRC:MED&resulttype=core&format=json

10 February 2020

issue

9

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20716022%20AND%20SRC:MED&resulttype=core&format=json

10 February 2020

page(s)

1147-1169

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20716022%20AND%20SRC:MED&resulttype=core&format=json

Auto-inhibition of brain histamine release mediated by a novel class (H3) of histamine receptor

10 February 2020

cites work

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

Histamine H3 receptors modulate the release of [3H]-acetylcholine from slices of rat entorhinal cortex: evidence for the possible existence of H3 receptor subtypes

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

Molecular cloning and characterization of a novel type of histamine receptor preferentially expressed in leukocytes

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

Molecular cloning and characterization of a new human histamine receptor, HH4R

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

Genetic and pharmacological aspects of histamine H3 receptor heterogeneity

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

The histamine H3 receptor: from gene cloning to H3 receptor drugs

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

Histamine H3-receptor isoforms

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

Constitutive activity of the histamine H3 receptor.

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

Protean agonism at histamine H3 receptors in vitro and in vivo

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

Pharmacological classification of histamine H3 receptor agents across species is attributable to transmembrane 3 sequence differences.

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

Medicinal chemical and pharmacological aspects of imidazole-containing histamine H3 receptor antagonists

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

Different antagonist binding properties of human and rat histamine H3 receptors

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

Coordination of histamine H3 receptor antagonists with human adrenal cytochrome P450 enzymes

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

Synthesis of potent non-imidazole histamine H3-receptor antagonists.

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

Histamine H3 receptor antagonists: preclinical promise for treating obesity and cognitive disorders

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

Recent advances in the development of histamine H3 antagonists

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

Histamine H3 receptor antagonists go to clinics

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

Histamine H3 antagonists as wake-promoting and pro-cognitive agents

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

The histamine H3 receptor as a therapeutic drug target for CNS disorders

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

Histamine H3 receptor ligands break ground in a remarkable plethora of therapeutic areas

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

The histamine H3 receptor: an attractive target for the treatment of cognitive disorders

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

Histamine H3 and H4 receptors as novel drug targets.

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

Histamine H3-receptor inverse agonists as novel antipsychotics

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

Histamine H3 antagonists for treatment of cognitive deficits in CNS diseases

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

Measurement of the pharmacokinetics and pharmacodynamics of neuroactive compounds

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

The challenge of drug discovery of a GPCR target: analysis of preclinical pharmacology of histamine H3 antagonists/inverse agonists

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

Histamine H3 receptor antagonists: from target identification to drug leads

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

Selective naphthalene H(3) receptor inverse agonists with reduced potential to induce phospholipidosis and their quinoline analogs.

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

Modulation of the partition coefficient between octanol and buffer at pH 7.4 and pKa to achieve the optimum balance of blood clearance and volume of distribution for a series of tetrahydropyran histamine type 3 receptor antagonists.

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

Minimization of potential hERG liability in histamine H3 receptor antagonists

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

In vitro studies on a class of quinoline containing histamine H3 antagonists

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

A robust and high-capacity [(35)S]GTPgammaS binding assay for determining antagonist and inverse agonist pharmacological parameters of histamine H(3) receptor ligands

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

Characterization of histamine H3-receptors in guinea-pig ileum with H3-selective ligands

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

Acidic elements in histamine H(3) receptor antagonists

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

A novel class of H3 antagonists derived from the natural product guided synthesis of unnatural analogs of the marine bromopyrrole alkaloid dispyrin

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

Total synthesis and biological evaluation of the marine bromopyrrole alkaloid dispyrin: elucidation of discrete molecular targets with therapeutic potential

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

Benzimidazole- and indole-substituted 1,3'-bipyrrolidine benzamides as histamine H3 receptor antagonists

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

Novel substituted pyrrolidines are high affinity histamine H3 receptor antagonists.

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

Aminoalkoxybiphenylnitriles as histamine-3 receptor ligands

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

Synthesis and SAR of aminoalkoxy-biaryl-4-carboxamides: novel and selective histamine H3 receptor antagonists

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

Design of a new histamine H3 receptor antagonist chemotype: (3aR,6aR)-5-alkyl-1-aryl-octahydropyrrolo[3,4-b]pyrroles, synthesis, and structure-activity relationships.

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

Design and evaluation of novel biphenyl sulfonamide derivatives with potent histamine H(3) receptor inverse agonist activity

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

4-acyl-1-(4-aminoalkoxyphenyl)-2-ketopiperazines as a novel class of non-brain-penetrant histamine H3 receptor antagonists

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

5-hydroxyindole-2-carboxylic acid amides: novel histamine-3 receptor inverse agonists for the treatment of obesity.

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

Development of novel 2-[4-(aminoalkoxy)phenyl]-4(3H)-quinazolinone derivatives as potent and selective histamine H3 receptor inverse agonists

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

Synthesis, structure-activity relationships, and biological profiles of a quinazolinone class of histamine H3 receptor inverse agonists

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

Synthesis and evaluation of structurally constrained quinazolinone derivatives as potent and selective histamine H3 receptor inverse agonists

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

A Systematic Review of Modafinil

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

Pharmacological characterization of JNJ-28583867, a histamine H(3) receptor antagonist and serotonin reuptake inhibitor

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

Exploration of structure-activity relationships for dual serotonin transporter reuptake inhibitors-histamine H3 receptor antagonists

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

Lead identification of acetylcholinesterase inhibitors-histamine H3 receptor antagonists from molecular modeling

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

Novel histamine H3 receptor antagonists GSK189254 and GSK334429 are efficacious in surgically-induced and virally-induced rat models of neuropathic pain

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2010.509346

10.1517/13543776.2010.509346

21 January 2018

Identifiers

DOI

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20716022%20AND%20SRC:MED&resulttype=core&format=json

10 February 2020

1 reference