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Substrate and drug binding sites in LeuT.
scientific article published on 16 June 2010
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2925194
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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20739005%20AND%20SRC:MED&resulttype=core&format=json
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11 February 2020
title
Substrate and drug binding sites in LeuT
(English)
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2925194
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11 February 2020
author
Juan Zhen
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3
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11 February 2020
Da-Neng Wang
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6
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11 February 2020
author name string
Ajeeta Nyola
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1
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11 February 2020
Nathan K Karpowich
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2
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11 February 2020
Jennifer Marden
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4
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11 February 2020
Maarten E Reith
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5
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11 February 2020
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English
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publication date
16 June 2010
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11 February 2020
published in
Current Opinion in Structural Biology
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11 February 2020
volume
20
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11 February 2020
issue
4
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11 February 2020
page(s)
415-422
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11 February 2020
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A competitive inhibitor traps LeuT in an open-to-out conformation
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Comparative molecular field analysis using selectivity fields reveals residues in the third transmembrane helix of the serotonin transporter associated with substrate and antagonist recognition
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Identification of a single amino acid, phenylalanine 586, that is responsible for high affinity interactions of tricyclic antidepressants with the human serotonin transporter
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Sibutramine: a novel anti-obesity drug. A review of the pharmacological evidence to differentiate it from d-amphetamine and d-fenfluramine
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Ligand-protein interaction in biomembrane carriers. The induced transition fit of transport catalysis
1 reference
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Identifiers
DOI
10.1016/J.SBI.2010.05.007
1 reference
stated in
Europe PubMed Central
PMC publication ID
2925194
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20739005%20AND%20SRC:MED&resulttype=core&format=json
retrieved
11 February 2020
PMC publication ID
2925194
1 reference
stated in
Europe PubMed Central
PMC publication ID
2925194
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20739005%20AND%20SRC:MED&resulttype=core&format=json
retrieved
11 February 2020
PubMed publication ID
20739005
1 reference
stated in
Europe PubMed Central
PMC publication ID
2925194
reference URL
https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20739005%20AND%20SRC:MED&resulttype=core&format=json
retrieved
11 February 2020
ResearchGate publication ID
45951279
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