(Q38149330)

29 August 2017

title

The therapeutic potential of GPR120: a patent review (English)

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29 August 2017

Somnath Halder

1

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29 August 2017

Sanjay Kumar

series ordinal

2

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29 August 2017

Rajiv Sharma

series ordinal

3

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29 August 2017

language of work or name

English

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publication date

6 October 2013

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Expert Opinion on Therapeutic Patents

29 August 2017

published in

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29 August 2017

volume

23

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29 August 2017

issue

12

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29 August 2017

page(s)

1581-1590

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G-protein-coupled receptors at a glance

29 August 2017

cites work

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2013.842977

The state of GPCR research in 2004.

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2013.842977

The G protein-coupled receptor repertoires of human and mouse

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2013.842977

Targeting GPR120 and other fatty acid-sensing GPCRs ameliorates insulin resistance and inflammatory diseases

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2013.842977

How activated receptors couple to G proteins

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2013.842977

G protein-coupled receptors for energy metabolites as new therapeutic targets

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2013.842977

New frontiers in gut nutrient sensor research: free fatty acid sensing in the gastrointestinal tract.

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2013.842977

Pleiotropic effects of fatty acids on pancreatic beta-cells

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2013.842977

Drug discovery opportunities and challenges at g protein coupled receptors for long chain free Fatty acids

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2013.842977

G protein-coupled receptors for free fatty acids.

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2013.842977

Discovery of TAK-875: A Potent, Selective, and Orally Bioavailable GPR40 Agonist

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2013.842977

AMG 837: a novel GPR40/FFA1 agonist that enhances insulin secretion and lowers glucose levels in rodents

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2013.842977

Identification of a potent and selective free fatty acid receptor 1 (FFA1/GPR40) agonist with favorable physicochemical and in vitro ADME properties.

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2013.842977

Pharmacological regulation of insulin secretion in MIN6 cells through the fatty acid receptor GPR40: identification of agonist and antagonist small molecules

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2013.842977

Free fatty acids regulate gut incretin glucagon-like peptide-1 secretion through GPR120

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2013.842977

Omega-3 and omega-6 PUFAs induce the same GPR120-mediated signalling events, but with different kinetics and intensity in Caco-2 cells.

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2013.842977

GPR120 is an omega-3 fatty acid receptor mediating potent anti-inflammatory and insulin-sensitizing effects

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2013.842977

Dysfunction of lipid sensor GPR120 leads to obesity in both mouse and human

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2013.842977

Discovery of a potent and selective GPR120 agonist.

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2013.842977

Novel selective ligands for free fatty acid receptors GPR120 and GPR40.

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2013.842977

Structure-activity relationships of GPR120 agonists based on a docking simulation.

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2013.842977

FFA1-selective agonistic activity based on docking simulation using FFA1 and GPR120 homology models

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2013.842977

Identification of G protein-coupled receptor 120-selective agonists derived from PPARgamma agonists.

21 January 2018

1 reference

https://api.crossref.org/works/10.1517%2F13543776.2013.842977

10.1517/13543776.2013.842977

21 January 2018

Identifiers

DOI

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29 August 2017

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