(Q39720138)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20358566%20AND%20SRC:MED&resulttype=core&format=json

29 January 2020

title

Antiplasmodial thiostrepton derivatives: proteasome inhibitors with a dual mode of action (English)

1 reference

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29 January 2020

4

1 reference

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29 January 2020

Yousef Najajreh

7

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20358566%20AND%20SRC:MED&resulttype=core&format=json

29 January 2020

2

Gabriele Pradel

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20358566%20AND%20SRC:MED&resulttype=core&format=json

29 January 2020

author name string

Sebastian Schoof

1

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20358566%20AND%20SRC:MED&resulttype=core&format=json

29 January 2020

Makoah N Aminake

3

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20358566%20AND%20SRC:MED&resulttype=core&format=json

29 January 2020

Sascha Baumann

5

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20358566%20AND%20SRC:MED&resulttype=core&format=json

29 January 2020

Marco Potowski

6

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20358566%20AND%20SRC:MED&resulttype=core&format=json

29 January 2020

Marc Kirschner

8

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20358566%20AND%20SRC:MED&resulttype=core&format=json

29 January 2020

Hans-Dieter Arndt

9

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20358566%20AND%20SRC:MED&resulttype=core&format=json

29 January 2020

language of work or name

English

0 references

publication date

1 April 2010

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20358566%20AND%20SRC:MED&resulttype=core&format=json

Angewandte Chemie International Edition

29 January 2020

published in

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20358566%20AND%20SRC:MED&resulttype=core&format=json

29 January 2020

volume

49

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20358566%20AND%20SRC:MED&resulttype=core&format=json

29 January 2020

issue

19

1 reference

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29 January 2020

page(s)

3317-3321

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:20358566%20AND%20SRC:MED&resulttype=core&format=json

New medicines to improve control and contribute to the eradication of malaria

29 January 2020

cites work

1 reference

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21 January 2018

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From amino acids to heteroaromatics--thiopeptide antibiotics, nature's heterocyclic peptides

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21 January 2018

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L11 domain rearrangement upon binding to RNA and thiostrepton studied by NMR spectroscopy

21 January 2018

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Translational regulation via L11: molecular switches on the ribosome turned on and off by thiostrepton and micrococcin

21 January 2018

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Mapping the binding site of thiopeptide antibiotics by proximity-induced covalent capture

21 January 2018

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A fluorescent probe for the 70 S-ribosomal GTPase-associated center

21 January 2018

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Suppressive effect of antibiotic siomycin on antibody production

21 January 2018

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Discovery of a biologically active thiostrepton fragment.

21 January 2018

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Inhibition of mitochondrial protein translation sensitizes melanoma cells to arsenic trioxide cytotoxicity via a reactive oxygen species dependent mechanism.

21 January 2018

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Novel anticancer compounds induce apoptosis in melanoma cells

21 January 2018

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Inhibition of Plasmodium falciparum protein synthesis. Targeting the plastid-like organelle with thiostrepton

21 January 2018

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Effects of interruption of apicoplast function on malaria infection, development, and transmission

21 January 2018

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The apicoplast of Plasmodium falciparum is translationally active.

21 January 2018

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Thiostrepton binds to malarial plastid rRNA.

21 January 2018

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Structure and functions of the 20S and 26S proteasomes

21 January 2018

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The 26S proteasome: a molecular machine designed for controlled proteolysis

21 January 2018

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20S proteasome and its inhibitors: crystallographic knowledge for drug development

21 January 2018

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Catalytic mechanism and assembly of the proteasome.

21 January 2018

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D-cysteine occurrence in thiostrepton may not necessitate an epimerase

21 January 2018

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Fluorescent phallotoxin, a tool for the visualization of cellular actin

21 January 2018

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Creating new fluorescent probes for cell biology.

21 January 2018

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A central strategy for converting natural products into fluorescent probes

21 January 2018

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Splicing factor SF3b as a target of the antitumor natural product pladienolide.

21 January 2018

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Antibiotic susceptibility of mammalian mitochondrial translation

21 January 2018

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Properties of human mitochondrial ribosomes

21 January 2018

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The proteasome inhibitor MLN-273 blocks exoerythrocytic and erythrocytic development of Plasmodium parasites

21 January 2018

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21 January 2018

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21 January 2018

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Epoxomicin, a potent and selective proteasome inhibitor, exhibits in vivo antiinflammatory activity

21 January 2018

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21 January 2018

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21 January 2018

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Selective inhibitors of the osteoblast proteasome stimulate bone formation in vivo and in vitro

21 January 2018

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Proteasome inhibition by fellutamide B induces nerve growth factor synthesis

21 January 2018

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21 January 2018

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21 January 2018

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Lack of proteasome active site allostery as revealed by subunit-specific inhibitors

21 January 2018

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21 January 2018

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FoxM1 is a general target for proteasome inhibitors

21 January 2018

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Plasmodia express two threonine-peptidase complexes during asexual development

21 January 2018

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21 January 2018

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The Structure of Thiostrepton

21 January 2018

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