(Q40461072)

20 September 2017

title

Structure-aided optimization of kinase inhibitors derived from alsterpaullone. (English)

1 reference

20 September 2017

1

Conrad Kunick

0 references

Christoph Schächtele

7

object named as

Christoph Schächtele

0 references

Laurent Meijer

9

object named as

Laurent Meijer

1 reference

20 September 2017

Conrad Kunick

1

1 reference

20 September 2017

Zhihong Zeng

2

1 reference

20 September 2017

Rick Gussio

3

1 reference

20 September 2017

Daniel Zaharevitz

4

1 reference

20 September 2017

Maryse Leost

5

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20 September 2017

Frank Totzke

6

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20 September 2017

Christoph Schächtele

7

1 reference

20 September 2017

Michael H G Kubbutat

8

1 reference

20 September 2017

Thomas Lemcke

10

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20 September 2017

language of work or name

1 reference

1 March 2005

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20 September 2017

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20 September 2017

volume

6

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20 September 2017

issue

3

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20 September 2017

page(s)

541-549

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The protein kinase complement of the human genome

20 September 2017

cites work

1 reference

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21 January 2018

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21 January 2018

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Paullones, a series of cyclin-dependent kinase inhibitors: synthesis, evaluation of CDK1/cyclin B inhibition, and in vitro antitumor activity

21 January 2018

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Paullones are potent inhibitors of glycogen synthase kinase-3beta and cyclin-dependent kinase 5/p25.

21 January 2018

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Intracellular Targets of Paullones. Identification following affinity purification on immobilized inhibitor

21 January 2018

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21 January 2018

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GSK-3: tricks of the trade for a multi-tasking kinase

21 January 2018

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GSK3 takes centre stage more than 20 years after its discovery

21 January 2018

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Structural basis for the synthesis of indirubins as potent and selective inhibitors of glycogen synthase kinase-3 and cyclin-dependent kinases

21 January 2018

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Aloisines, a new family of CDK/GSK-3 inhibitors. SAR study, crystal structure in complex with CDK2, enzyme selectivity, and cellular effects

21 January 2018

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Inhibition of cyclin-dependent kinases, GSK-3beta and CK1 by hymenialdisine, a marine sponge constituent

21 January 2018

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The specificities of protein kinase inhibitors: an update

21 January 2018

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21 January 2018

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Alzheimer's disease. The tangled tale of tau.

21 January 2018

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Role of tau phosphorylation by glycogen synthase kinase-3beta in the regulation of organelle transport

21 January 2018

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GSK-3alpha regulates production of Alzheimer's disease amyloid-beta peptides

21 January 2018

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Evaluation and comparison of 3D-QSAR CoMSIA models for CDK1, CDK5, and GSK-3 inhibition by paullones

21 January 2018

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21 January 2018

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2-Substituted paullones: CDK1/cyclin B-inhibiting property and in vitro antiproliferative activity.

21 January 2018

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Structural characterization of the GSK-3beta active site using selective and non-selective ATP-mimetic inhibitors

21 January 2018

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Baculovirus-mediated expression and characterisation of rat glycogen synthase kinase-3 beta, the mammalian homologue of the Drosophila melanogaster zeste-white 3sgg homeotic gene product

21 January 2018

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Intra-M phase-promoting factor phosphorylation of cyclin B at the prophase/metaphase transition.

21 January 2018

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21 January 2018

Identifiers

DOI

10.1002/CBIC.200400099

1 reference

release_ritequkd25f5zdxawpwagrxlym

20 September 2017

Fatcat ID

1 reference

Fatcat

https://api.fatcat.wiki/v0/release/ritequkd25f5zdxawpwagrxlym

mapped directly with Wikidata item

24 November 2022

based on heuristic

1 reference