(Q42015639)

15 October 2017

title

Synthesis and histamine H(3) and H(4) receptor activity of conformationally restricted cyanoguanidines related to UR-PI376. (English)

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15 October 2017

Roland Geyer

1

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15 October 2017

Armin Buschauer

series ordinal

2

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15 October 2017

publication date

11 October 2011

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Archiv der Pharmazie - Chemistry in Life Sciences

15 October 2017

published in

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15 October 2017

volume

344

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15 October 2017

issue

12

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15 October 2017

page(s)

775-785

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Molecular cloning and characterization of a novel type of histamine receptor preferentially expressed in leukocytes

15 October 2017

cites work

1 reference

https://api.crossref.org/works/10.1002%2FARDP.201100144

Molecular cloning and characterization of a new human histamine receptor, HH4R

21 January 2018

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Structure and expression of the human histamine H4-receptor gene.

21 January 2018

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Murine and human Langerhans cells express a functional histamine H4 receptor: modulation of cell migration and function

21 January 2018

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The role of histamine H4 receptor in immune and inflammatory disorders

21 January 2018

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Histamine h(4) and h(2) receptors control histamine-induced interleukin-16 release from human CD8(+) T cells

21 January 2018

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Histamine H4 receptors modulate dendritic cell migration through skin--immunomodulatory role of histamine

21 January 2018

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The histamine H4 receptor is functionally expressed on T(H)2 cells

21 January 2018

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Histamine H3 and H4 receptors as novel drug targets.

21 January 2018

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Histamine H4 receptor ligands and their potential therapeutic applications

21 January 2018

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Major advances in the development of histamine H4 receptor ligands

21 January 2018

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The histamine H4 receptor mediates inflammation and pruritus in Th2-dependent dermal inflammation

21 January 2018

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Histamine H4 receptor antagonism diminishes existing airway inflammation and dysfunction via modulation of Th2 cytokines

21 January 2018

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Agonist-biased signaling at the histamine H4 receptor: JNJ7777120 recruits β-arrestin without activating G proteins.

21 January 2018

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The first potent and selective non-imidazole human histamine H4 receptor antagonists

21 January 2018

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Does the histamine H4 receptor have a pro- or anti-inflammatory role in murine bronchial asthma?

21 January 2018

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Paradoxical stimulatory effects of the "standard" histamine H4-receptor antagonist JNJ7777120: the H4 receptor joins the club of 7 transmembrane domain receptors exhibiting functional selectivity.

21 January 2018

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Histamine H4 receptor agonists

21 January 2018

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Chiral NG-acylated hetarylpropylguanidine-type histamine H2 receptor agonists do not show significant stereoselectivity

21 January 2018

1 reference

https://api.crossref.org/works/10.1002%2FARDP.201100144

Acylguanidines as bioisosteres of guanidines: NG-acylated imidazolylpropylguanidines, a new class of histamine H2 receptor agonists.

21 January 2018

1 reference

https://api.crossref.org/works/10.1002%2FARDP.201100144

Synthesis and structure-activity relationships of cyanoguanidine-type and structurally related histamine H4 receptor agonists

21 January 2018

1 reference

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N(G)-acylated imidazolylpropylguanidines as potent histamine H4 receptor agonists: selectivity by variation of the N(G)-substituent.

21 January 2018

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Tritium-labeled N(1)-[3-(1H-imidazol-4-yl)propyl]-N(2)-propionylguanidine ([(3)H]UR-PI294), a high-affinity histamine H(3) and H(4) receptor radioligand

21 January 2018

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Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist

21 January 2018

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Discovery of S-(2-guanidylethyl)-isothiourea (VUF 8430) as a potent nonimidazole histamine H4 receptor agonist

21 January 2018

1 reference

https://api.crossref.org/works/10.1002%2FARDP.201100144

A selective human H(4)-receptor agonist: (-)-2-cyano-1-methyl-3-[(2R,5R)-5- [1H-imidazol-4(5)-yl]tetrahydrofuran-2-y] methylguanidine

21 January 2018

1 reference

https://api.crossref.org/works/10.1002%2FARDP.201100144

New high affinity H3 receptor agonists without a basic side chain

21 January 2018

1 reference

https://api.crossref.org/works/10.1002%2FARDP.201100144

2- and 3-substituted 1,4-naphthoquinone derivatives as subversive substrates of trypanothione reductase and lipoamide dehydrogenase from Trypanosoma cruzi: synthesis and correlation between redox cycling activities and in vitro cytotoxicity.

21 January 2018

1 reference

https://api.crossref.org/works/10.1002%2FARDP.201100144

Oxidation of alcohols by “activated” dimethyl sulfoxide. a preparative, steric and mechanistic study

21 January 2018

1 reference

https://api.crossref.org/works/10.1002%2FARDP.201100144

Histamine H3-receptor-mediated [35S]GTP gamma[S] binding: evidence for constitutive activity of the recombinant and native rat and human H3 receptors.

21 January 2018

1 reference

https://api.crossref.org/works/10.1002%2FARDP.201100144

No evidence for functional selectivity of proxyfan at the human histamine H3 receptor coupled to defined Gi/Go protein heterotrimers

21 January 2018

1 reference

https://api.crossref.org/works/10.1002%2FARDP.201100144

High constitutive activity and a G-protein-independent high-affinity state of the human histamine H(4)-receptor.

21 January 2018

1 reference

https://api.crossref.org/works/10.1002%2FARDP.201100144

Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

21 January 2018

1 reference

https://api.crossref.org/works/10.1002%2FARDP.201100144

21 January 2018

Identifiers

DOI

10.1002/ARDP.201100144

1 reference

15 October 2017

1 reference