(Q42020167)

15 October 2017

title

Comparison of the pharmacological properties of human and rat histamine H(3)-receptors (English)

1 reference

15 October 2017

Comparison of the pharmacological properties of human and rat histamine H3-receptors (English)

1 reference

https://api.crossref.org/works/10.1016/J.BCP.2010.07.027

17 June 2024

1 reference

David Schnell

1

1 reference

15 October 2017

Andrea Strasser

2

1 reference

15 October 2017

Roland Seifert

3

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15 October 2017

language of work or name

English

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publication date

3 August 2010

1 reference

full work available at URL

15 October 2017

https://hal.archives-ouvertes.fr/hal-00623303/file/PEER_stage2_10.1016%252Fj.bcp.2010.07.027.pdf

file format

Portable Document Format

online access status

open access

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?resulttype=core&format=json&query=SRC%3AMED%20AND%20EXT_ID%3A20688049

https://api.elsevier.com/content/article/PII:S0006295210005654?httpAccept=text/xml

17 June 2024

1 reference

https://api.crossref.org/works/10.1016/J.BCP.2010.07.027

https://api.elsevier.com/content/article/PII:S0006295210005654?httpAccept=text/plain

17 June 2024

1 reference

https://api.crossref.org/works/10.1016/J.BCP.2010.07.027

17 June 2024

published in

Biochemical Pharmacology

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15 October 2017

volume

80

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15 October 2017

issue

9

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15 October 2017

page(s)

1437-1449

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International Union of Pharmacology. XIII. Classification of histamine receptors

15 October 2017

cites work

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Histamine H3 and H4 receptors as novel drug targets.

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Molecular aspects of the histamine H3 receptor

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Constitutive activity of the histamine H3 receptor.

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High constitutive activity of native H3 receptors regulates histamine neurons in brain.

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The role of transmembrane helix 5 in agonist binding to the human H3 receptor

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Molecular modeling and pharmacological analysis of species-related histamine H(3) receptor heterogeneity

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Distinct pharmacology of rat and human histamine H(3) receptors: role of two amino acids in the third transmembrane domain

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Genetic and pharmacological aspects of histamine H3 receptor heterogeneity

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New G-protein-coupled receptor crystal structures: insights and limitations

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Crystal structure of the human beta2 adrenergic G-protein-coupled receptor

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The 2.6 angstrom crystal structure of a human A2A adenosine receptor bound to an antagonist

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Crystal structure of the ligand-free G-protein-coupled receptor opsin

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Different antagonist binding properties of human and rat histamine H3 receptors

17 June 2024

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Generation of a homology model of the human histamine H3 receptor for ligand docking and pharmacophore-based screening

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Modeling G protein-coupled receptors for structure-based drug discovery using low-frequency normal modes for refinement of homology models: application to H3 antagonists

17 June 2024

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No evidence for functional selectivity of proxyfan at the human histamine H3 receptor coupled to defined Gi/Go protein heterotrimers

17 June 2024

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High-resolution crystal structure of an engineered human beta2-adrenergic G protein-coupled receptor

17 June 2024

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Analysis of the activation mechanism of the guinea-pig Histamine H1-receptor

17 June 2024

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Ligand-specific contribution of the N terminus and E2-loop to pharmacological properties of the histamine H1-receptor

17 June 2024

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Synthesis and structure-activity relationships of cyanoguanidine-type and structurally related histamine H4 receptor agonists

17 June 2024

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Pharmacological profile of histaprodifens at four recombinant histamine H1 receptor species isoforms

17 June 2024

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GROMACS: fast, flexible, and free

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CLUSTAL W: improving the sensitivity of progressive multiple sequence alignment through sequence weighting, position-specific gap penalties and weight matrix choice

17 June 2024

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Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist

17 June 2024

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An 80-amino acid deletion in the third intracellular loop of a naturally occurring human histamine H3 isoform confers pharmacological differences and constitutive activity

17 June 2024

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New histamine H(3)-receptor ligands of the proxifan series: imoproxifan and other selective antagonists with high oral in vivo potency.

17 June 2024

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Multiple switches in G protein-coupled receptor activation

17 June 2024

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Pharmacological classification of histamine H3 receptor agents across species is attributable to transmembrane 3 sequence differences.

17 June 2024

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Quantitative analysis of formyl peptide receptor coupling to g(i)alpha(1), g(i)alpha(2), and g(i)alpha(3).

17 June 2024

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G protein-dependent pharmacology of histamine H3 receptor ligands: evidence for heterogeneous active state receptor conformations

17 June 2024

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https://api.crossref.org/works/10.1016/J.BCP.2010.07.027

High constitutive activity and a G-protein-independent high-affinity state of the human histamine H(4)-receptor.

17 June 2024

39

1 reference

https://api.crossref.org/works/10.1016/J.BCP.2010.07.027

Constitutive activity and ligand selectivity of human, guinea pig, rat, and canine histamine H2 receptors

17 June 2024

40

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Mutations of Cys-17 and Ala-271 in the human histamine H2 receptor determine the species selectivity of guanidine-type agonists and increase constitutive activity

17 June 2024

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Multiple differences in agonist and antagonist pharmacology between human and guinea pig histamine H1-receptor

17 June 2024

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Striking differences of action of lisuride stereoisomers at histamine H1 receptors

17 June 2024

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Molecular basis for the selective interaction of synthetic agonists with the human histamine H1-receptor compared with the guinea pig H1-receptor

17 June 2024

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1 reference

https://api.crossref.org/works/10.1016/J.BCP.2010.07.027

Distinct interaction of human and guinea pig histamine H2-receptor with guanidine-type agonists.

17 June 2024

45

1 reference

https://api.crossref.org/works/10.1016/J.BCP.2010.07.027

Phenylalanine 169 in the second extracellular loop of the human histamine H4 receptor is responsible for the difference in agonist binding between human and mouse H4 receptors

17 June 2024

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17 June 2024

Identifiers

1 reference

15 October 2017

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