(Q42112147)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:25525263%20AND%20SRC:MED&resulttype=core&format=json

25 February 2020

title

New insights on the mechanism of quinoline-based DNA Methyltransferase inhibitors (English)

1 reference

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25 February 2020

13

1 reference

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25 February 2020

Sergio Valente

5

1 reference

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25 February 2020

Frédéric Cantagrel

7

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:25525263%20AND%20SRC:MED&resulttype=core&format=json

25 February 2020

Laurent Lacroix

15

1 reference

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25 February 2020

author name string

Christina Gros

1

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:25525263%20AND%20SRC:MED&resulttype=core&format=json

25 February 2020

Laurence Fleury

2

1 reference

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25 February 2020

Virginie Nahoum

3

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:25525263%20AND%20SRC:MED&resulttype=core&format=json

25 February 2020

Céline Faux

4

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:25525263%20AND%20SRC:MED&resulttype=core&format=json

25 February 2020

Donatella Labella

6

1 reference

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25 February 2020

Elodie Rilova

8

1 reference

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25 February 2020

Mohamed Amine Bouhlel

9

1 reference

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25 February 2020

Marie-Hélène David-Cordonnier

10

1 reference

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25 February 2020

Isabelle Dufau

11

1 reference

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25 February 2020

Frédéric Ausseil

12

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:25525263%20AND%20SRC:MED&resulttype=core&format=json

25 February 2020

Lionel Mourey

14

1 reference

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25 February 2020

Paola B Arimondo

16

1 reference

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25 February 2020

language of work or name

English

0 references

publication date

18 December 2014

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:25525263%20AND%20SRC:MED&resulttype=core&format=json

Journal of Biological Chemistry

25 February 2020

published in

1 reference

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25 February 2020

volume

290

1 reference

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25 February 2020

issue

10

1 reference

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25 February 2020

page(s)

6293-6302

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:25525263%20AND%20SRC:MED&resulttype=core&format=json

Design, synthesis and biological evaluation of 4-amino-N- (4-aminophenyl)benzamide analogues of quinoline-based SGI-1027 as inhibitors of DNA methylation

25 February 2020

cites work

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4358266

Selective non-nucleoside inhibitors of human DNA methyltransferases active in cancer including in cancer stem cells

29 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4358266

Development of a universal radioactive DNA methyltransferase inhibition test for high-throughput screening and mechanistic studies

29 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4358266

Laccaic acid A is a direct, DNA-competitive inhibitor of DNA methyltransferase 1.

29 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4358266

New anticancer active and selective phenylene-bisbenzothiazoles: synthesis, antiproliferative evaluation and DNA binding

29 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4358266

The future of epigenetic therapy in solid tumours--lessons from the past.

29 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4358266

DNA methyltransferase-1 inhibitors as epigenetic therapy for cancer

29 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4358266

DNA methyltransferase inhibitors in cancer: a chemical and therapeutic patent overview and selected clinical studies

29 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4358266

DNA methylation inhibitors in cancer: recent and future approaches

29 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4358266

Towards the chemoinformatic-based identification of DNA methyltransferase inhibitors: 2D- and 3D-similarity profile of screening libraries

29 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4358266

Combination epigenetic therapy has efficacy in patients with refractory advanced non-small cell lung cancer

29 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4358266

Structural insight into maintenance methylation by mouse DNA methyltransferase 1 (Dnmt1)

29 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4358266

The replication focus targeting sequence (RFTS) domain is a DNA-competitive inhibitor of Dnmt1

29 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4358266

Structure and function of mammalian DNA methyltransferases.

29 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4358266

Targeting DNA methylation for epigenetic therapy

29 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4358266

A new class of quinoline-based DNA hypomethylating agents reactivates tumor suppressor genes by blocking DNA methyltransferase 1 activity and inducing its degradation

29 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4358266

Cancer epigenomics: DNA methylomes and histone-modification maps

29 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4358266

Procainamide is a specific inhibitor of DNA methyltransferase 1.

29 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4358266

Analysis of thermal melting curves.

29 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4358266

Mechanistic considerations in high-throughput screening

29 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4358266

Chemical modification of pyrimidine TFOs: effect on i-motif and triple helix formation

29 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4358266

Sequence-specific DNA recognition by polyamides

29 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4358266

Footprinting studies on the effect of echinomycin on the structure of a bent DNA fragment

29 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4358266

Structure-activity relationships for 4-anilinoquinoline derivatives as inhibitors of the DNA methyltransferase enzyme DNMT1.

29 May 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4358266

Clinical outcome of treatment with a combined regimen of decitabine and aclacinomycin/cytarabine for patients with refractory acute myeloid leukemia

17 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4358266

Photochemical electrocyclisation of 3-vinylindoles to pyrido[2,3-a]-, pyrido[4,3-a]- and thieno[2,3-a]-carbazoles: design, synthesis, DNA binding and antitumor cell cytotoxicity

17 August 2018

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=4358266

Kinetic effects due to nonspecific substrate-inhibitor interactions in enzymatic reactions

17 August 2018

1 reference

PubMed

https://pubmed.ncbi.nlm.nih.gov/25525263

inferred from PubMed ID database lookup

12 December 2020

based on heuristic

Identifiers

DOI

10.1074/JBC.M114.594671

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:25525263%20AND%20SRC:MED&resulttype=core&format=json

25 February 2020

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:25525263%20AND%20SRC:MED&resulttype=core&format=json

25 February 2020

1 reference