(Q35863536)

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Design, synthesis and biological evaluation of 4-amino-N- (4-aminophenyl)benzamide analogues of quinoline-based SGI-1027 as inhibitors of DNA methylation

scientific article published in March 2014

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scholarly article

1 reference

Europe PubMed Central

10 August 2017

Design, synthesis and biological evaluation of 4-amino-N- (4-aminophenyl)benzamide analogues of quinoline-based SGI-1027 as inhibitors of DNA methylation (English)

1 reference

Europe PubMed Central

10 August 2017

0 references

DNA methylation

0 references

8

1 reference

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12 June 2020

Arumugam Rajavelu

7

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12 June 2020

Frédéric Cantagrel

17

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12 June 2020

Alexandre Erdmann

2

object named as

Alexandre Erdmann

1 reference

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12 June 2020

Philippe Schambel

13

object named as

Philippe Schambel

1 reference

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12 June 2020

Paola B Arimondo

16

object named as

Paola B Arimondo

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12 June 2020

author name string

Elodie Rilova

1

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12 June 2020

Christina Gros

3

1 reference

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12 June 2020

Véronique Masson

4

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12 June 2020

Yannick Aussagues

5

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12 June 2020

Valérie Poughon-Cassabois

6

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12 June 2020

Yoann Menon

9

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12 June 2020

Natacha Novosad

10

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12 June 2020

Jean-Marc Gregoire

11

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12 June 2020

Stéphane Vispé

12

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12 June 2020

Fréderic Ausseil

14

1 reference

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12 June 2020

François Sautel

15

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12 June 2020

publication date

1 March 2014

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10 August 2017

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12 June 2020

9

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12 June 2020

3

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12 June 2020

590-601

1 reference

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12 June 2020

Development of a universal radioactive DNA methyltransferase inhibition test for high-throughput screening and mechanistic studies

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DNA methyltransferase inhibitors in cancer: a chemical and therapeutic patent overview and selected clinical studies

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11 July 2018

Molecular modeling and virtual screening of DNA methyltransferase inhibitors

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11 July 2018

DNA methylation inhibitors in cancer: recent and future approaches

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Cancer epigenetics: from mechanism to therapy

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11 July 2018

Towards the chemoinformatic-based identification of DNA methyltransferase inhibitors: 2D- and 3D-similarity profile of screening libraries

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11 July 2018

Inhibitors of DNA methyltransferases: insights from computational studies

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11 July 2018

Mechanisms of DNA methylation and demethylation in mammals

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11 July 2018

Molecular modeling of inhibitors of human DNA methyltransferase with a crystal structure: discovery of a novel DNMT1 inhibitor

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Combination epigenetic therapy has efficacy in patients with refractory advanced non-small cell lung cancer

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11 July 2018

Structure-Based Mechanistic Insights into DNMT1-Mediated Maintenance DNA Methylation

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11 July 2018

Epigenetic drug discovery: targeting DNA methyltransferases

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11 July 2018

A decade of exploring the cancer epigenome - biological and translational implications

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11 July 2018

C5-DNA methyltransferase inhibitors: from screening to effects on zebrafish embryo development.

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11 July 2018

Structural insight into maintenance methylation by mouse DNA methyltransferase 1 (Dnmt1)

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11 July 2018

Advances in the computational development of DNA methyltransferase inhibitors

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Structure and function of mammalian DNA methyltransferases.

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11 July 2018

Structure of DNMT1-DNA Complex Reveals a Role for Autoinhibition in Maintenance DNA Methylation

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11 July 2018

DNA methylation predicts survival and response to therapy in patients with myelodysplastic syndromes

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11 July 2018

Epigenetics in cancer

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11 July 2018

A new class of quinoline-based DNA hypomethylating agents reactivates tumor suppressor genes by blocking DNA methyltransferase 1 activity and inducing its degradation

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11 July 2018

An operational definition of epigenetics

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11 July 2018

DNA methylation landscapes: provocative insights from epigenomics

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11 July 2018

Epigenetics in cancer

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11 July 2018

Mammalian DNA methyltransferases: a structural perspective

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11 July 2018

Structure of Dnmt3a bound to Dnmt3L suggests a model for de novo DNA methylation

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11 July 2018

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11 July 2018

Procainamide is a specific inhibitor of DNA methyltransferase 1.

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11 July 2018

Natural products as DNA methyltransferase inhibitors: a computer-aided discovery approach

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21 January 2018

Docking of a novel DNA methyltransferase inhibitor identified from high-throughput screening: insights to unveil inhibitors in chemical databases

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21 January 2018

Molecular modeling studies of the novel inhibitors of DNA methyltransferases SGI-1027 and CBC12: implications for the mechanism of inhibition of DNMTs

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21 January 2018

The role of Arg165 towards base flipping, base stabilization and catalysis in M.HhaI.

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21 January 2018

The use of formamidine protection for the derivatization of aminobenzoic acids

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21 January 2018

Structure-activity relationships for 4-anilinoquinoline derivatives as inhibitors of the DNA methyltransferase enzyme DNMT1.

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21 January 2018

Potential antitumor agents. 13. Bisquaternary salts

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12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Homology modeling, docking and structure-based pharmacophore of inhibitors of DNA methyltransferase

1 reference

https://pubmed.ncbi.nlm.nih.gov/24678024

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identifiers

10.1002/CMDC.201300420

1 reference

Europe PubMed Central

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:24678024%20AND%20SRC:MED&resulttype=core&format=json

12 June 2020

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12 June 2020

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12 June 2020

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