(Q43263223)

English

A different molecular interaction of bradykinin and the synthetic agonist FR190997 with the human B2 receptor: evidence from mutational analysis

scientific article published on 26 August 2003

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scholarly article

1 reference

Europe PubMed Central

PMC publication ID

17 November 2017

A different molecular interaction of bradykinin and the synthetic agonist FR190997 with the human B2 receptor: evidence from mutational analysis (English)

1 reference

Europe PubMed Central

PMC publication ID

17 November 2017

molecular interaction

1 reference

based on heuristic

inferred from title

2

1 reference

Europe PubMed Central

PMC publication ID

17 November 2017

author name string

Francesca Bellucci

1

1 reference

Europe PubMed Central

PMC publication ID

17 November 2017

Paola Cucchi

3

1 reference

Europe PubMed Central

PMC publication ID

17 November 2017

Claudio Catalani

4

1 reference

Europe PubMed Central

PMC publication ID

17 November 2017

Wolfgang Reichert

5

1 reference

Europe PubMed Central

PMC publication ID

17 November 2017

Sabrina Zappitelli

6

1 reference

Europe PubMed Central

PMC publication ID

17 November 2017

Luigi Rotondaro

7

1 reference

Europe PubMed Central

PMC publication ID

17 November 2017

Laura Quartara

8

1 reference

Europe PubMed Central

PMC publication ID

17 November 2017

Alessandro Giolitti

9

1 reference

Europe PubMed Central

PMC publication ID

17 November 2017

Carlo Alberto Maggi

10

1 reference

Europe PubMed Central

PMC publication ID

17 November 2017

language of work or name

0 references

publication date

26 August 2003

1 reference

Europe PubMed Central

PMC publication ID

17 November 2017

British Journal of Pharmacology

1 reference

Europe PubMed Central

PMC publication ID

17 November 2017

140

1 reference

Europe PubMed Central

PMC publication ID

17 November 2017

3

1 reference

Europe PubMed Central

PMC publication ID

17 November 2017

500-506

1 reference

Europe PubMed Central

PMC publication ID

17 November 2017

The therapeutic potential of bradykinin B2 receptor agonists in the treatment of cardiovascular disease

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1574048

25 May 2018

Bradykinin inhibits development of myocardial infarction through B2 receptor signalling by increment of regional blood flow around the ischaemic lesions in rats

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1574048

25 May 2018

The ligand paradox between affinity and efficacy: can you be there and not make a difference?

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1574048

25 May 2018

Role of bradykinin in preconditioning and protection of the ischaemic myocardium

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1574048

25 May 2018

Receptor activation: what does the rhodopsin structure tell us?

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1574048

25 May 2018

Determination of bradykinin B2 receptor in vivo phosphorylation sites and their role in receptor function

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1574048

25 May 2018

Proinflammatory characteristics of a nonpeptide bradykinin mimic, FR190997, in vivo

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1574048

25 May 2018

The development of the bradykinin agonist labradimil as a means to increase the permeability of the blood-brain barrier: from concept to clinical evaluation

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1574048

25 May 2018

Differences in electromechanical coupling between bradykinin and the nonpeptide kinin B2 receptor agonist, FR 190997, in the circular muscle of guinea-pig colon.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1574048

25 May 2018

Peptide and non-peptide bradykinin B2 receptor agonists and antagonists: a reappraisal of their pharmacology in the guinea-pig ileum

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1574048

25 May 2018

Uncovering molecular mechanisms involved in activation of G protein-coupled receptors

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1574048

25 May 2018

Nonpeptide antagonists for kinin receptors.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1574048

25 May 2018

Binding, gating, affinity and efficacy: the interpretation of structure-activity relationships for agonists and of the effects of mutating receptors

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1574048

25 May 2018

Mutations within the cholecystokinin-B/gastrin receptor ligand 'pocket' interconvert the functions of nonpeptide agonists and antagonists.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1574048

25 May 2018

Cloning, sequencing and functional expression of a guinea pig lung bradykinin B2 receptor

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1574048

25 May 2018

Nonpeptide mimic of bradykinin with long-acting properties at the bradykinin B2 receptor

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1574048

25 May 2018

Mutations in the B2 bradykinin receptor reveal a different pattern of contacts for peptidic agonists and peptidic antagonists

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1574048

25 May 2018

Expression cloning of a human B1 bradykinin receptor

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1574048

25 May 2018

Pharmacology of bradykinin and related kinins.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1574048

25 May 2018

Bradykinin receptors: pharmacological properties and biological roles

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1574048

25 May 2018

Molecular cloning, functional expression and pharmacological characterization of a human bradykinin B2 receptor gene

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1574048

25 May 2018

Cloning and pharmacological characterization of a human bradykinin (BK-2) receptor

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1574048

25 May 2018

A rapid and sensitive method for the quantitation of microgram quantities of protein utilizing the principle of protein-dye binding

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1574048

25 May 2018

Characterization of non-peptide bradykinin B2 receptor agonist (FR 190997) and antagonist (FR 173657).

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1574048

25 May 2018

Preliminary mutational analysis of the human kinin B2 receptor for nonpeptide antagonist ligands recognition

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1574048

15 August 2018

Control of conformational equilibria in the human B2 bradykinin receptor. Modeling of nonpeptidic ligand action and comparison to the rhodopsin structure.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1574048

15 August 2018

Two active molecular phenotypes of the tachykinin NK1 receptor revealed by G-protein fusions and mutagenesis.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1574048

15 August 2018

Controlled modulation of BBB permeability using the bradykinin agonist, RMP-7.

1 reference

https://eutils.ncbi.nlm.nih.gov/entrez/eutils/elink.fcgi?dbfrom=pmc&linkname=pmc_refs_pubmed&retmode=json&id=1574048

15 August 2018

FR190997, a novel bradykinin B2 agonist, expresses longer action than bradykinin in paw edema formation and hypotensive response

1 reference

https://pubmed.ncbi.nlm.nih.gov/12970081

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Mouse paw edema induced by a novel bradykinin agonist and its inhibition by B2-antagonists

1 reference

https://pubmed.ncbi.nlm.nih.gov/12970081

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Can peptides be mimicked?

1 reference

https://pubmed.ncbi.nlm.nih.gov/12970081

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Anion secretory effects of a non-peptide mimic of bradykinin (FR190997) on mouse colon epithelium

1 reference

https://pubmed.ncbi.nlm.nih.gov/12970081

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

A molecular model of agonist and nonpeptide antagonist binding to the human V(1) vascular vasopressin receptor

1 reference

https://pubmed.ncbi.nlm.nih.gov/12970081

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Dual agonistic and antagonistic property of nonpeptide angiotensin AT1 ligands: susceptibility to receptor mutations

1 reference

https://pubmed.ncbi.nlm.nih.gov/12970081

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Pharmacological characterisation of the first non-peptide bradykinin B2 receptor agonist FR 190997: an in vitro study on human, rabbit and pig vascular B2 receptors

1 reference

https://pubmed.ncbi.nlm.nih.gov/12970081

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

CCK-B/Gastrin receptor transmembrane domain mutations selectively alter synthetic agonist efficacy without affecting the activity of endogenous peptides

1 reference

https://pubmed.ncbi.nlm.nih.gov/12970081

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identifiers

10.1038/SJ.BJP.0705454

1 reference

Europe PubMed Central

PMC publication ID

17 November 2017

PMC publication ID

1 reference

Europe PubMed Central

PMC publication ID

17 November 2017

PubMed publication ID

1 reference

Europe PubMed Central

PMC publication ID

17 November 2017

ResearchGate publication ID

0 references

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