(Q44784411)

English

Structure-activity studies on the corticotropin releasing factor antagonist astressin, leading to a minimal sequence necessary for antagonistic activity

scientific article published in March 2004

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scholarly article

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Europe PubMed Central

PubMed publication ID

6 December 2017

Structure-activity studies on the corticotropin releasing factor antagonist astressin, leading to a minimal sequence necessary for antagonistic activity (English)

1 reference

Europe PubMed Central

PubMed publication ID

6 December 2017

Rob M.J. Liskamp

6

object named as

Rob M J Liskamp

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Europe PubMed Central

PubMed publication ID

6 December 2017

author name string

Dirk T S Rijkers

1

1 reference

Europe PubMed Central

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6 December 2017

John A W Kruijtzer

2

1 reference

Europe PubMed Central

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6 December 2017

Marja van Oostenbrugge

3

1 reference

Europe PubMed Central

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6 December 2017

Eric Ronken

4

1 reference

Europe PubMed Central

PubMed publication ID

6 December 2017

Jack A J den Hartog

5

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Europe PubMed Central

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6 December 2017

language of work or name

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publication date

1 March 2004

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Europe PubMed Central

PubMed publication ID

6 December 2017

1 reference

Europe PubMed Central

PubMed publication ID

6 December 2017

5

1 reference

Europe PubMed Central

PubMed publication ID

6 December 2017

3

1 reference

Europe PubMed Central

PubMed publication ID

6 December 2017

340-348

1 reference

Europe PubMed Central

PubMed publication ID

6 December 2017

Corticotropin releasing hormone: therapeutic implications and medicinal chemistry developments.

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Characterization of a 41-Residue Ovine Hypothalamic Peptide That Stimulates Secretion of Corticotropin and β-Endorphin

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Characterization of rat hypothalamic corticotropin-releasing factor

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Persistent elevations of cerebrospinal fluid concentrations of corticotropin-releasing factor in adult nonhuman primates exposed to early-life stressors: implications for the pathophysiology of mood and anxiety disorders

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Alanine series of ovine corticotropin releasing factor (oCRF): a structure-activity relationship study

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Identification of a seven transmembrane helix receptor for corticotropin-releasing factor and sauvagine in mammalian brain.

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Cloning and functional expression of a rat brain corticotropin releasing factor (CRF) receptor

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Cloning and characterization of a functionally distinct corticotropin-releasing factor receptor subtype from rat brain.

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A sauvagine/corticotropin-releasing factor receptor expressed in heart and skeletal muscle

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Identification of a second corticotropin-releasing factor receptor gene and characterization of a cDNA expressed in heart

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Identification of a novel murine receptor for corticotropin-releasing hormone expressed in the heart

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CP-154,526: a potent and selective nonpeptide antagonist of corticotropin releasing factor receptors.

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Synthesis and oral efficacy of a 4-(butylethylamino)pyrrolo[2,3-d]pyrimidine: a centrally active corticotropin-releasing factor1 receptor antagonist.

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Rapid microscale synthesis, a new method for lead optimization using robotics and solution phase chemistry: application to the synthesis and optimization of corticotropin-releasing factor1 receptor antagonists

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Design and synthesis of a series of non-peptide high-affinity human corticotropin-releasing factor1 receptor antagonists

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Pyrazolo[1,5-a]pyrimidine CRF-1 receptor antagonists.

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Synthesis and biological activity of oxo-7H-benzo[e]perimidine-4-carboxylic acid derivatives as potent, nonpeptide corticotropin releasing factor (CRF) receptor antagonists

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Thiazolo[4,5-d]pyrimidine thiones and -ones as corticotropin-releasing hormone (CRH-R1) receptor antagonists

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Non-peptide corticotropin-releasing hormone antagonists: syntheses and structure-activity relationships of 2-anilinopyrimidines and -triazines

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Synthesis, corticotropin-releasing factor receptor binding affinity, and pharmacokinetic properties of triazolo-, imidazo-, and pyrrolopyrimidines and -pyridines

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The discovery of 4-(3-pentylamino)-2,7-dimethyl-8-(2-methyl-4-methoxyphenyl)-pyrazolo-[1 ,5-a]-pyrimidine: a corticotropin-releasing factor (hCRF1) antagonist

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Synthesis and structure-affinity relationships of 4-(5-Aryl-1,2,3,6-tetrahydropyridino)pyrimidine derivatives as corticotropin-releasing factor(1) receptor antagonists.

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Chemical modification of aryl-1,2,3,6-tetrahydropyridinopyrimidine derivative to discover corticotropin-releasing factor(1) receptor antagonists: aryl-1,2,3,6-tetrahydropyridino-purine, -3H-1,2,3-triazolo[4,5-d)pyrimidine, -purin-8-one, and -7H-pyrr

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CRHR1 Receptor binding and lipophilicity of pyrrolopyrimidines, potential nonpeptide corticotropin-releasing hormone type 1 receptor antagonists

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Imidazo[4,5-b]pyridines as corticotropin releasing factor receptor ligands

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Pharmacophore development for corticotropin-releasing hormone: new insights into inhibitor activity.

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Compounds that activate the mouse melanocortin-1 receptor identified by screening a small molecule library based upon the beta-turn

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An optimized solid phase synthesis strategy--including on-resin lactamization--of astressin, its retro-, inverso-, and retro-inverso isomers as corticotropin releasing factor antagonists

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Ligand requirements of the human corticotropin-releasing factor-binding protein

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Identifiers

10.1002/CBIC.200300769

1 reference

Europe PubMed Central

PubMed publication ID

6 December 2017

PubMed publication ID

1 reference

Europe PubMed Central

PubMed publication ID

6 December 2017

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