(Q46871307)

26 December 2017

title

Peptidic macrocyclization via palladium-catalyzed chemoselective indole C-2 arylation (English)

1 reference

26 December 2017

author name string

Huijun Dong

1

1 reference

26 December 2017

Chris Limberakis

2

1 reference

26 December 2017

Spiros Liras

3

1 reference

26 December 2017

David Price

4

1 reference

26 December 2017

Keith James

5

1 reference

26 December 2017

language of work or name

English

0 references

publication date

1 December 2012

1 reference

26 December 2017

published in

Chemical Communications

1 reference

26 December 2017

volume

48

1 reference

26 December 2017

issue

95

1 reference

26 December 2017

page(s)

11644-11646

1 reference

26 December 2017

Protein-protein interactions: principles, techniques, and their potential role in new drug development

cites work

1 reference

https://api.crossref.org/works/10.1039%2FC2CC36962A

Synthesis of chemically modified bioactive peptides: recent advances, challenges and developments for medicinal chemistry.

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC2CC36962A

Eleven amino acid glucagon-like peptide-1 receptor agonists with antidiabetic activity

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC2CC36962A

Emerging approaches in the molecular design of receptor-selective peptide ligands: conformational, topographical and dynamic considerations

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC2CC36962A

Constrained peptides: models of bioactive peptides and protein substructures

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC2CC36962A

Solid-phase synthesis of cyclic homodetic peptides

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC2CC36962A

Converting a peptide into a drug: strategies to improve stability and bioavailability

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC2CC36962A

New Structural Insights into the Inhibition of Serine Proteases by Cyclic Peptides from Bacteria

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC2CC36962A

Histone Deacetylase Inhibitors

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC2CC36962A

Chemistry and biology of cyclic depsipeptides of medicinal and biological interest

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC2CC36962A

Proteases universally recognize beta strands in their active sites

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC2CC36962A

Round and round we go: cyclic peptides in disease

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC2CC36962A

Effect of structural and conformation modifications, including backbone cyclization, of hydrophilic hexapeptides on their intestinal permeability and enzymatic stability

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC2CC36962A

Quantitative comparison of the relative cell permeability of cyclic and linear peptides.

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC2CC36962A

Peptoid macrocycles: making the rounds with peptidomimetic oligomers

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC2CC36962A

The exploration of macrocycles for drug discovery--an underexploited structural class

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC2CC36962A

Macrocycles are great cycles: applications, opportunities, and challenges of synthetic macrocycles in drug discovery

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC2CC36962A

Contemporary strategies for peptide macrocyclization

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC2CC36962A

Single turn peptide alpha helices with exceptional stability in water

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC2CC36962A

Biaryl-bridged macrocyclic peptides: conformational constraint via carbogenic fusion of natural amino acid side chains

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC2CC36962A

Total synthesis of chloropeptin II (complestatin) and chloropeptin I.

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC2CC36962A

Sigma-chelation-directed C-H functionalizations using Pd(II) and Cu(II) catalysts: regioselectivity, stereoselectivity and catalytic turnover

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC2CC36962A

Aryl-aryl bond formation by transition-metal-catalyzed direct arylation.

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC2CC36962A

Transition-metal-catalyzed direct arylation of (hetero)arenes by C-H bond cleavage.

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC2CC36962A

Palladium- and copper-catalyzed arylation of carbon-hydrogen bonds

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC2CC36962A

Recent advances in aryl-aryl bond formation by direct arylation.

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC2CC36962A

Intermolecular oxidative cross-coupling of arenes

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC2CC36962A

Direct C-H transformation via iron catalysis

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC2CC36962A

Towards mild metal-catalyzed C-H bond activation

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC2CC36962A

Palladium-Catalyzed Ligand-Directed C−H Functionalization Reactions

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC2CC36962A

Direct transition metal-catalyzed functionalization of heteroaromatic compounds

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC2CC36962A

Direct palladium-catalyzed C-2 and C-3 arylation of indoles: a mechanistic rationale for regioselectivity

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC2CC36962A

Room temperature and phosphine free palladium catalyzed direct C-2 arylation of indoles.

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC2CC36962A

Increasing rates of reaction: microwave-assisted organic synthesis for combinatorial chemistry

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC2CC36962A

CuI-Catalyzed Azideâ Alkyne Intramoleculari-to-(i+4) Side-Chain-to-Side-Chain Cyclization Promotes the Formation of Helix-Like Secondary Structures

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC2CC36962A

Room Temperature Palladium-Catalyzed 2-Arylation of Indoles

21 January 2018

1 reference

https://api.crossref.org/works/10.1039%2FC2CC36962A

21 January 2018

Identifiers

DOI

10.1039/C2CC36962A

1 reference

26 December 2017

1 reference

26 December 2017