(Q58200853)

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:17530729%20AND%20SRC:MED&resulttype=core&format=json

31 December 2019

title

Synthesis and evaluation of 3-phenylpyrazolo[3,4-d]pyrimidine-peptide conjugates as Src kinase inhibitors (English)

1 reference

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31 December 2019

0 references

1

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31 December 2019

author name string

Yuehao Wang

2

1 reference

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31 December 2019

Xiaofeng Lin

3

1 reference

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31 December 2019

Gongqin Sun

4

1 reference

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31 December 2019

Keykavous Parang

5

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31 December 2019

publication date

1 September 2007

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31 December 2019

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31 December 2019

volume

2

1 reference

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31 December 2019

issue

9

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31 December 2019

page(s)

1346-1360

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https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:17530729%20AND%20SRC:MED&resulttype=core&format=json

The catalytic activity of the Src family kinases is required to disrupt cadherin-dependent cell-cell contacts

31 December 2019

cites work

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700074

Protein tyrosine kinase structure and function

21 January 2018

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700074

7 January 2021

Src Family Kinases: Potential Targets for the Treatment of Human Cancer and Leukemia

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700074

7 January 2021

Cellular functions regulated by Src family kinases

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700074

7 January 2021

c-Src, receptor tyrosine kinases, and human cancer

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700074

7 January 2021

A renaissance for SRC

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700074

7 January 2021

The hunting of the Src

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700074

7 January 2021

Selected glimpses into the activation and function of Src kinase

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700074

7 January 2021

Src inhibitors: genomics to therapeutics

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700074

7 January 2021

Targeted disruption of the c-src proto-oncogene leads to osteopetrosis in mice

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700074

7 January 2021

Role of Src expression and activation in human cancer

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700074

7 January 2021

Activation of c-Src by receptor tyrosine kinases in human colon cancer cells with high metastatic potential

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700074

7 January 2021

Selective requirement for Src kinases during VEGF-induced angiogenesis and vascular permeability

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700074

7 January 2021

Src deficiency or blockade of Src activity in mice provides cerebral protection following stroke

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700074

7 January 2021

Crystal structure of Hck in complex with a Src family-selective tyrosine kinase inhibitor

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700074

7 January 2021

Crystal structure of the Src family tyrosine kinase Hck

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700074

7 January 2021

Three protein kinase structures define a common motif

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700074

7 January 2021

Designing bisubstrate analog inhibitors for protein kinases

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700074

7 January 2021

Chemical mechanism of the adenosine cyclic 3',5'-monophosphate dependent protein kinase from pH studies

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700074

7 January 2021

Multiple modes of ligand recognition: crystal structures of cyclin-dependent protein kinase 2 in complex with ATP and two inhibitors, olomoucine and isopentenyladenine

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700074

7 January 2021

Structural analysis of the lymphocyte-specific kinase Lck in complex with non-selective and Src family selective kinase inhibitors

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700074

7 January 2021

New pyrazolo[3,4-d]pyrimidines endowed with A431 antiproliferative activity and inhibitory properties of Src phosphorylation.

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700074

7 January 2021

Use of synthetic peptides and copolymers to study the substrate specificity and inhibition of the protein tyrosine kinase pp60c-src

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700074

7 January 2021

Development and characterization of potent and specific peptide inhibitors of p60c-src protein tyrosine kinase using pseudosubstrate-based inhibitor design approach

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700074

7 January 2021

Identification and characterization of a novel synthetic peptide substrate specific for Src-family protein tyrosine kinases.

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700074

7 January 2021

Catalytic specificity of protein-tyrosine kinases is critical for selective signalling

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700074

7 January 2021

Identification of GIYWHHY as a novel peptide substrate for human p60c-src protein tyrosine kinase

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700074

7 January 2021

The Src-selective kinase inhibitor PP1 also inhibits Kit and Bcr-Abl tyrosine kinases

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700074

7 January 2021

Bone-targeted Src kinase inhibitors: novel pyrrolo- and pyrazolopyrimidine analogues

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700074

7 January 2021

Discovery of a novel, potent, and Src family-selective tyrosine kinase inhibitor. Study of Lck- and FynT-dependent T cell activation

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700074

7 January 2021

The specificities of protein kinase inhibitors: an update

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700074

7 January 2021

Discovery of a novel series of potent and selective substrate-based inhibitors of p60c-src protein tyrosine kinase: conformational and topographical constraints in peptide design

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700074

7 January 2021

Synthesis and structure-activity relationships of linear and conformationally constrained peptide analogues of CIYKYY as Src tyrosine kinase inhibitors

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700074

7 January 2021

Mechanism-based design of a protein kinase inhibitor

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700074

7 January 2021

ATP-phosphopeptide conjugates as inhibitors of Src tyrosine kinases

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700074

7 January 2021

Pyrazolo[3,4-d]pyrimidines containing an extended 3-substituent as potent inhibitors of Lck -- a selectivity insight

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700074

7 January 2021

Design of tetrapeptide ligands as inhibitors of the Src SH2 domain

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700074

7 January 2021

Conformationally constrained peptide analogues of pTyr-Glu-Glu-Ile as inhibitors of the Src SH2 domain binding

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700074

7 January 2021

Docking interactions in the mitogen-activated protein kinase cascades

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700074

7 January 2021

Molecular determinants for Csk-catalyzed tyrosine phosphorylation of the Src tail

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700074

7 January 2021

Determination of the substrate-docking site of protein tyrosine kinase C-terminal Src kinase

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700074

7 January 2021

Docking-based substrate recognition by the catalytic domain of a protein tyrosine kinase, C-terminal Src kinase (Csk).

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700074

7 January 2021

Design of allele-specific inhibitors to probe protein kinase signaling

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700074

7 January 2021

Engineering unnatural nucleotide specificity for Rous sarcoma virus tyrosine kinase to uniquely label its direct substrates

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700074

7 January 2021

A molecular gate which controls unnatural ATP analogue recognition by the tyrosine kinase v-Src

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700074

7 January 2021

Engineering Src family protein kinases with unnatural nucleotide specificity

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700074

7 January 2021

Crystal structures of c-Src reveal features of its autoinhibitory mechanism

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700074

7 January 2021

Peptide chips for the quantitative evaluation of protein kinase activity

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700074

7 January 2021

The pp60c-Src inhibitor PP1 is non-competitive against ATP.

1 reference

https://api.crossref.org/works/10.1002%2FCMDC.200700074

7 January 2021

Identifiers

DOI

10.1002/CMDC.200700074

1 reference

https://www.ebi.ac.uk/europepmc/webservices/rest/search?query=EXT_ID:17530729%20AND%20SRC:MED&resulttype=core&format=json

31 December 2019

1 reference