(Q64944773)

1 July 2019

title

Discovery of New Sulfonamide Carbonic Anhydrase IX Inhibitors Incorporating Nitrogenous Bases. (English)

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1 July 2019

author

Silvia Bua

2

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1 July 2019

Gianluca Bartolucci

6

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1 July 2019

Paola Gratteri

10

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1 July 2019

Carla Ghelardini

9

object named as

Carla Ghelardini

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1 July 2019

Claudiu T Supuran

11

object named as

Claudiu T Supuran

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1 July 2019

author name string

Alessio Nocentini

1

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1 July 2019

Carrie L Lomelino

3

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1 July 2019

Robert McKenna

4

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1 July 2019

Marta Menicatti

5

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1 July 2019

Barbara Tenci

7

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1 July 2019

Lorenzo Di Cesare Mannelli

8

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1 July 2019

publication date

21 November 2017

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1 July 2019

ACS Medicinal Chemistry Letters

published in

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1 July 2019

volume

8

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issue

12

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1 July 2019

page(s)

1314-1319

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1 July 2019

The carbon dioxide hydration activity of carbonic anhydrase. I. Stop-flow kinetic studies on the native human isoenzymes B and C

cites work

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12 December 2020

Synthesis and antitumor activities of novel pyrimidine derivatives of 2,3-O,O-dibenzyl-6-deoxy-L-ascorbic acid and 4,5-didehydro-5,6- dideoxy-L-ascorbic acid

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The purines: potent and versatile small molecule inhibitors and modulators of key biological targets

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Carbonic anhydrases: novel therapeutic applications for inhibitors and activators

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Enzymology of purine and pyrimidine antimetabolites used in the treatment of cancer

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Carbonic anhydrase IX: Biochemical and crystallographic characterization of a novel antitumor target

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12 December 2020

Ureido-substituted benzenesulfonamides potently inhibit carbonic anhydrase IX and show antimetastatic activity in a model of breast cancer metastasis.

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12 December 2020

Interfering with pH regulation in tumours as a therapeutic strategy

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12 December 2020

Structure-based drug discovery of carbonic anhydrase inhibitors

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12 December 2020

Multiple binding modes of inhibitors to carbonic anhydrases: how to design specific drugs targeting 15 different isoforms?

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12 December 2020

Promise and challenges in drug discovery and development of hybrid anticancer drugs

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12 December 2020

Anticancer carbonic anhydrase inhibitors: a patent review (2008 - 2013).

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12 December 2020

Combining the tail and the ring approaches for obtaining potent and isoform-selective carbonic anhydrase inhibitors: solution and X-ray crystallographic studies

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12 December 2020

Rational approaches, design strategies, structure activity relationship and mechanistic insights for anticancer hybrids.

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12 December 2020

Hypoxia-induced carbonic anhydrase IX as a target for cancer therapy: from biology to clinical use.

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12 December 2020

In search of uracil derivatives as bioactive agents. Uracils and fused uracils: Synthesis, biological activity and applications.

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12 December 2020

Synthesis and pharmacophore modelling of 2,6,9-trisubstituted purine derivatives and their potential role as apoptosis-inducing agents in cancer cell lines

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12 December 2020

Click-tailed coumarins with potent and selective inhibitory action against the tumor-associated carbonic anhydrases IX and XII

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12 December 2020

How many carbonic anhydrase inhibition mechanisms exist?

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12 December 2020

Advances in structure-based drug discovery of carbonic anhydrase inhibitors

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12 December 2020

Benzenesulfonamides Incorporating Flexible Triazole Moieties Are Highly Effective Carbonic Anhydrase Inhibitors: Synthesis and Kinetic, Crystallographic, Computational, and Intraocular Pressure Lowering Investigations

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12 December 2020

Synthesis of isoxazole-containing sulfonamides with potent carbonic anhydrase II and VII inhibitory properties

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12 December 2020

Carbonic Anhydrase Inhibition and the Management of Hypoxic Tumors

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12 December 2020

10.1021/ACSMEDCHEMLETT.7B00399

Identifiers

DOI

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1 July 2019

PMC publication ID

5733260

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1 July 2019

PubMed publication ID

29259754

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1 July 2019