(Q27657268)

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Binding and Inactivation Mechanism of a Humanized Fatty Acid Amide Hydrolase by α-Ketoheterocycle Inhibitors Revealed from Cocrystal Structures

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scholarly article

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Binding and Inactivation Mechanism of a Humanized Fatty Acid Amide Hydrolase by α-Ketoheterocycle Inhibitors Revealed from Cocrystal Structures (English)

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crystal structure

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1 reference

based on heuristic

inferred from title

1 reference

based on heuristic

inferred from title

Benjamin Cravatt

4

object named as

Benjamin F Cravatt

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author name string

Mauro Mileni

1

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Joie Garfunkle

2

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Jessica K DeMartino

3

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Dale L Boger

5

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Raymond C Stevens

6

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language of work or name

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publication date

5 August 2009

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Journal of the American Chemical Society

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131

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10497-506

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30

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Discovery and Characterization of a Highly Selective FAAH Inhibitor that Reduces Inflammatory Pain

1 reference

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Structure-guided inhibitor design for human FAAH by interspecies active site conversion

1 reference

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Structural adaptations in a membrane enzyme that terminates endocannabinoid signaling

1 reference

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1 reference

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1 reference

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1 reference

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1 reference

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1 reference

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1 reference

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1 reference

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1 reference

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1 reference

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1 reference

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1 reference

https://pubmed.ncbi.nlm.nih.gov/19722626

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

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1 reference

https://pubmed.ncbi.nlm.nih.gov/19722626

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based on heuristic

inferred from PubMed ID database lookup

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1 reference

https://pubmed.ncbi.nlm.nih.gov/19722626

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based on heuristic

inferred from PubMed ID database lookup

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https://pubmed.ncbi.nlm.nih.gov/19722626

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1 reference

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Identifiers

10.1021/JA902694N

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release_o3dkvwakmvff7fwukwgtjk4ghy

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