(Q34313778)

English

Synthesis and structure-activity relationship studies of N-benzyl-2-phenylpyrimidin-4-amine derivatives as potent USP1/UAF1 deubiquitinase inhibitors with anticancer activity against nonsmall cell lung cancer

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scholarly article

1 reference

Europe PubMed Central

1 August 2017

Synthesis and structure-activity relationship studies of N-benzyl-2-phenylpyrimidin-4-amine derivatives as potent USP1/UAF1 deubiquitinase inhibitors with anticancer activity against nonsmall cell lung cancer (English)

1 reference

Europe PubMed Central

1 August 2017

object named as

Ajit Jadhav

10

0 references

9

object named as

Anton Simeonov

1 reference

Europe PubMed Central

1 August 2017

author name string

Thomas S Dexheimer

1

1 reference

Europe PubMed Central

1 August 2017

Andrew S Rosenthal

2

1 reference

Europe PubMed Central

1 August 2017

Diane K Luci

3

1 reference

Europe PubMed Central

1 August 2017

Qin Liang

4

1 reference

Europe PubMed Central

1 August 2017

Mark A Villamil

5

1 reference

Europe PubMed Central

1 August 2017

Junjun Chen

6

1 reference

Europe PubMed Central

1 August 2017

Hongmao Sun

7

1 reference

Europe PubMed Central

1 August 2017

Edward H Kerns

8

1 reference

Europe PubMed Central

1 August 2017

Zhihao Zhuang

11

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Europe PubMed Central

1 August 2017

David J Maloney

12

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Europe PubMed Central

1 August 2017

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publication date

17 September 2014

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Europe PubMed Central

1 August 2017

Journal of Medicinal Chemistry

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Europe PubMed Central

1 August 2017

57

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Europe PubMed Central

1 August 2017

19

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Europe PubMed Central

1 August 2017

8099-8110

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Europe PubMed Central

1 August 2017

describes a project that uses

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Europe PubMed Central

11 June 2022

https://www.ebi.ac.uk/europepmc/webservices/rest/PMC4191588/fullTextXML

based on heuristic

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A selective USP1-UAF1 inhibitor links deubiquitination to DNA damage responses.

1 reference

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1 reference

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1 reference

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1 reference

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1 reference

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1 reference

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1 reference

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The ubiquitin code

1 reference

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1 reference

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Selective and cell-active inhibitors of the USP1/ UAF1 deubiquitinase complex reverse cisplatin resistance in non-small cell lung cancer cells

1 reference

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USP1 deubiquitinates ID proteins to preserve a mesenchymal stem cell program in osteosarcoma

1 reference

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6 July 2018

The USP1/UAF1 complex promotes double-strand break repair through homologous recombination

1 reference

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The STAT5 inhibitor pimozide decreases survival of chronic myelogenous leukemia cells resistant to kinase inhibitors

1 reference

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1 reference

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Will the ubiquitin system furnish as many drug targets as protein kinases?

1 reference

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1 reference

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1 reference

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1 reference

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1 reference

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1 reference

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1 reference

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A UAF1-containing multisubunit protein complex regulates the Fanconi anemia pathway

1 reference

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1 reference

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Proteasome-independent functions of ubiquitin in endocytosis and signaling

1 reference

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1 reference

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1 reference

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1 reference

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1 reference

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1 reference

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1 reference

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1 reference

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based on heuristic

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Identification of chemokine receptor CCR4 antagonist

1 reference

https://pubmed.ncbi.nlm.nih.gov/25229643

12 December 2020

based on heuristic

inferred from PubMed ID database lookup

Identifiers

10.1021/JM5010495

1 reference

Europe PubMed Central

1 August 2017

release_3j2vxzispfgwbghe4beytfaq2q

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https://api.fatcat.wiki/v0/release/3j2vxzispfgwbghe4beytfaq2q

24 November 2022

based on heuristic

mapped directly with Wikidata item

1 reference

Europe PubMed Central

1 August 2017

1 reference

Europe PubMed Central

1 August 2017

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